BE872023A - 4-AMINO-2-PIPERIDINOQUINAZOLINE DERIVATIVES, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM - Google Patents
4-AMINO-2-PIPERIDINOQUINAZOLINE DERIVATIVES, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITION CONTAINING THEMInfo
- Publication number
- BE872023A BE872023A BE191743A BE191743A BE872023A BE 872023 A BE872023 A BE 872023A BE 191743 A BE191743 A BE 191743A BE 191743 A BE191743 A BE 191743A BE 872023 A BE872023 A BE 872023A
- Authority
- BE
- Belgium
- Prior art keywords
- piperidinoquinazoline
- derivatives
- amino
- pharmaceutical composition
- composition containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Heart & Thoracic Surgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Cardiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB4758377 | 1977-11-16 | ||
GB7844533A GB2010824B (en) | 1977-11-16 | 1978-11-15 | Therapeutic agents |
Publications (1)
Publication Number | Publication Date |
---|---|
BE872023A true BE872023A (en) | 1979-05-14 |
Family
ID=26266083
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE191743A BE872023A (en) | 1977-11-16 | 1978-11-14 | 4-AMINO-2-PIPERIDINOQUINAZOLINE DERIVATIVES, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM |
Country Status (12)
Country | Link |
---|---|
JP (1) | JPS5481282A (en) |
AT (1) | AT365183B (en) |
AU (1) | AU509348B2 (en) |
BE (1) | BE872023A (en) |
CA (1) | CA1088068A (en) |
CH (1) | CH637131A5 (en) |
DE (1) | DE2849392A1 (en) |
FR (1) | FR2409267A1 (en) |
GB (1) | GB2010824B (en) |
LU (1) | LU80531A1 (en) |
NL (1) | NL174646C (en) |
SE (1) | SE7811770L (en) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IE800178L (en) * | 1979-01-31 | 1980-07-31 | Pfizer Ltd | Derivatives of 4-amino-2-piperidinoquinazoline |
FR2514353A2 (en) * | 1980-04-28 | 1983-04-15 | Synthelabo | Antidepressant 4-benzyloxy-piperidine derivs. - prepd. by react-ng piperidine deriv. with benzyl deriv. |
FR2481278A1 (en) * | 1980-04-28 | 1981-10-30 | Synthelabo | Antidepressant 4:benzyloxy piperidine(s) - are prepd. from 4:hydroxy piperidine and benzyl halide |
JPS62212385A (en) * | 1986-03-13 | 1987-09-18 | Kotobuki Seiyaku Kk | Quinazoline derivative and hypotensive agent and production thereof |
-
1978
- 1978-10-24 CA CA314,082A patent/CA1088068A/en not_active Expired
- 1978-11-14 DE DE19782849392 patent/DE2849392A1/en not_active Withdrawn
- 1978-11-14 SE SE7811770A patent/SE7811770L/en unknown
- 1978-11-14 BE BE191743A patent/BE872023A/en not_active IP Right Cessation
- 1978-11-14 NL NLAANVRAGE7811236,A patent/NL174646C/en not_active IP Right Cessation
- 1978-11-14 AU AU41576/78A patent/AU509348B2/en not_active Expired
- 1978-11-15 FR FR7832235A patent/FR2409267A1/en active Granted
- 1978-11-15 AT AT0816678A patent/AT365183B/en active
- 1978-11-15 CH CH1175578A patent/CH637131A5/en not_active IP Right Cessation
- 1978-11-15 GB GB7844533A patent/GB2010824B/en not_active Expired
- 1978-11-15 LU LU80531A patent/LU80531A1/en unknown
- 1978-11-15 JP JP14094678A patent/JPS5481282A/en active Granted
Also Published As
Publication number | Publication date |
---|---|
LU80531A1 (en) | 1980-06-05 |
NL174646B (en) | 1984-02-16 |
AU4157678A (en) | 1979-05-24 |
NL7811236A (en) | 1979-05-18 |
CH637131A5 (en) | 1983-07-15 |
GB2010824B (en) | 1982-06-16 |
FR2409267B1 (en) | 1981-02-27 |
JPS5623991B2 (en) | 1981-06-03 |
ATA816678A (en) | 1981-05-15 |
NL174646C (en) | 1984-07-16 |
AT365183B (en) | 1981-12-28 |
FR2409267A1 (en) | 1979-06-15 |
JPS5481282A (en) | 1979-06-28 |
SE7811770L (en) | 1979-05-17 |
CA1088068A (en) | 1980-10-21 |
GB2010824A (en) | 1979-07-04 |
AU509348B2 (en) | 1980-05-08 |
DE2849392A1 (en) | 1979-05-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: PFIZER CORP. Effective date: 19841114 |