BE904724A - Derives de piperazine 1,4-disubstitues, composition pharmaceutique les contenant; leur procede d'obtention. - Google Patents
Derives de piperazine 1,4-disubstitues, composition pharmaceutique les contenant; leur procede d'obtention.Info
- Publication number
- BE904724A BE904724A BE0/216623A BE216623A BE904724A BE 904724 A BE904724 A BE 904724A BE 0/216623 A BE0/216623 A BE 0/216623A BE 216623 A BE216623 A BE 216623A BE 904724 A BE904724 A BE 904724A
- Authority
- BE
- Belgium
- Prior art keywords
- obtaining
- pharmaceutical composition
- composition containing
- piperazine derivatives
- disubstituted piperazine
- Prior art date
Links
- -1 1,4-DISUBSTITUTED PIPERAZINE Chemical class 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 229940066771 systemic antihistamines piperazine derivative Drugs 0.000 title abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
- 125000001118 alkylidene group Chemical group 0.000 abstract 1
- 125000002618 bicyclic heterocycle group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- DBDCNCCRPKTRSD-UHFFFAOYSA-N thieno[3,2-b]pyridine Chemical class C1=CC=C2SC=CC2=N1 DBDCNCCRPKTRSD-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US73120185A | 1985-05-06 | 1985-05-06 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE904724A true BE904724A (fr) | 1986-11-05 |
Family
ID=24938510
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE0/216623A BE904724A (fr) | 1985-05-06 | 1986-05-05 | Derives de piperazine 1,4-disubstitues, composition pharmaceutique les contenant; leur procede d'obtention. |
Country Status (25)
Country | Link |
---|---|
JP (1) | JPH0753728B2 (xx) |
KR (1) | KR940000829B1 (xx) |
CN (1) | CN1017901B (xx) |
AT (1) | AT398572B (xx) |
AU (1) | AU593244B2 (xx) |
BE (1) | BE904724A (xx) |
CA (1) | CA1278792C (xx) |
CH (1) | CH672787A5 (xx) |
DE (1) | DE3615180C2 (xx) |
DK (1) | DK165745C (xx) |
EG (1) | EG18206A (xx) |
ES (6) | ES8801250A1 (xx) |
FI (1) | FI85484C (xx) |
FR (1) | FR2581385B1 (xx) |
GB (1) | GB2174703B (xx) |
GR (1) | GR861149B (xx) |
HU (1) | HU195509B (xx) |
IE (1) | IE59201B1 (xx) |
IT (1) | IT1208607B (xx) |
LU (1) | LU86421A1 (xx) |
MY (1) | MY100777A (xx) |
NL (1) | NL8601146A (xx) |
PT (1) | PT82523B (xx) |
SE (1) | SE465270B (xx) |
ZA (1) | ZA862046B (xx) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5801186A (en) * | 1987-11-20 | 1998-09-01 | Hoechst Marion Roussel, Inc. | 3- 4-(1-substituted-4-piperazinyl)butyl!-4-thiazolidinone and related compounds |
US4880930A (en) * | 1987-11-30 | 1989-11-14 | New James S | Psychotropic acyclic amide derivatives |
US4780466A (en) * | 1988-03-17 | 1988-10-25 | Hoechst-Roussel Pharmaceuticals, Inc. | Arylpiperazinylalkoxy derivatives of cyclic imides |
IE903410A1 (en) * | 1989-10-09 | 1991-04-10 | Novo Nordisk As | Indole derivatives, their preparation and use |
US5272148A (en) * | 1992-09-09 | 1993-12-21 | Hoechst-Roussel Pharmaceuticals Incorporated | Heteroarenylpiperazines |
FR2738823B1 (fr) * | 1995-09-15 | 1997-10-31 | Synthelabo | Derives de 3-(omega-(4-(thieno(3,2-c)pyridin-4-yl)piperazin- 1-yl)alkyl)-3,4-dihydroquinolein-2(1h)-one,leur preparation et leur application en therapeutique |
