AU2003256006A8 - Improved process for preparation of risperidone - Google Patents
Improved process for preparation of risperidoneInfo
- Publication number
- AU2003256006A8 AU2003256006A8 AU2003256006A AU2003256006A AU2003256006A8 AU 2003256006 A8 AU2003256006 A8 AU 2003256006A8 AU 2003256006 A AU2003256006 A AU 2003256006A AU 2003256006 A AU2003256006 A AU 2003256006A AU 2003256006 A8 AU2003256006 A8 AU 2003256006A8
- Authority
- AU
- Australia
- Prior art keywords
- risperidone
- preparation
- improved process
- improved
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- RAPZEAPATHNIPO-UHFFFAOYSA-N risperidone Chemical compound FC1=CC=C2C(C3CCN(CC3)CCC=3C(=O)N4CCCCC4=NC=3C)=NOC2=C1 RAPZEAPATHNIPO-UHFFFAOYSA-N 0.000 title 1
- 229960001534 risperidone Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN507CA2002 | 2002-08-30 | ||
IN507CAL2002 | 2002-08-30 | ||
PCT/IB2003/003830 WO2004020439A2 (en) | 2002-08-30 | 2003-08-25 | Improved process for preparation of risperidone |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2003256006A8 true AU2003256006A8 (en) | 2004-03-19 |
AU2003256006A1 AU2003256006A1 (en) | 2004-03-19 |
Family
ID=31972123
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2003256006A Abandoned AU2003256006A1 (en) | 2002-08-30 | 2003-08-25 | Improved process for preparation of risperidone |
Country Status (3)
Country | Link |
---|---|
AU (1) | AU2003256006A1 (en) |
BR (1) | BR0306204A (en) |
WO (1) | WO2004020439A2 (en) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IS7290A (en) * | 2004-05-28 | 2005-11-29 | Actavis Group | Pharmaceutical formulations containing risperidone |
US8852638B2 (en) | 2005-09-30 | 2014-10-07 | Durect Corporation | Sustained release small molecule drug formulation |
MX337286B (en) | 2007-05-25 | 2016-02-22 | Indivior Uk Ltd | Sustained delivery formulations of risperidone compounds. |
CN105481854B (en) * | 2015-12-08 | 2017-11-10 | 天津市亨必达化学合成物有限公司 | A kind of preparation method of the brilliant III type material of Risperidone |
CN105367570B (en) * | 2015-12-08 | 2017-10-10 | 天津市亨必达化学合成物有限公司 | A kind of preparation method of Risperidone crystalline substance I type materials |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4804663A (en) * | 1985-03-27 | 1989-02-14 | Janssen Pharmaceutica N.V. | 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles |
US4957916A (en) * | 1988-08-05 | 1990-09-18 | Janssen Pharmaceutica N.V. | Antipsychotic 3-piperazinylbenzazole derivatives |
GB9008850D0 (en) * | 1990-04-19 | 1990-06-13 | Janssen Pharmaceutica Nv | Novel 2,9-disubstituted-4h-pyridol(1,2-a)pyrimidin-4-ones |
ES2050069B1 (en) * | 1992-07-10 | 1994-12-16 | Vita Invest Sa | PROCEDURE FOR OBTAINING 3- (2- (4- (6-FLUORO-1,2-BENZISOXAZOL-3-IL) PIPERIDINO) ETIL) -2-METHYL-6,7,8,9-TETRAHIDRO-4H-PIRIDO (1,2-A) PIRIMIDIN-4-ONA. |
WO1995014691A1 (en) * | 1993-11-23 | 1995-06-01 | Janssen Pharmaceutica N.V. | NOVEL 9-HYDROXY-PYRIDO[1,2-a]PYRIMIDIN-4-ONE ETHER DERIVATIVES |
US6331317B1 (en) * | 1999-11-12 | 2001-12-18 | Alkermes Controlled Therapeutics Ii Inc. | Apparatus and method for preparing microparticles |
SK2982003A3 (en) * | 2000-08-14 | 2004-10-05 | Teva Pharma | Preparation of risperidone |
US20020193386A1 (en) * | 2002-03-28 | 2002-12-19 | Inigo Pfeiffer | Polymorphic form of 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-alpha]pyrimidin-4-one and formulations thereof |
-
2003
- 2003-08-25 AU AU2003256006A patent/AU2003256006A1/en not_active Abandoned
- 2003-08-25 WO PCT/IB2003/003830 patent/WO2004020439A2/en not_active Application Discontinuation
- 2003-08-25 BR BR0306204-0A patent/BR0306204A/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2004020439A2 (en) | 2004-03-11 |
WO2004020439A3 (en) | 2004-07-01 |
AU2003256006A1 (en) | 2004-03-19 |
BR0306204A (en) | 2004-09-08 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |