AU2001227757A1 - Inhibitors of prenyl-protein transferase - Google Patents
Inhibitors of prenyl-protein transferaseInfo
- Publication number
- AU2001227757A1 AU2001227757A1 AU2001227757A AU2775701A AU2001227757A1 AU 2001227757 A1 AU2001227757 A1 AU 2001227757A1 AU 2001227757 A AU2001227757 A AU 2001227757A AU 2775701 A AU2775701 A AU 2775701A AU 2001227757 A1 AU2001227757 A1 AU 2001227757A1
- Authority
- AU
- Australia
- Prior art keywords
- prenyl
- inhibitors
- protein transferase
- transferase
- protein
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D515/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D515/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
- C07D515/18—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17570300P | 2000-01-12 | 2000-01-12 | |
| US60175703 | 2000-01-12 | ||
| PCT/US2001/000635 WO2001051128A1 (en) | 2000-01-12 | 2001-01-09 | Inhibitors of prenyl-protein transferase |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2001227757A1 true AU2001227757A1 (en) | 2001-07-24 |
Family
ID=22641289
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001227757A Abandoned AU2001227757A1 (en) | 2000-01-12 | 2001-01-09 | Inhibitors of prenyl-protein transferase |
Country Status (3)
| Country | Link |
|---|---|
| US (1) | US6350755B1 (en) |
| AU (1) | AU2001227757A1 (en) |
| WO (1) | WO2001051128A1 (en) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2001077116A1 (en) * | 2000-04-10 | 2001-10-18 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferase |
| ATE457995T1 (en) | 2003-06-18 | 2010-03-15 | Tranzyme Pharma Inc | MACROCYCLIC MOTILIN RECEPTOR ANTAGONISTS |
| TW200944530A (en) * | 2008-04-09 | 2009-11-01 | Gruenenthal Chemie | Substituted sulfonamide derivatives |
| CA2938311C (en) | 2014-02-03 | 2023-03-07 | Vitae Pharmaceuticals, Inc. | Dihydropyrrolopyridine inhibitors of ror-gamma |
| CN112245565A (en) * | 2014-09-24 | 2021-01-22 | 艾瑞朗医疗公司 | Peptidomimetic macrocycles and uses thereof |
| JP6564029B2 (en) | 2014-10-14 | 2019-08-21 | ヴァイティー ファーマシューティカルズ，エルエルシー | Dihydropyrrolopyridine inhibitors of ROR-gamma |
| US9845308B2 (en) | 2014-11-05 | 2017-12-19 | Vitae Pharmaceuticals, Inc. | Isoindoline inhibitors of ROR-gamma |
| US9663515B2 (en) | 2014-11-05 | 2017-05-30 | Vitae Pharmaceuticals, Inc. | Dihydropyrrolopyridine inhibitors of ROR-gamma |
| DK3331876T3 (en) | 2015-08-05 | 2021-01-11 | Vitae Pharmaceuticals Llc | MODULATORS OF ROR-GAMMA |
| BR112018010018A2 (en) | 2015-11-20 | 2018-11-21 | Vitae Pharmaceuticals Inc | ror-gamma modulators |
| TW202220968A (en) | 2016-01-29 | 2022-06-01 | 美商維它藥物有限責任公司 | Modulators of ror-gamma |
| US9481674B1 (en) | 2016-06-10 | 2016-11-01 | Vitae Pharmaceuticals, Inc. | Dihydropyrrolopyridine inhibitors of ROR-gamma |
| WO2019018975A1 (en) | 2017-07-24 | 2019-01-31 | Vitae Pharmaceuticals, Inc. | Inhibitors of ror gamma |
| KR20200053481A (en) | 2017-07-24 | 2020-05-18 | 비타이 파마슈티컬즈, 엘엘씨 | Inhibitors of RORγ |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5719148A (en) | 1993-10-15 | 1998-02-17 | Schering Corporation | Tricyclic amide and urea compounds useful for inhibition of g-protein function and for treatment of proliferative diseases |
| US5721236A (en) | 1993-10-15 | 1998-02-24 | Schering Corporation | Tricyclic carbamate compounds useful for inhibition of G-protein function and for treatment of proliferative diseases |
| US5891872A (en) | 1995-04-07 | 1999-04-06 | Schering Corporation | Tricyclic compounds |
| US5712280A (en) | 1995-04-07 | 1998-01-27 | Schering Corporation | Tricyclic compounds useful for inhibition of G-protein function and for treatment of proliferative diseases |
| US5801175A (en) | 1995-04-07 | 1998-09-01 | Schering Corporation | Tricyclic compounds useful for inhibition of G-protein function and for treatment of proliferative diseases |
| US5756528A (en) | 1995-06-06 | 1998-05-26 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| US6090948A (en) | 1996-01-30 | 2000-07-18 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| US5981562A (en) | 1996-01-30 | 1999-11-09 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| US6028201A (en) | 1996-01-30 | 2000-02-22 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| US5968965A (en) | 1996-01-30 | 1999-10-19 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| US5922883A (en) | 1996-04-03 | 1999-07-13 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| US5780488A (en) | 1996-04-03 | 1998-07-14 | Merck & Co., Inc. | Inhibitors of farnesyl-protein transferase |
| AU5196698A (en) | 1996-09-13 | 1998-04-02 | Schering Corporation | Compounds useful for inhibition of farnesyl protein transferase |
| WO2000001382A1 (en) | 1998-07-02 | 2000-01-13 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferase |
| AU754554B2 (en) | 1998-07-02 | 2002-11-21 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferase |
| AU760028B2 (en) * | 1998-07-02 | 2003-05-08 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferase |
-
2001
- 2001-01-09 WO PCT/US2001/000635 patent/WO2001051128A1/en active Application Filing
- 2001-01-09 US US09/757,218 patent/US6350755B1/en not_active Expired - Fee Related
- 2001-01-09 AU AU2001227757A patent/AU2001227757A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2001051128A1 (en) | 2001-07-19 |
| US6350755B1 (en) | 2002-02-26 |
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