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AU9393601A - Association of the cb1 receptor antagonist and a sibutramin, pharmaceutical compositions containing same and use thereof for treating obesity - Google Patents

Association of the cb1 receptor antagonist and a sibutramin, pharmaceutical compositions containing same and use thereof for treating obesity

Info

Publication number
AU9393601A
AU9393601A AU9393601A AU9393601A AU9393601A AU 9393601 A AU9393601 A AU 9393601A AU 9393601 A AU9393601 A AU 9393601A AU 9393601 A AU9393601 A AU 9393601A AU 9393601 A AU9393601 A AU 9393601A
Authority
AU
Australia
Prior art keywords
sibutramin
association
pharmaceutical compositions
compositions containing
receptor antagonist
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
AU9393601A
Inventor
Odile Piot-Grosjean
Philippe Picaut
Francois Petitet
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharma SA
Original Assignee
Aventis Pharma SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8854974&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU9393601(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aventis Pharma SA filed Critical Aventis Pharma SA
Publication of AU9393601A publication Critical patent/AU9393601A/en
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

The invention concerns the association of the CB1 receptor antagonist and a sibutramin, pharmaceutical compositions containing same and use thereof for treating obesity.
AU9393601A 2000-10-04 2001-10-01 Association of the cb1 receptor antagonist and a sibutramin, pharmaceutical compositions containing same and use thereof for treating obesity Pending AU9393601A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0012646A FR2814678B1 (en) 2000-10-04 2000-10-04 COMBINATION OF AN ANTAGONIST OF THE CB1 RECEPTOR AND SIBUTRAMINE, THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USE FOR THE TREATMENT OF OBESITY
PCT/FR2001/003022 WO2002028346A2 (en) 2000-10-04 2001-10-01 Association of the cb1 receptor antagonist and sibutramin, for treating obesity

Publications (1)

Publication Number Publication Date
AU9393601A true AU9393601A (en) 2002-04-15

Family

ID=8854974

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2001293936A Ceased AU2001293936B2 (en) 2000-10-04 2001-10-01 Association of the CB1 receptor antagonist and sibutramin, for treating obesity
AU9393601A Pending AU9393601A (en) 2000-10-04 2001-10-01 Association of the cb1 receptor antagonist and a sibutramin, pharmaceutical compositions containing same and use thereof for treating obesity

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AU2001293936A Ceased AU2001293936B2 (en) 2000-10-04 2001-10-01 Association of the CB1 receptor antagonist and sibutramin, for treating obesity

Country Status (29)

Country Link
EP (1) EP1328269B2 (en)
JP (1) JP4221221B2 (en)
KR (1) KR20030036885A (en)
CN (1) CN100409845C (en)
AT (1) ATE267595T1 (en)
AU (2) AU2001293936B2 (en)
BG (1) BG107739A (en)
BR (1) BR0114410A (en)
CA (1) CA2424934A1 (en)
DE (1) DE60103556T3 (en)
DK (1) DK1328269T5 (en)
EA (1) EA005924B1 (en)
EE (1) EE200300121A (en)
ES (1) ES2217191T5 (en)
FR (1) FR2814678B1 (en)
HR (1) HRP20030249A2 (en)
HU (1) HUP0302044A3 (en)
IL (1) IL155236A0 (en)
MX (1) MXPA03002845A (en)
NO (1) NO20031521L (en)
NZ (1) NZ524904A (en)
PL (1) PL362833A1 (en)
PT (1) PT1328269E (en)
SI (1) SI1328269T2 (en)
SK (1) SK4032003A3 (en)
TR (1) TR200401264T4 (en)
WO (1) WO2002028346A2 (en)
YU (1) YU26103A (en)
ZA (1) ZA200303015B (en)

