AU2001279700A1 - 5-aminoalkyl-pyrazolo(4,3-d)pyrimidines with a phosphodiesterase v-inhibiting effect - Google Patents

5-aminoalkyl-pyrazolo(4,3-d)pyrimidines with a phosphodiesterase v-inhibiting effect

Info

Publication number: AU2001279700A1
Authority: AU; Australia
Prior art keywords: pyrazolo; phosphodiesterase; pyrimidines; aminoalkyl; inhibiting effect
Prior art date: 2000-06-29
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU2001279700A

Other versions

AU2001279700B2 (en

Inventor

Norbert Beier

Maria Christadler

Rochus Jonas

Pierre Schelling

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Merck Patent GmbH

Original Assignee

Merck Patent GmbH

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-06-29

Filing date

2001-06-28

Publication date

2002-03-28

2000-06-29 Priority claimed from DE10031584A external-priority patent/DE10031584A1/en

2001-06-28 Application filed by Merck Patent GmbH filed Critical Merck Patent GmbH

2002-03-28 Publication of AU2001279700A1 publication Critical patent/AU2001279700A1/en

2006-08-24 Application granted granted Critical

2006-08-24 Publication of AU2001279700B2 publication Critical patent/AU2001279700B2/en

2021-06-28 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DE10031584A DE10031584A1 (en)	2000-06-29	2000-06-29	5-aminoalkyl-pyrazolo [4,3-d] pyrimidine
DE10031584.4		2000-06-29
PCT/EP2001/007378 WO2002000660A1 (en)	2000-06-29	2001-06-28	5-aminoalkyl-pyrazolo[4,3-d]pyrimidines with a phosphodiesterase v-inhibiting effect

Publications (2)

Publication Number	Publication Date
AU2001279700A1 true AU2001279700A1 (en)	2002-03-28
AU2001279700B2 AU2001279700B2 (en)	2006-08-24

Family

ID=7647151

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AU2001279700A Ceased AU2001279700B2 (en)	2000-06-29	2001-06-28	5-aminoalkyl-pyrazolo(4,3-d)pyrimidines with a phosphodiesterase v-inhibiting effect
AU7970001A Pending AU7970001A (en)	2000-06-29	2001-06-28	5-aminoalkyl-pyrazolo(4,3-d)pyrimidines with a phosphodiesterase v-inhibiting effect

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
AU7970001A Pending AU7970001A (en)	2000-06-29	2001-06-28	5-aminoalkyl-pyrazolo(4,3-d)pyrimidines with a phosphodiesterase v-inhibiting effect

Country Status (21)

