AU2002251481A1 - Carboxylic acid derivative and salt thereof - Google Patents
Carboxylic acid derivative and salt thereofInfo
- Publication number
- AU2002251481A1 AU2002251481A1 AU2002251481A AU2002251481A AU2002251481A1 AU 2002251481 A1 AU2002251481 A1 AU 2002251481A1 AU 2002251481 A AU2002251481 A AU 2002251481A AU 2002251481 A AU2002251481 A AU 2002251481A AU 2002251481 A1 AU2002251481 A1 AU 2002251481A1
- Authority
- AU
- Australia
- Prior art keywords
- salt
- carboxylic acid
- acid derivative
- derivative
- carboxylic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2001123346 | 2001-04-20 | ||
JP2001-123346 | 2001-04-20 | ||
JP2002-36274 | 2002-02-14 | ||
JP2002036274 | 2002-02-14 | ||
PCT/JP2002/003866 WO2002100812A1 (en) | 2001-04-20 | 2002-04-18 | Carboxylic acid derivative and salt thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2002251481A1 true AU2002251481A1 (en) | 2003-05-15 |
AU2002251481B2 AU2002251481B2 (en) | 2007-08-09 |
Family
ID=26613950
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2002251481A Ceased AU2002251481B2 (en) | 2001-04-20 | 2002-04-18 | Carboxylic acid derivative and salt thereof |
Country Status (19)
Country | Link |
---|---|
US (1) | US7544835B2 (en) |
EP (1) | EP1380562A4 (en) |
JP (1) | JP4131698B2 (en) |
KR (1) | KR100888001B1 (en) |
CN (1) | CN100522944C (en) |
AU (1) | AU2002251481B2 (en) |
BR (1) | BR0209027A (en) |
CA (1) | CA2442319C (en) |
CZ (1) | CZ20032727A3 (en) |
HU (1) | HUP0303810A3 (en) |
IL (1) | IL157731A0 (en) |
MX (1) | MXPA03009565A (en) |
NO (1) | NO329995B1 (en) |
NZ (2) | NZ528655A (en) |
PL (1) | PL206767B1 (en) |
RU (1) | RU2316537C2 (en) |
SG (1) | SG161743A1 (en) |
TW (1) | TWI311133B (en) |
WO (1) | WO2002100812A1 (en) |
Families Citing this family (54)
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EP1375472A4 (en) | 2001-03-30 | 2008-12-10 | Eisai R&D Man Co Ltd | Benzene compound and salt thereof |
TWI311133B (en) | 2001-04-20 | 2009-06-21 | Eisai R&D Man Co Ltd | Carboxylic acid derivativeand the salt thereof |
WO2002098840A1 (en) | 2001-06-04 | 2002-12-12 | Eisai Co., Ltd. | Carboxylic acid derivative and medicine comprising salt or ester of the same |
CN1543451A (en) * | 2001-06-07 | 2004-11-03 | Receptor modulators activated by peroxizonal proliferators (ppar) | |
US7371777B2 (en) | 2001-08-17 | 2008-05-13 | Eisai Co., Ltd. | Cyclic compound and PPAR agonist |
SE0104333D0 (en) | 2001-12-19 | 2001-12-19 | Astrazeneca Ab | Therapeutic agents |
US7816385B2 (en) * | 2002-12-20 | 2010-10-19 | High Point Pharmaceuticals, Llc | Dimeric dicarboxylic acid derivatives, their preparation and use |
US20060177444A1 (en) * | 2003-03-20 | 2006-08-10 | Tatsuo Horizoe | Concomitant drug as therapeutic agent for inflammatory bowel disease |
JP2007186515A (en) * | 2003-05-02 | 2007-07-26 | Takara Bio Inc | Curative agent |
MY150088A (en) | 2003-05-19 | 2013-11-29 | Irm Llc | Immunosuppressant compounds and compositions |
GB0314131D0 (en) * | 2003-06-18 | 2003-07-23 | Astrazeneca Ab | Therapeutic agents |
WO2005014755A1 (en) * | 2003-08-08 | 2005-02-17 | Ube Industries, Ltd. | Alkynyl group-substituted condensed heterocyclic compound, method for producing same, and organic electroluminescent device using same |
AU2004267085B2 (en) * | 2003-08-20 | 2010-09-16 | Pharmacyclics, Inc. | Acetylene derivatives as inhibitors of histone deacetylase |
WO2005086661A2 (en) | 2004-02-27 | 2005-09-22 | Amgen Inc. | Compounds, pharmaceutical compositions and methods for use in treating metabolic disorders |