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CA2479618A1 (en) 2002-03-26 2003-10-09 William K. Hagmann Spirocyclic amides as cannabinoid receptor modulators
WO2003082191A2 (en) 2002-03-28 2003-10-09 Merck & Co., Inc. Substituted 2,3-diphenyl pyridines
EP1499306A4 (en) 2002-04-12 2007-03-28 Merck & Co Inc Bicyclic amides
ATE389646T1 (en) 2002-07-29 2008-04-15 Hoffmann La Roche NEW BENZODIOXOLS
RU2330035C2 (en) 2003-01-02 2008-07-27 Ф.Хоффманн-Ля Рош Аг Pyrroleylthiazoles and their application as reverse agonists of receptor cb1
TW200413328A (en) 2003-01-02 2004-08-01 Hoffmann La Roche Novel CB 1 receptor inverse agonists
US7329658B2 (en) * 2003-02-06 2008-02-12 Pfizer Inc Cannabinoid receptor ligands and uses thereof
US20040224962A1 (en) * 2003-05-09 2004-11-11 Pfizer Inc Pharmaceutical composition for the treatment of obesity or to facilitate or promote weight loss
RU2006100298A (en) 2003-06-11 2006-05-10 Мерк энд Ко., Инк. (US) SUBSTITUTED 3-ALKYL-AND 3-ALKENYLASETIDINE DERIVATIVES
DE602004012858T2 (en) 2003-06-20 2009-05-14 F. Hoffmann-La Roche Ag 2-AMINOBENZOTHIAZOLE AS CB1 RECEPTOR INVERSE AGONISTS
EP1498123A1 (en) * 2003-07-18 2005-01-19 Aventis Pharma S.A. Emulsifying systems containing azetidine derivatives
EP1498122A1 (en) * 2003-07-18 2005-01-19 Aventis Pharma S.A. Semi-solid systems containing azetidine derivatives
EP1663215A1 (en) * 2003-09-02 2006-06-07 Solvay Pharmaceuticals GmbH Novel medical use of selective cb1- receptor antagonists
FR2861303A1 (en) * 2003-10-24 2005-04-29 Sanofi Synthelabo Use of pyrazole derivative as cannabinoid CB1 receptor antagonist, for treatment and prevention of metabolic syndrome, particularly cardiovascular risks, dyslipidemia and liver disease associated with obesity
WO2005049615A1 (en) * 2003-11-21 2005-06-02 Pfizer Products Inc. Pyrazolo`1,5-a!`1,3,5! triazin -4-one derivatives as cb1 receptor antagonists
AU2004299198A1 (en) 2003-12-08 2005-06-30 F. Hoffmann-La Roche Ag Novel thiazole derivates
ATE478856T1 (en) 2004-01-28 2010-09-15 Hoffmann La Roche SPIROBENZODIOXOLS AND THEIR USE AS CB1 ANTAGONISTS
ATE432275T1 (en) 2004-05-10 2009-06-15 Hoffmann La Roche PYRROLE OR IMIDAZOLAMIDE FOR THE TREATMENT OF OBESITAS
US20060025448A1 (en) 2004-07-22 2006-02-02 Cadila Healthcare Limited Hair growth stimulators
JP2008514718A (en) * 2004-09-29 2008-05-08 シェーリング コーポレイション Combinations of substituted azetidonones and CB1 antagonists
FR2876689B1 (en) 2004-10-14 2008-02-22 Aventis Pharma Sa NOVEL PROCESS AND INTERMEDIATES FOR PREPARING N- (1-BENZHYDRYL-AZETIDIN-3-YL) -N-PHENYL-METHYLSULFONAMIDE DERIVATIVES
WO2006045799A2 (en) 2004-10-25 2006-05-04 Solvay Pharmaceuticals Gmbh Pharmaceutical compositions comprising cb1 cannabinoid receptor antagonists and potassium channel openers for the treatment of diabetes mellitus type i, obesity and related conditions
ES2309812T3 (en) 2004-10-27 2008-12-16 F. Hoffmann-La Roche Ag NEW DERIVATIVES OF INDOL OR BENZIMIDAZOL.
WO2006050842A1 (en) 2004-11-09 2006-05-18 F. Hoffmann-La Roche Ag Dibenzosuberone derivatives
BRPI0609685A2 (en) 2005-04-06 2010-04-20 Hoffmann La Roche compounds, process for their manufacture, pharmaceutical compositions comprising them, method for treating and / or prophylaxis of diseases that are associated with modulating cb1 receptors, and using them
US7906652B2 (en) 2005-11-28 2011-03-15 Merck Sharp & Dohme Corp. Heterocycle-substituted 3-alkyl azetidine derivatives
US20090264470A1 (en) * 2006-02-21 2009-10-22 Bennett Teresa A CB1 Antagonists and Inverse Agonists
US8247442B2 (en) 2006-03-29 2012-08-21 Purdue Pharma L.P. Benzenesulfonamide compounds and their use
WO2007118853A1 (en) 2006-04-13 2007-10-25 Euro-Celtique S.A. Benzenesulfonamide compounds and their use as blockers of calcium channels
WO2007118854A1 (en) 2006-04-13 2007-10-25 Euro-Celtique S.A. Benzenesulfonamide compounds and the use thereof
US7629346B2 (en) 2006-06-19 2009-12-08 Hoffmann-La Roche Inc. Pyrazinecarboxamide derivatives as CB1 antagonists
WO2008038143A2 (en) * 2006-06-22 2008-04-03 Medichem, S.A. Novel solid forms of rimonabant and synthetic processes for their preparation
EP2057144A4 (en) * 2006-09-01 2010-06-02 Hetero Drugs Ltd Novel polymorphs of rimonabant
US7781593B2 (en) 2006-09-14 2010-08-24 Hoffmann-La Roche Inc. 5-phenyl-nicotinamide derivatives
AU2007300295A1 (en) * 2006-09-25 2008-04-03 Boehringer Ingelheim International Gmbh Compounds which modulate the CB2 receptor
DE102007002260A1 (en) 2007-01-16 2008-07-31 Sanofi-Aventis Use of substituted pyranonic acid derivatives for the preparation of medicaments for the treatment of the metabolic syndrome
EP1953144A1 (en) * 2007-01-30 2008-08-06 Sandoz AG Novel polymorphic forms of N-piperidino-5-(4-chlorophenyl)-1-(2, 4-dichlorphenyl)-4-methyl-3-pyrazolecarboxamide
US8399486B2 (en) 2007-04-09 2013-03-19 Purdue Pharma L.P. Benzenesulfonyl compounds and the use thereof
US8765736B2 (en) 2007-09-28 2014-07-01 Purdue Pharma L.P. Benzenesulfonamide compounds and the use thereof
PT2234966E (en) * 2007-12-18 2013-12-19 Sanofi Sa Azetidine derivatives, their preparation and their application in therapy
WO2010079241A1 (en) 2009-01-12 2010-07-15 Fundacion Hospital Nacional De Paraplejicos Para La Investigacion Y La Integracion Use of antagonists and/or inverse agonists of cb1 receptors for the preparation of drugs that increase motor neuron excitability
BRPI0902481B8 (en) 2009-07-31 2021-05-25 Soc Beneficente De Senhoras Hospital Sirio Libanes pharmaceutical composition comprising hemopressin and its use.
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Also Published As