FR2738822B1 (fr) * | 1995-09-15 | 1997-10-31 | Synthelabo | Derives de 4-(omega-(4-(thieno(3,2-c)pyridin-4-yl)piperazin- 1-yl)alkyl)quinolein-2(1h)-one, leur preparation et leur application en therapeutique |
FR2738824B1 (fr) * | 1995-09-15 | 1997-10-31 | Synthelabo | Derives de 3-(omega(4-(thieno(3,2-c)pyridin-4-yl)piperazin-1 -yl)alkyl)-3,4-dihydroquinazolin-2(1h)-one,leur preparation et leur application en therapeutique |
SI0850235T1 (en) * | 1995-09-15 | 2000-04-30 | Sanofi-Synthelabo | Quinolein-2(1h)-one derivatives as serotonin antagonists |
FR2761071B1 (fr) * | 1997-03-20 | 1999-12-03 | Synthelabo | Derives de quinolein-2(1h)-one et de dihydroquinolein-2(1h)- one, leur preparation et leur application en therapeutique |
FR2797874B1 (fr) * | 1999-08-27 | 2002-03-29 | Adir | Nouveaux derives de la pyridine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
US20040077605A1 (en) | 2001-06-20 | 2004-04-22 | Salvati Mark E. | Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4367335A (en) * | 1981-08-03 | 1983-01-04 | Mead Johnson & Company | Thiazolidinylalkylene piperazine derivatives |
US4452799A (en) * | 1981-12-23 | 1984-06-05 | Mead Johnson & Company | Benzisothiazole and benzisoxazole piperazine derivatives |
US4361565A (en) * | 1981-12-28 | 1982-11-30 | Mead Johnson & Company | 2-[4-[(4,4-Dialkyl-2,6-piperidinedion-1-yl)butyl]-1-piperazinyl]pyridines |
-
1986
- 1986-03-11 CA CA000503794A patent/CA1278792C/en not_active Expired - Fee Related
- 1986-03-19 ZA ZA862046A patent/ZA862046B/xx unknown
- 1986-04-29 AU AU56795/86A patent/AU593244B2/en not_active Expired
- 1986-04-29 EG EG250/86A patent/EG18206A/xx active
- 1986-04-29 GR GR861149A patent/GR861149B/el unknown
- 1986-04-30 FI FI861820A patent/FI85484C/fi not_active IP Right Cessation
- 1986-05-02 KR KR1019860003445A patent/KR940000829B1/ko not_active Expired - Fee Related
- 1986-05-02 GB GB08610810A patent/GB2174703B/en not_active Expired
- 1986-05-05 BE BE0/216623A patent/BE904724A/fr not_active IP Right Cessation
- 1986-05-05 FR FR8606471A patent/FR2581385B1/fr not_active Expired - Lifetime
- 1986-05-05 IE IE119386A patent/IE59201B1/en not_active IP Right Cessation
- 1986-05-05 NL NL8601146A patent/NL8601146A/nl active Search and Examination
- 1986-05-05 CN CN86103071A patent/CN1017901B/zh not_active Expired
- 1986-05-05 DE DE3615180A patent/DE3615180C2/de not_active Expired - Lifetime
- 1986-05-05 ES ES554659A patent/ES8801250A1/es not_active Expired
- 1986-05-05 DK DK207186A patent/DK165745C/da not_active IP Right Cessation
- 1986-05-05 LU LU86421A patent/LU86421A1/fr unknown
- 1986-05-05 SE SE8602061A patent/SE465270B/sv not_active IP Right Cessation
- 1986-05-05 CH CH1830/86A patent/CH672787A5/de not_active IP Right Cessation
- 1986-05-06 HU HU861860A patent/HU195509B/hu unknown
- 1986-05-06 JP JP61103726A patent/JPH0753728B2/ja not_active Expired - Lifetime
- 1986-05-06 IT IT8620313A patent/IT1208607B/it active
- 1986-05-06 PT PT82523A patent/PT82523B/pt unknown
- 1986-05-06 AT AT0121486A patent/AT398572B/de not_active IP Right Cessation
-
1987
- 1987-09-25 ES ES557757A patent/ES8802149A1/es not_active Expired
- 1987-10-01 MY MYPI87002712A patent/MY100777A/en unknown
-
1988
- 1988-01-28 ES ES557809A patent/ES8802614A1/es not_active Expired
- 1988-05-26 ES ES557839A patent/ES8900138A1/es not_active Expired