WO2005093423A2 (en) * | 2004-03-26 | 2005-10-06 | Bayer Healthcare Ag | Diagnostics and therapeutics for diseases associated with peroxisome proliferative activated receptor alpha (ppara) |
WO2005105726A1 (en) | 2004-05-05 | 2005-11-10 | Novo Nordisk A/S | Novel compounds, their preparation and use |
JP4981662B2 (en) | 2004-05-05 | 2012-07-25 | ハイ・ポイント・ファーマスーティカルズ、エルエルシー | New compounds, their preparation and use |
FR2872159B1 (en) * | 2004-06-28 | 2007-10-05 | Merck Sante Soc Par Actions Si | NOVEL PHENYL CARBOXYLIC ACID DERIVATIVES AND THEIR USE IN THE TREATMENT OF DIABETES |
AU2005259579A1 (en) * | 2004-07-01 | 2006-01-12 | F. Hoffmann-La Roche Ag | Phenyl derivatives comprising an acetylene group |
US7405236B2 (en) * | 2004-08-16 | 2008-07-29 | Hoffman-La Roche Inc. | Indole derivatives comprising an acetylene group |
ITMI20041825A1 (en) * | 2004-09-24 | 2004-12-24 | Medestea Res & Production Srl | RECEPTOR AGONISTS ACTIVATING THE PROLIFERATION OF PEROXYSOMES, USEFUL IN THE PREVENTION OR TREATMENT OF GASTRITIS |
US20090069591A1 (en) * | 2005-04-19 | 2009-03-12 | Eisai R & D Management Co., Ltd. | Calcium Bis [ (2S) -3- [3-[ (2S) -3- (4-Chloro-2-Cyanophenoxy) -2- Fluoropropoxy]Phenyl] -2- Isopropoxypropionate] and Intermediate Thereof |
US7816405B2 (en) * | 2005-04-19 | 2010-10-19 | Eisai R&D Management Co., Ltd. | Calcium bis [(2S)-3-[3-[(2S)-3-(4-chloro-2-cyanophenoxy)-2-fluoropropoxy]phenyl ]-2-isopropoxypropionate] and intermediate thereof |
US7465804B2 (en) | 2005-05-20 | 2008-12-16 | Amgen Inc. | Compounds, pharmaceutical compositions and methods for their use in treating metabolic disorders |
ES2382876T3 (en) | 2005-05-31 | 2012-06-14 | Pfizer, Inc. | Aryloxy-N-bicyclomethyl-acetamide compounds substituted as VR1 antagonists |
TW200718691A (en) * | 2005-06-10 | 2007-05-16 | Sigma Tau Ind Farmaceuti | Cinnamic and phenylpropiolic acid derivatives useful as anti-tumour agents |
ES2372617T3 (en) | 2005-06-30 | 2012-01-24 | High Point Pharmaceuticals, Llc | PHENOXYACETIC ACIDS AS ACTIVATORS OF PPAR-DELTA. |
CA2621949A1 (en) | 2005-09-14 | 2007-03-22 | Amgen Inc. | Conformationally constrained 3- (4-hydroxy-phenyl) - substituted-propanoic acids useful for treating metabolic disorders |
JP2007166908A (en) * | 2005-12-19 | 2007-07-05 | Sumitomo Chemical Co Ltd | Process for producing optically active 3- (3-hydroxyphenyl) -2-alkoxypropanoic acid or 3- (3-hydroxyphenyl) -2-alkoxypropanoic acid ester |
EA201101084A1 (en) | 2005-12-22 | 2012-04-30 | ХАЙ ПОЙНТ ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи | PHENOXYACIC ACIDS AS PPAR DELTA ACTIVATORS |
JP2009529512A (en) | 2006-03-09 | 2009-08-20 | ハイ ポイント ファーマシューティカルズ,リミティド ライアビリティ カンパニー | Novel compounds, methods for their production and use |
NZ574038A (en) | 2006-06-27 | 2011-12-22 | Takeda Pharmaceutical | Fused cyclic compounds as GPR40 receptor function modulators, for treating diabetes |
WO2008030618A1 (en) | 2006-09-07 | 2008-03-13 | Amgen Inc. | Benzo-fused compounds for use in treating metabolic disorders |
AU2007293028B2 (en) | 2006-09-07 | 2012-05-31 | Amgen Inc. | Heterocyclic GPR40 modulators |
CA2679514A1 (en) * | 2007-03-01 | 2008-09-04 | Bayer Schering Pharma Aktiengesellschaft | 18f fluoro-benzoyl labelled biologically active compounds as diagnostic imaging agents as well as benzotriazol-1-yloxy-benzoyl, 2,5-dioxo-pyrrolidin-1-yloxy-benzoyl and trimethylammonio-benzoyl precursers |