Publication number Publication date
NZ524904A (en) 2004-11-26
EP1328269B1 (en) 2004-05-26
JP2004512279A (en) 2004-04-22
JP4221221B2 (en) 2009-02-12
TR200401264T4 (en) 2004-07-21
NO20031521L (en) 2003-04-24
EP1328269A2 (en) 2003-07-23
DK1328269T5 (en) 2009-03-16
YU26103A (en) 2006-08-17
SK4032003A3 (en) 2003-09-11
AU2001293936B2 (en) 2007-01-25
CN100409845C (en) 2008-08-13
PL362833A1 (en) 2004-11-02
DE60103556T3 (en) 2009-04-09
IL155236A0 (en) 2003-11-23
MXPA03002845A (en) 2004-09-10
EA200300441A1 (en) 2003-08-28
ES2217191T5 (en) 2009-02-16
SI1328269T2 (en) 2008-12-31
EE200300121A (en) 2005-04-15
BR0114410A (en) 2004-02-17
WO2002028346A3 (en) 2002-08-29
WO2002028346A2 (en) 2002-04-11
ES2217191T3 (en) 2004-11-01
FR2814678A1 (en) 2002-04-05
ZA200303015B (en) 2004-02-26
CN1473040A (en) 2004-02-04
FR2814678B1 (en) 2002-12-20
HRP20030249A2 (en) 2005-02-28
BG107739A (en) 2004-01-30
HUP0302044A3 (en) 2005-05-30
NO20031521D0 (en) 2003-04-03
SI1328269T1 (en) 2004-10-31
DK1328269T4 (en) 2008-11-24
DE60103556D1 (en) 2004-07-01
CA2424934A1 (en) 2002-04-11
DE60103556T2 (en) 2005-06-30
EP1328269B2 (en) 2008-07-30
DK1328269T3 (en) 2004-09-20
HUP0302044A2 (en) 2003-11-28
ATE267595T1 (en) 2004-06-15
PT1328269E (en) 2004-08-31
KR20030036885A (en) 2003-05-09
EA005924B1 (en) 2005-08-25

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