- 1988-11-16 ES ES557855A patent/ES8900253A1/es not_active Expired
-
1989
- 1989-02-27 ES ES557865A patent/ES9000005A1/es not_active Expired
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
FR2430412A1 (fr) | Derives substitues de propanolamine utiles comme medicaments et procede de leur preparation | |
ES2044836T3 (es) | Derivado de la piperidina, su utilizacion y compuesto farmaceutico que lo contiene. | |
BE904724A (fr) | Derives de piperazine 1,4-disubstitues, composition pharmaceutique les contenant; leur procede d'obtention. | |
FR2371437A1 (fr) | Nouveaux derives de pipepidine ou de morpholine utiles comme medicaments et comme fongicides | |
PT91121A (pt) | Processo para a preparacao de derivados da quinolina e de composicoes farmaceuticas que os contem | |
FR2453133A1 (fr) | Nouveaux acides acetohydroxamiques, leur procede de preparation et leur application en therapeutique | |
DE3574702D1 (de) | Antitumor-platin-komplexe. | |
FR2374307A1 (fr) | Derives de la 1,4-dihydropyridine, leur procede d'obtention et composition pharmaceutique les contenant | |
FR2357556A1 (fr) | Procede de transformation de cis-hexahydrodibenzo(b,d) pyran-9-ones en trans-hexahydrodibenzo(b,d) pyran-9-ones | |
FR2375187A1 (fr) | Cyclopentane-1-amines, procede pour leur preparation et produits contenant ces composes | |
FR2403989A1 (fr) | Nouveaux derives a-halogenomethyles d'amines utiles comme medicaments et procedes de leur preparation | |
DK165109C (da) | 4-anilino-cyklopentaoedaapyrimidinderivater samt farmaceutiske midler indeholdende saadanne | |
HU906360D0 (en) | Process for producing quinoline derivatives and pharmaceutical preparatives containing such compounds | |
FR2372818A1 (fr) | Acide 5-(hydroxy (substitue) methyl)-2,3-dihydrobenzofuran-2-carboxylique et ses derives utiles comme medicaments | |
FR2363559A1 (fr) | Nouveaux derives de perhydro-aza-heterocycles utiles comme medicaments et procede pour leur preparation | |
FR2403330A1 (fr) | Nouveaux derives de benzoyl-2-chloro-4-glycinanilides substitues, leur procede de preparation et leur application en tant que medicaments | |
FR2369287A1 (fr) | Procede de preparation de derives organiques d'etain d'esters mercaptoalcooliques | |
DK183789A (da) | 2-alkyl-3-benzoylbenzofuraner og laegemidler indeholdende disse | |
FR2358415A1 (fr) | Derives peptidiques, leur preparation et leur application en tant que medicaments | |
ES8706148A1 (es) | Un procedimiento para preparar nuevos derivados de carbapenem. | |
FI870090A0 (fi) | Laongkedjade alkylresorcinolfosfiter. | |
FR2371460A1 (fr) | Procede de preparation de kanamycine c et de ses derives desoxy | |
FR2453162A1 (fr) | Procede pour la preparation de derives de 4-acetoxy-azetidine-2-one par condensation avec un b-thiocetoester et composes obtenus | |
BE905654A (fr) | Derives de la armstrong 2-1,2,4-triazoline-5-one, procede pour leur preparation et leurs utilisations. | |
BE904588A (fr) | (-)-1Beta-ETHYL-1ALPHA-HYDROXYMETHYL-1,2,3,4,6,7,12,12beta alpha-OCTAHYDROINDOLO (2,3-a) QUINOLIZINE, PROCEDE POUR LA PREPARER ET COMPOSITIONS PHARMACEUTIQUES CONTENANT CELLE-CI. |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE20 | Patent expired |
Owner name: *BRISTOL-MYERS CY Effective date: 20060505 |