Country	Link
US (1)	US7060823B2 (en)
EP (1)	EP1296986B1 (en)
JP (1)	JP4964388B2 (en)
KR (1)	KR20030017558A (en)
CN (1)	CN1439011A (en)
AR (1)	AR028772A1 (en)
AT (1)	ATE519761T1 (en)
AU (2)	AU2001279700B2 (en)
BR (1)	BR0111915A (en)
CA (1)	CA2410399C (en)
CZ (1)	CZ20024054A3 (en)
DE (1)	DE10031584A1 (en)
ES (1)	ES2367704T3 (en)
HU (1)	HUP0301587A3 (en)
MX (1)	MXPA02012263A (en)
NO (1)	NO20026247D0 (en)
PL (1)	PL358551A1 (en)
RU (1)	RU2271359C2 (en)
SK (1)	SK17632002A3 (en)
WO (1)	WO2002000660A1 (en)
ZA (1)	ZA200209728B (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE19942474A1 (en) *	1999-09-06	2001-03-15	Merck Patent Gmbh	Pyrazolo [4,3-d] pyrimidines
DE10031585A1 (en) *	2000-06-29	2002-01-10	Merck Patent Gmbh	2-aminoalkyl-thieno [2,3-d] pyrimidine
DE10058662A1 (en) *	2000-11-25	2002-05-29	Merck Patent Gmbh	Use of pyrazolo [4,3-d] pyrimidines
CN100439371C (en) *	2003-04-29	2008-12-03	辉瑞大药厂	5,7-Diaminopyrazolo[4,3-d]pyrimidines useful in the treatment of hypertension
BRPI0409903A (en)	2003-04-29	2006-04-25	Pfizer Ltd	5,7-diamino pyrazol [4,3-d] pyrimidine useful in treating hypertension
GB0327319D0 (en) *	2003-11-24	2003-12-24	Pfizer Ltd	Novel pharmaceuticals
US7572799B2 (en)	2003-11-24	2009-08-11	Pfizer Inc	Pyrazolo[4,3-d]pyrimidines as Phosphodiesterase Inhibitors
GB0327323D0 (en) *	2003-11-24	2003-12-31	Pfizer Ltd	Novel pharmaceuticals
US7569572B2 (en) *	2004-04-07	2009-08-04	Pfizer Inc	Pyrazolo[4,3-D]pyrimidines
EP1809632A2 (en) *	2004-10-28	2007-07-25	Pharmacia & Upjohn Company LLC	Pyrazolo[4,3-d]pyrimidine derivatives useful as pde-5 inhibitors
PT1881985E (en)	2005-05-12	2011-02-01	Pfizer	Anhydrous crystalline forms of n-ý1-(2-ethoxyethyl)-5-(n-ethyl-n-methylamino)-7-(4-methylpyridin-2-yl-amino)-1h-pyrazolo[4,3-d]pyrimidine-3-carbonyl¨methanesulfonamide
NL2000291C2 (en)	2005-11-10	2009-02-17	Pfizer Prod Inc	1- (1- (2-ethoxyethyl) -3-ethyl-7- (4-methylpyridin-2-ylamino) -1 H -pyrazole (4,3-d) pyrimidin-5-yl) piperidine-4-carboxylic acid and salts thereof.
DE102012200360A1 (en) *	2012-01-11	2013-07-11	Bayer Intellectual Property Gmbh	Substituted triazines and their use
CA2782774A1 (en) *	2012-07-06	2014-01-06	Pharmascience Inc.	Protein kinase inhibitors

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SU1739850A3 (en) *	1987-08-31	1992-06-07	Такеда Кемикал Индастриз, Лтд (Фирма)	Method for synthesis of condensed derivatives of pyrazolo-[3,4-d]-pyrimidine
US5075310A (en) *	1988-07-01	1991-12-24	Smith Kline & French Laboratories, Ltd.	Pyrimidone derivatives as bronchodilators
GB9119704D0 (en) *	1991-09-14	1991-10-30	Pfizer Ltd	Therapeutic agents
JP2657760B2 (en) *	1992-07-15	1997-09-24	小野薬品工業株式会社	4-aminoquinazoline derivatives and pharmaceuticals containing them
GB9301192D0 (en)	1993-06-09	1993-06-09	Trott Francis W	Flower shaped mechanised table
GB9423911D0 (en) *	1994-11-26	1995-01-11	Pfizer Ltd	Therapeutic agents
US5869486A (en) *	1995-02-24	1999-02-09	Ono Pharmaceutical Co., Ltd.	Fused pyrimidines and pyriazines as pharmaceutical compounds
DE19644228A1 (en)	1996-10-24	1998-04-30	Merck Patent Gmbh	Thienopyrimidines
DE19752952A1 (en)	1997-11-28	1999-06-02	Merck Patent Gmbh	Thienopyrimidines
DE19942474A1 (en) *	1999-09-06	2001-03-15	Merck Patent Gmbh	Pyrazolo [4,3-d] pyrimidines

2000
- 2000-06-29 DE DE10031584A patent/DE10031584A1/en not_active Withdrawn
2001
- 2001-06-28 ES ES01957901T patent/ES2367704T3/en not_active Expired - Lifetime
- 2001-06-28 EP EP01957901A patent/EP1296986B1/en not_active Expired - Lifetime
- 2001-06-28 KR KR1020027017571A patent/KR20030017558A/en not_active Withdrawn
- 2001-06-28 CN CN01811801A patent/CN1439011A/en active Pending
- 2001-06-28 SK SK1763-2002A patent/SK17632002A3/en unknown
- 2001-06-28 US US10/312,766 patent/US7060823B2/en not_active Expired - Fee Related
- 2001-06-28 BR BR0111915-0A patent/BR0111915A/en not_active IP Right Cessation
- 2001-06-28 RU RU2003100508/04A patent/RU2271359C2/en not_active IP Right Cessation
- 2001-06-28 HU HU0301587A patent/HUP0301587A3/en unknown
- 2001-06-28 AU AU2001279700A patent/AU2001279700B2/en not_active Ceased
- 2001-06-28 MX MXPA02012263A patent/MXPA02012263A/en unknown
- 2001-06-28 WO PCT/EP2001/007378 patent/WO2002000660A1/en active Application Filing
- 2001-06-28 JP JP2002505784A patent/JP4964388B2/en not_active Expired - Fee Related
- 2001-06-28 PL PL01358551A patent/PL358551A1/en unknown
- 2001-06-28 CZ CZ20024054A patent/CZ20024054A3/en unknown
- 2001-06-28 AT AT01957901T patent/ATE519761T1/en active
- 2001-06-28 CA CA2410399A patent/CA2410399C/en not_active Expired - Fee Related
- 2001-06-28 AU AU7970001A patent/AU7970001A/en active Pending
- 2001-06-29 AR ARP010103144A patent/AR028772A1/en unknown
2002
- 2002-11-29 ZA ZA200209728A patent/ZA200209728B/en unknown
- 2002-12-27 NO NO20026247A patent/NO20026247D0/en not_active Application Discontinuation

Publication	Publication Date	Title
EP1416935B8 (en)	2008-08-27	4-amino-6-phenyl-pyrrolo[2,3-d]pyrimidine derivatives
IL158697A0 (en)	2004-05-12	4-amino-5-phenyl-7-cyclobutyl-pyrrolo (2,3-d) pyrimidine derivatives
SI1220856T1 (en)	2005-06-30	Pyrazolo(4,3-d)pyrimidine derivatives
AU2002221344A1 (en)	2002-09-05	Antiviral agents
HRP20020798A2 (en)	2004-02-29	5-ALKYLPYRIDO[2,3-d]PYRIMIDINES TYROZINE KINASE INHIBITORS
EP1255764B8 (en)	2006-06-28	Purine derivatives
NO20022738D0 (en)	2002-06-07	Pyrrolo (2,3-d) pyrimidine
MXPA03002269A (en)	2003-06-06	Purine derivatives.
MXPA03000078A (en)	2003-08-19	Purine derivatives.
AU2003292007A1 (en)	2004-06-03	4-AMINO-5-PHENYL-7-CYCLOHEXYL-PYRROLO(2,3-d)PYRIMIDINE DERIVATIVES
AU2001279700A1 (en)	2002-03-28	5-aminoalkyl-pyrazolo(4,3-d)pyrimidines with a phosphodiesterase v-inhibiting effect
PL353366A1 (en)	2003-11-17	Pyrazolo[4,3-d]pyrimidines
AU7970001A (en)	2002-01-08	5-aminoalkyl-pyrazolo(4,3-d)pyrimidines with a phosphodiesterase v-inhibiting effect
MXPA03004453A (en)	2003-08-19	Pyrimidine derivatives.
AU2001236065A1 (en)	2001-09-12	Antiviral compounds
AU2002215979A1 (en)	2002-06-03	Use of pyrazolo(4,3-D)pyrimidines
AU2002216033A1 (en)	2002-06-18	Use of pyrazolo(4,3-d)pyrimidines
AU2001285785A1 (en)	2002-03-28	2-aminoalkyl-thieno[2,3-d]pyrimidines
AU8578501A (en)	2002-01-08	2-aminoalkyl-thieno(2,3-d)pyrimidines
MXPA03000504A (en)	2003-06-24	Pyrimidine derivatives.
AU2001233026A1 (en)	2001-08-07	Phosphodiesterases
AU2002210526A1 (en)	2002-06-27	Substituted 3.4-dihydro-pyrido[1,2-A]pyrimidines
PL361915A1 (en)	2004-10-04	Substituted 3.4-dihydro-pyrido[1,2-a]pyrimidines
SI1210349T1 (en)	2003-06-30	PYRAZOLO 4,3-d)PYRIMIDINES
AUPQ806700A0 (en)	2000-07-06	Antiviral agents