ES2550479T3 (en) * | 2007-04-05 | 2015-11-10 | Daiichi Sankyo Company, Limited | Condensed bicyclic heteroaryl derivatives |
US7572934B2 (en) | 2007-04-16 | 2009-08-11 | Amgen Inc. | Substituted biphenyl GPR40 modulators |
KR101196680B1 (en) | 2007-06-29 | 2012-11-06 | 어큐셀라 인코포레이티드 | Alkynyl phenyl derivative compounds for treating ophthalmic diseases and disorders |
BRPI0818253A2 (en) | 2007-10-10 | 2015-04-07 | Amgen Inc | Substituted biphenyl gpr40 modulators |
US8450522B2 (en) | 2008-03-06 | 2013-05-28 | Amgen Inc. | Conformationally constrained carboxylic acid derivatives useful for treating metabolic disorders |
ES2450567T3 (en) | 2008-10-15 | 2014-03-25 | Amgen, Inc | GPR40 spirocyclic modulators |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
TW201215387A (en) | 2010-07-05 | 2012-04-16 | Sanofi Aventis | Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament |
TW201215388A (en) | 2010-07-05 | 2012-04-16 | Sanofi Sa | (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments |
EP2759533B1 (en) * | 2011-09-22 | 2017-08-02 | Takeda Pharmaceutical Company Limited | Condensed heterocyclic compound |
KR102157912B1 (en) * | 2012-08-03 | 2020-09-21 | 더 보드 오브 트러스티즈 오브 더 유니버시티 오브 일리노이 | Enzyme-activating compounds and compositions |
CN109400502A (en) * | 2013-07-22 | 2019-03-01 | 新陈代谢解决方案开发公司 | The regulated compound of PPAR- for treating metabolic disease |
PE20160901A1 (en) * | 2013-12-18 | 2016-08-27 | Astex Therapeutics Ltd | NRF2 REGULATORS |
EP3240785B1 (en) | 2014-12-29 | 2021-07-07 | The United States of America, as represented by The Secretary, Department of Health and Human Services | Small molecule inhibitors of lactate dehydrogenase and methods of use thereof |
PL3307739T3 (en) | 2015-06-15 | 2021-05-31 | Glaxosmithkline Intellectual Property Development Limited | Nrf2 regulators |
US10272095B2 (en) | 2015-06-15 | 2019-04-30 | GlaxoSmithKline Intellectual Propert Development Limited | NRF2 regulators |
EP3359532A1 (en) | 2015-10-06 | 2018-08-15 | GlaxoSmithKline Intellectual Property Development Limited | Biaryl pyrazoles as nrf2 regulators |
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JPS5649336A (en) | 1979-09-05 | 1981-05-02 | Glaxo Group Ltd | Phenol derivative* its manufacture and its use |
DE3026924A1 (en) * | 1980-07-16 | 1982-02-18 | Klinge Pharma GmbH & Co, 8000 München | 1,3-Di:phenoxy-propan-2-ol derivs. - used as hypolipaemics to reduce tri:glyceride and cholesterol levels in the blood |
JPS5764639A (en) * | 1980-10-04 | 1982-04-19 | Nippon Zoki Pharmaceut Co Ltd | Novel stilbene derivative, its preparation, and medical composition containing the same as active ingredent |
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GB9225386D0 (en) * | 1992-12-04 | 1993-01-27 | Smithkline Beecham Plc | Novel compounds |
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US6130214A (en) | 1997-10-27 | 2000-10-10 | Dr. Reddy's Research Foundation | Benzothiazin and benzoxazin derivatives; their preparation and uses |
JPH11152269A (en) | 1997-11-20 | 1999-06-08 | Teijin Ltd | Biphenylamindine derivative |
MY153569A (en) | 1998-01-20 | 2015-02-27 | Mitsubishi Tanabe Pharma Corp | Inhibitors of ?4 mediated cell adhesion |
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FR2781222A1 (en) | 1998-07-17 | 2000-01-21 | Lipha | New cyclic peroxisome proliferator activated receptor activators, used to prevent or treat dyslipidemia, atherosclerosis and diabetes |
