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BE852641A - Derives de benzimidazole-2-carbamate substitues sur le noyau benzenique en 5(6) - Google Patents

Derives de benzimidazole-2-carbamate substitues sur le noyau benzenique en 5(6)

Info

Publication number
BE852641A
BE852641A BE175923A BE175923A BE852641A BE 852641 A BE852641 A BE 852641A BE 175923 A BE175923 A BE 175923A BE 175923 A BE175923 A BE 175923A BE 852641 A BE852641 A BE 852641A
Authority
BE
Belgium
Prior art keywords
benzimidazole
benzene nucleus
derivatives substituted
carbamate derivatives
carbamate
Prior art date
Application number
BE175923A
Other languages
English (en)
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of BE852641A publication Critical patent/BE852641A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30Nitrogen atoms not forming part of a nitro radical
    • C07D235/32Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C335/00Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C335/30Isothioureas
    • C07C335/38Isothioureas containing any of the groups, X being a hetero atom, Y being any atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE175923A 1976-03-19 1977-03-18 Derives de benzimidazole-2-carbamate substitues sur le noyau benzenique en 5(6) BE852641A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US66877876A 1976-03-19 1976-03-19

Publications (1)

Publication Number Publication Date
BE852641A true BE852641A (fr) 1977-09-19

Family

ID=24683698

Family Applications (1)

Application Number Title Priority Date Filing Date
BE175923A BE852641A (fr) 1976-03-19 1977-03-18 Derives de benzimidazole-2-carbamate substitues sur le noyau benzenique en 5(6)

Country Status (4)

Country Link
US (1) US4139626A (fr)
BE (1) BE852641A (fr)
HU (1) HU176329B (fr)
ZA (1) ZA771591B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4297365A (en) * 1978-08-04 1981-10-27 Ciba-Geigy Corporation Benzimidazoles and pharmaceutical preparations containing such compounds
US4386097A (en) * 1978-08-04 1983-05-31 Ciba-Geigy Corporation Benzimidazoles, processes for their preparation and pharmaceutical preparations containing such compounds
US4312873A (en) * 1978-09-29 1982-01-26 Syntex (U.S.A.) Inc. 5(6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity
CN1612733A (zh) 2001-11-09 2005-05-04 贝林格尔·英格海姆药物公司 用作蛋白激酶抑制剂的苯并咪唑类
CA2494942A1 (fr) * 2002-08-08 2004-02-19 Boehringer Ingelheim Pharmaceuticals, Inc. Composes benzimidazole substitues
WO2005079791A1 (fr) * 2004-02-12 2005-09-01 Boehringer Ingelheim Pharmaceuticals, Inc. Derives d'acide thiophene-2-carboxylique (1h-benzimidazol-2 yl)-amide et composes associes utilises comme inhibiteurs de la tec kinase itk (kinase des lymphocites inductibles par l'interleukine -2) pour traiter une inflammation et des troubles immunologiques et allergiques

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1032171A (fr) * 1972-12-29 1978-05-30 Colin C. Beard Noyau benzene 5-6 substitue par des derives benzimidazole -2- carbamate a action authelonintique
US3935209A (en) * 1973-03-12 1976-01-27 Syntex (U.S.A.) Inc. 5(6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity
US4026936A (en) * 1975-08-07 1977-05-31 Hoffmann-La Roche Inc. Anthelmintic pyridine and thiazole substituted benzimidazole carbamates

Also Published As

Publication number Publication date
US4139626A (en) 1979-02-13
HU176329B (en) 1981-01-28
ZA771591B (en) 1978-10-25

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