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AU3141197A - Antagonists of gonadotropin releasing hormone - Google Patents

Antagonists of gonadotropin releasing hormone

Info

Publication number
AU3141197A
AU3141197A AU31411/97A AU3141197A AU3141197A AU 3141197 A AU3141197 A AU 3141197A AU 31411/97 A AU31411/97 A AU 31411/97A AU 3141197 A AU3141197 A AU 3141197A AU 3141197 A AU3141197 A AU 3141197A
Authority
AU
Australia
Prior art keywords
antagonists
releasing hormone
gonadotropin releasing
gonadotropin
hormone
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU31411/97A
Other versions
AU712019B2 (en
Inventor
Robert J Devita
Mark Goulet
Matthew J. Wyvratt Jr.
Jonathan R. Young
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9613525.6A external-priority patent/GB9613525D0/en
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of AU3141197A publication Critical patent/AU3141197A/en
Application granted granted Critical
Publication of AU712019B2 publication Critical patent/AU712019B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU31411/97A 1996-05-20 1997-05-16 Antagonists of gonadotropin releasing hormone Ceased AU712019B2 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US1715196P 1996-05-20 1996-05-20
US60/017151 1996-05-20
GBGB9613525.6A GB9613525D0 (en) 1996-06-27 1996-06-27 Antagonists of gonadotropin releasing hormone
GB9613525 1996-06-27
PCT/US1997/008782 WO1997044041A1 (en) 1996-05-20 1997-05-16 Antagonists of gonadotropin releasing hormone

Publications (2)

Publication Number Publication Date
AU3141197A true AU3141197A (en) 1997-12-09
AU712019B2 AU712019B2 (en) 1999-10-28

Family

ID=26309582

Family Applications (1)

Application Number Title Priority Date Filing Date
AU31411/97A Ceased AU712019B2 (en) 1996-05-20 1997-05-16 Antagonists of gonadotropin releasing hormone

Country Status (5)

Country Link
EP (1) EP0920319A4 (en)
JP (1) JP2000511186A (en)
AU (1) AU712019B2 (en)
CA (1) CA2254974A1 (en)
WO (1) WO1997044041A1 (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2000511182A (en) * 1996-05-20 2000-08-29 メルク エンド カンパニー インコーポレーテッド Gonadotropin-releasing hormone antagonists
US6346534B1 (en) 1998-09-23 2002-02-12 Neurocrine Biosciences, Inc. Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
US6537998B1 (en) 1999-10-15 2003-03-25 Neurocrine Biosciences, Inc. Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
WO2001055119A2 (en) 2000-01-25 2001-08-02 Neurocrine Biosciences, Inc. Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
IL154624A0 (en) * 2000-09-22 2003-09-17 Akzo Nobel Nv Bicyclic heteroaromatic compounds
US6583153B2 (en) 2000-12-12 2003-06-24 Ortho-Mcneil Pharmaceutical, Inc. 7-heterocyclyl quinoline and thieno[2,3-b]yridine derivatives useful as antagonists of gonadotropin releasing hormone
AU2002247737B2 (en) * 2001-02-21 2006-05-18 Zentaris Gmbh Quinoline, isoquinoline and phthalazine derivatives as antagonists of the gonadotropin-releasing hormone
DE10108271A1 (en) 2001-02-21 2002-08-22 Schering Ag New oxo substituted quinoline, isoquinoline and phthalazine derivatives useful as GnRH antagonists in male fertility control, female infertility and contraception and tumor control
US6740656B2 (en) 2001-08-02 2004-05-25 Neurocrine Biosciences, Inc. Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
WO2003011293A2 (en) 2001-08-02 2003-02-13 Neurocrine Biosciences, Inc. Pyridinone and pyridazinone derivatives as gonadotropin-releasing hormone receptor antagonists
US6673796B2 (en) 2001-08-02 2004-01-06 Neurocrine Biosciences, Inc. Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
WO2003013528A1 (en) 2001-08-02 2003-02-20 Neurocrine Biosciences, Inc. Substituted pyridin-4-ones and their use as gonadotropin-releasing hormone receptor antagonists.
AU2002324586B2 (en) 2001-08-02 2008-04-24 Neurocrine Biosciences, Inc. 1,3,5-triazine-2,4,6-triones, preparation and use as gonadotropin-releasing hormone receptor antagonists
GB0223730D0 (en) * 2002-10-11 2002-11-20 Novartis Ag Organic compounds
GB0307777D0 (en) 2003-04-04 2003-05-07 Medical Res Council Conjugate compounds
GB0412769D0 (en) 2004-06-08 2004-07-07 Novartis Ag Organic compounds
TW201130854A (en) 2009-12-22 2011-09-16 Bayer Schering Pharma Ag Pyridinone derivatives and pharmaceutical compositions thereof
WO2012175514A1 (en) 2011-06-21 2012-12-27 Bayer Intellectual Property Gmbh Pyridinone derivatives and pharmaceutical compositions thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI80022C (en) * 1982-07-05 1990-04-10 Otsuka Pharma Co Ltd FOERFARANDE FOER FRAMSTAELLNING AV ETT NYTT, TERAPEUTISKT ANVAENDBART KARBOSTYRILDERIVAT.
GB9125515D0 (en) * 1991-11-29 1992-01-29 Merck Sharp & Dohme Therapeutic agents
US5656643A (en) * 1993-11-08 1997-08-12 Rhone-Poulenc Rorer Pharmaceuticals Inc. Bis mono-and bicyclic aryl and heteroaryl compounds which inhibit EGF and/or PDGF receptor tyrosine kinase
US5607939A (en) * 1994-04-28 1997-03-04 Takeda Chemical Industries, Ltd. Condensed heterocyclic compounds, their production and use
JP2000511182A (en) * 1996-05-20 2000-08-29 メルク エンド カンパニー インコーポレーテッド Gonadotropin-releasing hormone antagonists

Also Published As

Publication number Publication date
EP0920319A4 (en) 2002-05-02
EP0920319A1 (en) 1999-06-09
CA2254974A1 (en) 1997-11-27
JP2000511186A (en) 2000-08-29
AU712019B2 (en) 1999-10-28
WO1997044041A1 (en) 1997-11-27

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Legal Events

Date Code Title Description
MK14 Patent ceased section 143(a) (annual fees not paid) or expired