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AU5044499A - 2-ethyl-2,3-dihydrobenzofuran-carboxylic acid ester derivative, preparation method and use for preparing efaroxan derivatives - Google Patents

2-ethyl-2,3-dihydrobenzofuran-carboxylic acid ester derivative, preparation method and use for preparing efaroxan derivatives

Info

Publication number
AU5044499A
AU5044499A AU50444/99A AU5044499A AU5044499A AU 5044499 A AU5044499 A AU 5044499A AU 50444/99 A AU50444/99 A AU 50444/99A AU 5044499 A AU5044499 A AU 5044499A AU 5044499 A AU5044499 A AU 5044499A
Authority
AU
Australia
Prior art keywords
preparing
efaroxan
dihydrobenzofuran
ethyl
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU50444/99A
Inventor
Jean-Marie Autret
Karine Couture
Veronique Gouverneur
Patrick Lesimple
Charles Mioskowski
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pierre Fabre Sante
Original Assignee
Pierre Fabre Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pierre Fabre Sante filed Critical Pierre Fabre Sante
Publication of AU5044499A publication Critical patent/AU5044499A/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/82—Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/84—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D307/85—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

The invention concerns a 2-ethyl-3-hydroxy-2,3-dihydrobenzofuran of general formula (F) wherein: R represents a hydrogen atom, a halogen, a lower alkyl, lower alkoxy or hydroxy radical; and Z represents a C1-C3 alkoxy group or an amino group, and its use for preparing an Efaroxan derivative. The invention also concerns the method for preparing the derivative of general formula (F) from a corresponding salicylic aldehyde derivative.
AU50444/99A 1998-09-10 1999-07-26 2-ethyl-2,3-dihydrobenzofuran-carboxylic acid ester derivative, preparation method and use for preparing efaroxan derivatives Abandoned AU5044499A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9811303A FR2784989B1 (en) 1998-09-10 1998-09-10 2-ETHYL-2,3-DIHYDROBENZOFURANE-CARBOXYLIC ACID ESTER DERIVATIVE, PREPARATION METHOD AND USE FOR THE PREPARATION OF EFAROXAN DERIVATIVES
FR9811303 1998-09-10
PCT/FR1999/001848 WO2000015624A1 (en) 1998-09-10 1999-07-26 2-ethyl-2,3-dihydrobenzofuran-carboxylic acid ester derivative, preparation method and use for preparing efaroxan derivatives

Publications (1)

Publication Number Publication Date
AU5044499A true AU5044499A (en) 2000-04-03

Family

ID=9530300

Family Applications (1)

Application Number Title Priority Date Filing Date
AU50444/99A Abandoned AU5044499A (en) 1998-09-10 1999-07-26 2-ethyl-2,3-dihydrobenzofuran-carboxylic acid ester derivative, preparation method and use for preparing efaroxan derivatives

Country Status (7)

Country Link
EP (1) EP1112261B1 (en)
AT (1) ATE215940T1 (en)
AU (1) AU5044499A (en)
DE (1) DE69901262T2 (en)
ES (1) ES2176000T3 (en)
FR (1) FR2784989B1 (en)
WO (1) WO2000015624A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3997917B2 (en) * 2003-01-10 2007-10-24 株式会社デンソー Map search device

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZW13782A1 (en) * 1981-07-28 1982-10-06 Reckitt & Colmann Prod Ltd Imidazoline derivatives
GB2167408B (en) * 1984-11-23 1988-05-25 Farmos Oy Substituted imidazole derivatives and their preparation and use
GB9020128D0 (en) * 1990-09-14 1990-10-24 Reckitt & Colmann Prod Ltd Imidazoline derivatives
FR2733983B1 (en) * 1995-05-10 1997-08-01 Pf Medicament PROCESS FOR THE PREPARATION OF AN OPTICALLY PURE BENZOFURANE CARBOXYLIC ACID DERIVATIVE AND THE USE THEREOF FOR THE PREPARATION OF EFAROXAN

Also Published As

Publication number Publication date
WO2000015624A1 (en) 2000-03-23
EP1112261B1 (en) 2002-04-10
ES2176000T3 (en) 2002-11-16
ATE215940T1 (en) 2002-04-15
EP1112261A1 (en) 2001-07-04
FR2784989A1 (en) 2000-04-28
DE69901262D1 (en) 2002-05-16
FR2784989B1 (en) 2002-09-27
DE69901262T2 (en) 2002-11-21

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase