AU2001278980A1 - Coumarin derivatives useful as tnfalpha inhibitors - Google Patents
Coumarin derivatives useful as tnfalpha inhibitorsInfo
- Publication number
- AU2001278980A1 AU2001278980A1 AU2001278980A AU7898001A AU2001278980A1 AU 2001278980 A1 AU2001278980 A1 AU 2001278980A1 AU 2001278980 A AU2001278980 A AU 2001278980A AU 7898001 A AU7898001 A AU 7898001A AU 2001278980 A1 AU2001278980 A1 AU 2001278980A1
- Authority
- AU
- Australia
- Prior art keywords
- derivatives useful
- coumarin derivatives
- tnfalpha inhibitors
- tnfalpha
- inhibitors
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/365—Lactones
- A61K31/366—Lactones having six-membered rings, e.g. delta-lactones
- A61K31/37—Coumarins, e.g. psoralen
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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Applications Claiming Priority (7)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US22004800P | 2000-07-21 | 2000-07-21 | |
US60220048 | 2000-07-21 | ||
US22544800P | 2000-08-14 | 2000-08-14 | |
US60225448 | 2000-08-14 | ||
US30303001P | 2001-07-03 | 2001-07-03 | |
US60303030 | 2001-07-03 | ||
PCT/US2001/022950 WO2002008217A2 (en) | 2000-07-21 | 2001-07-19 | COUMARIN DERIVATIVES USEFUL AS TNFα INHIBITORS |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2001278980A1 true AU2001278980A1 (en) | 2002-02-05 |
Family
ID=27396753
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001278980A Abandoned AU2001278980A1 (en) | 2000-07-21 | 2001-07-19 | Coumarin derivatives useful as tnfalpha inhibitors |
Country Status (4)
Country | Link |
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US (4) | US7026491B2 (en) |
JP (1) | JP4890723B2 (en) |
AU (1) | AU2001278980A1 (en) |
WO (1) | WO2002008217A2 (en) |
Families Citing this family (33)
Publication number | Priority date | Publication date | Assignee | Title |
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WO2003105842A1 (en) * | 2002-06-13 | 2003-12-24 | Novuspharma S.P.A. | Derivatives of chromen-2-one as inhibitors of vegf production in mammalian cells |
AR059339A1 (en) | 2006-02-09 | 2008-03-26 | Chugai Pharmaceutical Co Ltd | CUMARINE DERIVATIVES FOR PROLIFERATIVE DISORDERS OF CELLS, PHARMACEUTICAL COMPOSITION AND THERAPEUTIC AGENT CONTAINING THEM |
US8569378B2 (en) | 2007-07-20 | 2013-10-29 | Toshiyuki Sakai | p27 protein inducer |
JP2009084269A (en) * | 2007-09-05 | 2009-04-23 | Sumitomo Chemical Co Ltd | Coumarin compounds and their uses |
US10867298B1 (en) | 2008-10-31 | 2020-12-15 | Wells Fargo Bank, N.A. | Payment vehicle with on and off function |
US20100114768A1 (en) | 2008-10-31 | 2010-05-06 | Wachovia Corporation | Payment vehicle with on and off function |
JP5848712B2 (en) * | 2009-12-11 | 2016-01-27 | ノノ インコーポレイテッド | Agents and methods for treating ischemic diseases and other diseases |
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CH522631A (en) * | 1961-08-12 | 1972-06-30 | Cassella Farbwerke Mainkur Ag | 7-hydroxy-coumarin derivs |
US3259635A (en) * | 1962-07-26 | 1966-07-05 | Cassella Farbwerke Mainkur Ag | 7-hydroxy coumarin derivative |
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DE59010069D1 (en) * | 1989-11-21 | 1996-02-29 | Bayer Ag | Coumarin derivatives, processes for their preparation, their use and thiazolyl acetic acid derivatives as intermediates |
GB9109645D0 (en) | 1991-05-03 | 1991-06-26 | Celltech Ltd | Recombinant antibodies |
WO1996031206A2 (en) * | 1995-04-07 | 1996-10-10 | Warner-Lambert Company | Flavones and coumarins as agents for the treatment of atherosclerosis |
BR9813216A (en) | 1997-09-24 | 2000-08-29 | Orion Corp | Biesters of 1-oxa, aza and tianaftalen-2-ones as phospholamban inhibitors |
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- 2001-07-19 WO PCT/US2001/022950 patent/WO2002008217A2/en active Application Filing
- 2001-07-19 JP JP2002514123A patent/JP4890723B2/en not_active Expired - Lifetime
- 2001-07-19 AU AU2001278980A patent/AU2001278980A1/en not_active Abandoned
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2005
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WO2002008217A3 (en) | 2002-04-18 |
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WO2002008217A2 (en) | 2002-01-31 |
US20100174076A1 (en) | 2010-07-08 |
US20050014705A1 (en) | 2005-01-20 |
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