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DE60025621T2 (en) | 1999-09-17 | 2006-11-23 | Kyorin Pharmaceutical Co., Ltd. | O anisamide DERIVATIVES |
TWI262185B (en) | 1999-10-01 | 2006-09-21 | Eisai Co Ltd | Carboxylic acid derivatives having anti-hyperglycemia and anti-hyperlipemia action, and pharmaceutical composition containing the derivatives |
DE19947457A1 (en) | 1999-10-02 | 2001-04-05 | Aventis Pharma Gmbh | New 2'-aminomethyl-biphenyl-2-carboxamide derivatives, are potassium channel blockers especially useful for treating re-entry or supraventricular arrhythmia or atrial fibrillation or flutter |
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JP2001261612A (en) | 2000-03-22 | 2001-09-26 | Mitsui Chemicals Inc | Catecholpropionic acid derivative and nuclear receptor agonist containing the same as active ingredient |
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JP4256166B2 (en) * | 2001-03-28 | 2009-04-22 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | Carboxylic acid compound |
EP1375472A4 (en) * | 2001-03-30 | 2008-12-10 | Eisai R&D Man Co Ltd | Benzene compound and salt thereof |
WO2002080899A1 (en) | 2001-03-30 | 2002-10-17 | Eisai Co., Ltd. | Remedial agent for digestive disease |
WO2002083616A1 (en) | 2001-04-10 | 2002-10-24 | Sankyo Company, Limited | α-SUBSTITUTED φ-ARYLFATTY ACID DERIVATIVE |
TWI311133B (en) | 2001-04-20 | 2009-06-21 | Eisai R&D Man Co Ltd | Carboxylic acid derivativeand the salt thereof |
WO2002098840A1 (en) * | 2001-06-04 | 2002-12-12 | Eisai Co., Ltd. | Carboxylic acid derivative and medicine comprising salt or ester of the same |
US7371777B2 (en) * | 2001-08-17 | 2008-05-13 | Eisai Co., Ltd. | Cyclic compound and PPAR agonist |
FR2833949B1 (en) | 2001-12-21 | 2005-08-05 | Galderma Res & Dev | NOVEL PPARy RECEPTOR ACTIVATION LIGANDS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN HUMAN MEDICINE AND COSMETICS |
-
2002
- 2002-04-17 TW TW091107890A patent/TWI311133B/en not_active IP Right Cessation
- 2002-04-18 CA CA2442319A patent/CA2442319C/en not_active Expired - Fee Related
- 2002-04-18 RU RU2003133744/04A patent/RU2316537C2/en not_active IP Right Cessation
- 2002-04-18 WO PCT/JP2002/003866 patent/WO2002100812A1/en active IP Right Grant
- 2002-04-18 NZ NZ528655A patent/NZ528655A/en unknown
- 2002-04-18 KR KR1020037013180A patent/KR100888001B1/en not_active Expired - Fee Related
- 2002-04-18 CZ CZ20032727A patent/CZ20032727A3/en unknown
- 2002-04-18 JP JP2003503583A patent/JP4131698B2/en not_active Expired - Fee Related
- 2002-04-18 CN CNB028084985A patent/CN100522944C/en not_active Expired - Fee Related
- 2002-04-18 BR BR0209027-9A patent/BR0209027A/en not_active Application Discontinuation
- 2002-04-18 NZ NZ539708A patent/NZ539708A/en unknown
- 2002-04-18 EP EP02720489A patent/EP1380562A4/en not_active Withdrawn
- 2002-04-18 AU AU2002251481A patent/AU2002251481B2/en not_active Ceased
- 2002-04-18 IL IL15773102A patent/IL157731A0/en unknown
- 2002-04-18 PL PL367196A patent/PL206767B1/en not_active IP Right Cessation
- 2002-04-18 SG SG200608047-7A patent/SG161743A1/en unknown
- 2002-04-18 HU HU0303810A patent/HUP0303810A3/en unknown
- 2002-04-18 MX MXPA03009565A patent/MXPA03009565A/en active IP Right Grant
- 2002-04-18 US US10/472,543 patent/US7544835B2/en not_active Expired - Fee Related
-
2003
- 2003-10-17 NO NO20034669A patent/NO329995B1/en not_active IP Right Cessation
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