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BE759493A - Nouvelles 2-(5-nitro-2-furyl)-thieno(3,2-d) pyrimidines et procedes pour les fabriquer - Google Patents

Nouvelles 2-(5-nitro-2-furyl)-thieno(3,2-d) pyrimidines et procedes pour les fabriquer

Info

Publication number
BE759493A
BE759493A BE759493DA BE759493A BE 759493 A BE759493 A BE 759493A BE 759493D A BE759493D A BE 759493DA BE 759493 A BE759493 A BE 759493A
Authority
BE
Belgium
Prior art keywords
thieno
pyrimidines
furyl
news
nitro
Prior art date
Application number
Other languages
English (en)
French (fr)
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Publication date
Priority claimed from DE19691959403 external-priority patent/DE1959403A1/de
Priority claimed from DE19702050816 external-priority patent/DE2050816A1/de
Priority claimed from DE19702050815 external-priority patent/DE2050815A1/de
Priority claimed from DE19702050814 external-priority patent/DE2050814A1/de
Publication of BE759493A publication Critical patent/BE759493A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
BE759493D 1969-11-26 Nouvelles 2-(5-nitro-2-furyl)-thieno(3,2-d) pyrimidines et procedes pour les fabriquer BE759493A (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE19691959403 DE1959403A1 (de) 1969-11-26 1969-11-26 Neue 2-(5-Nitro-2-furyl)-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
DE19702050816 DE2050816A1 (de) 1970-10-16 1970-10-16 Neue 2-(Nitro-2-furyl>thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine
DE19702050815 DE2050815A1 (de) 1970-10-16 1970-10-16 Neue 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidine
DE19702050814 DE2050814A1 (de) 1970-10-16 1970-10-16 Neue Verfahren zur Herstellung von 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 3,2-d eckige Klammer zu pyrimidinen

Publications (1)

Publication Number Publication Date
BE759493A true BE759493A (fr) 1971-05-25

Family

ID=27430978

Family Applications (1)

Application Number Title Priority Date Filing Date
BE759493D BE759493A (fr) 1969-11-26 Nouvelles 2-(5-nitro-2-furyl)-thieno(3,2-d) pyrimidines et procedes pour les fabriquer

Country Status (13)

Country Link
US (1) US3661908A (de)
BE (1) BE759493A (de)
BG (2) BG17799A3 (de)
CA (1) CA926865A (de)
CH (3) CH568324A5 (de)
DK (1) DK128781B (de)
FR (1) FR2073416B1 (de)
GB (1) GB1321316A (de)
IE (1) IE34765B1 (de)
IL (1) IL35729A (de)
NL (1) NL7017210A (de)
NO (1) NO129954B (de)
SE (1) SE377938B (de)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3932642A (en) * 1971-04-10 1976-01-13 Boehringer Ingelheim Gmbh Biocidal compositions containing a 2- (5'-nitro-2'-furyl)-thieno(2,3-d) pyrimidine and methods of use
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
US6608053B2 (en) * 2000-04-27 2003-08-19 Yamanouchi Pharmaceutical Co., Ltd. Fused heteroaryl derivatives
US20040138238A1 (en) * 2002-08-08 2004-07-15 Dhanoa Dale S. Substituted aminopyrimidine compounds as neurokinin antagonists
GB0423653D0 (en) * 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds
EP2041139B1 (de) 2006-04-26 2011-11-09 F. Hoffmann-La Roche AG Pharmazeutische verbindungen
WO2007127183A1 (en) * 2006-04-26 2007-11-08 Genentech, Inc. Phosphoinositide 3-kinase inhibitor compounds and pharmaceutical compositions containing them
JP5148597B2 (ja) 2006-04-26 2013-02-20 エフ.ホフマン−ラ ロシュ アーゲー 医薬化合物
BRPI0717923A2 (pt) * 2006-12-07 2013-10-22 Genentech In '' composto, composição farmacêutica, método para tratar um câncer, processo para a produção de uma composição farmacêutica, usos, métodos para inibir ou modular a atividade da lipídeo quinase e kit ' '
AR064154A1 (es) * 2006-12-07 2009-03-18 Piramed Ltd Compuestos inhibidores de fodfoinostida 3- quinasas y composiciones farmaceuticas
ATE510841T1 (de) * 2007-06-12 2011-06-15 Hoffmann La Roche Thiazoliopyrimidine und ihre verwendung als hemmer der phosphatidylinositol-3 kinase
EP2207781B1 (de) * 2007-09-24 2012-11-28 Genentech, Inc. Thiazolopyrimidinverbindungen als p13k-inhibitoren und anwendungsverfahren
CA2701292C (en) * 2007-10-25 2015-03-24 Genentech, Inc. Process for making thienopyrimidine compounds
GB0721095D0 (en) * 2007-10-26 2007-12-05 Piramed Ltd Pharmaceutical compounds
JP5709766B2 (ja) 2009-03-12 2015-04-30 ジェネンテック, インコーポレイテッド 造血器腫瘍の治療のためのホスホイノシチド3キナーゼ阻害剤化合物と化学療法剤の併用
EP2451811A1 (de) * 2009-05-27 2012-05-16 F. Hoffmann-La Roche AG Für p110 delta selektive bicyclische indol-pyrimidin-pi3k-hemmerverbindungen und anwendungsverfahren
KR20130026364A (ko) 2009-05-27 2013-03-13 제넨테크, 인크. P110 델타에 대해 선택적인 비시클릭 피리미딘 pi3k 억제제 화합물 및 사용 방법
MA33974B1 (fr) * 2009-10-12 2013-02-01 Hoffmann La Roche Combinaisons d'un inhibiteur de pi3k et d'un inhibiteur de mek
WO2011130654A1 (en) 2010-04-16 2011-10-20 Genentech, Inc. Fox03a as predictive biomarker for pi3k/akt kinase pathway inhibitor efficacy
WO2012088254A1 (en) 2010-12-22 2012-06-28 Genentech, Inc. Autophagy inducer and inhibitor combination therapy for the treatment of neoplasms
JP6669500B2 (ja) 2013-02-25 2020-03-18 ジェネンテック, インコーポレイテッド 薬物耐性akt変異体を検出し治療するための方法及び組成物

Also Published As

Publication number Publication date
IL35729A0 (en) 1971-01-28
CH567029A5 (de) 1975-09-30
IE34765L (en) 1971-05-26
CA926865A (en) 1973-05-22
DK128781B (da) 1974-07-01
US3661908A (en) 1972-05-09
CH568324A5 (de) 1975-10-31
FR2073416B1 (de) 1975-04-18
GB1321316A (en) 1973-06-27
BG17800A3 (bg) 1973-12-25
CH559210A5 (de) 1975-02-28
IL35729A (en) 1974-01-14
FR2073416A1 (de) 1971-10-01
BG17799A3 (bg) 1973-12-25
NO129954B (de) 1974-06-17
IE34765B1 (en) 1975-08-06
SE377938B (de) 1975-08-04
NL7017210A (de) 1971-05-28

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