AU1123088A - Enantiomers of absolute configurations of amide derivatives of 3-aminoquinuclidine, the process for preparing them and their application in therapy - Google Patents
Enantiomers of absolute configurations of amide derivatives of 3-aminoquinuclidine, the process for preparing them and their application in therapyInfo
- Publication number
- AU1123088A AU1123088A AU11230/88A AU1123088A AU1123088A AU 1123088 A AU1123088 A AU 1123088A AU 11230/88 A AU11230/88 A AU 11230/88A AU 1123088 A AU1123088 A AU 1123088A AU 1123088 A AU1123088 A AU 1123088A
- Authority
- AU
- Australia
- Prior art keywords
- aminoquinuclidine
- enantiomers
- therapy
- preparing
- application
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- HBAQYPYDRFILMT-UHFFFAOYSA-N 8-[3-(1-cyclopropylpyrazol-4-yl)-1H-pyrazolo[4,3-d]pyrimidin-5-yl]-3-methyl-3,8-diazabicyclo[3.2.1]octan-2-one Chemical class C1(CC1)N1N=CC(=C1)C1=NNC2=C1N=C(N=C2)N1C2C(N(CC1CC2)C)=O HBAQYPYDRFILMT-UHFFFAOYSA-N 0.000 title 1
- -1 amide derivatives of 3-aminoquinuclidine Chemical class 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 238000002560 therapeutic procedure Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR8701355 | 1987-02-04 | ||
FR8701355A FR2610323B1 (en) | 1987-02-04 | 1987-02-04 | ENANTIOMERS OF ABSOLUTE CONFIGURATION OF AMINO-3 QUINUCLIDINE AMIDE DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR THERAPEUTIC APPLICATION |
Publications (2)
Publication Number | Publication Date |
---|---|
AU1123088A true AU1123088A (en) | 1988-08-11 |
AU619731B2 AU619731B2 (en) | 1992-02-06 |
Family
ID=9347585
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU11230/88A Ceased AU619731B2 (en) | 1987-02-04 | 1988-02-03 | Enantiomers of absolute configurations of amide derivatives of 3-aminoquinuclidine, the process for preparing them and their application in therapy |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP0280603A1 (en) |
JP (1) | JPH0681754B2 (en) |
AU (1) | AU619731B2 (en) |
DE (1) | DE280603T1 (en) |
ES (1) | ES2009718A4 (en) |
FR (1) | FR2610323B1 (en) |
ZA (1) | ZA88723B (en) |
Cited By (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU618027B2 (en) * | 1987-10-16 | 1991-12-12 | A.H. Robins Company, Incorporated | Anxiolytic-r-n-(1-azabicyclo(2.2.2)oct-3-yl) benzamides and thiobenzamides |
US5360820A (en) * | 1991-09-20 | 1994-11-01 | Glaxo Group Limited | Medical use for tachykinin antagonists |
US5547964A (en) * | 1993-03-19 | 1996-08-20 | Glaxo Group Limited | Medical use for tachykinin antagonists |
US7043496B2 (en) | 2000-11-10 | 2006-05-09 | Masae Yanagi | Data managing method, data managing system, data managing apparatus, data handling apparatus, computer program, and recording medium |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5126343A (en) * | 1989-09-11 | 1992-06-30 | G. D. Searle & Co. | N-azabicyclo [3.3.0]octane amides of aromatic acids |
NO168529C (en) * | 1989-09-15 | 1992-03-04 | Chiron Lab As | PROCEDURE FOR THE PREPARATION OF S - (-) AND R - (+) - N- (QUINUCLIDINYL-3) AMIDES. |
US5290938A (en) * | 1989-09-15 | 1994-03-01 | Chiron Laboratories A.S. | Preparation of S-(-)- and R-(+)-N-(quinuclidinyl-3)-amide |
IN187238B (en) * | 1995-06-30 | 2002-03-09 | Astra Ab |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2529548A1 (en) * | 1982-07-02 | 1984-01-06 | Delalande Sa | NOVEL DERIVATIVES OF AMINO-3 QUINUCLIDINE, THEIR PROCESS AND THEIR THERAPEUTIC APPLICATION |
US4593034A (en) * | 1984-04-06 | 1986-06-03 | A. H. Robins Company, Inc. | 2-alkoxy-N-(1-azabicyclo[2.2.2]oct-3-yl)benzamides and thiobenzamides |
US4870181A (en) * | 1985-02-04 | 1989-09-26 | A. H. Robins Company, Incorporated | Process for the preparation of 2-alkoxy-N-(1-azabicyclo[2.2.2])octan-3-yl)aminobenzamides |
JPS63146850A (en) * | 1986-11-12 | 1988-06-18 | メルク エンド カムパニー インコーポレーテツド | Renin inhibitor having phenylalanyl-histidine substitute component |
GB8629962D0 (en) * | 1986-12-16 | 1987-01-28 | Naylor R J | Benzamides & thiobenzamides |
-
1987
- 1987-02-04 FR FR8701355A patent/FR2610323B1/en not_active Expired
-
1988
- 1988-02-02 ZA ZA88723A patent/ZA88723B/en unknown
- 1988-02-03 DE DE198888400253T patent/DE280603T1/en active Pending
- 1988-02-03 EP EP88400253A patent/EP0280603A1/en not_active Withdrawn
- 1988-02-03 ES ES88400253T patent/ES2009718A4/en active Pending
- 1988-02-03 AU AU11230/88A patent/AU619731B2/en not_active Ceased
- 1988-02-04 JP JP63022969A patent/JPH0681754B2/en not_active Expired - Lifetime
Cited By (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU618027B2 (en) * | 1987-10-16 | 1991-12-12 | A.H. Robins Company, Incorporated | Anxiolytic-r-n-(1-azabicyclo(2.2.2)oct-3-yl) benzamides and thiobenzamides |
US5360820A (en) * | 1991-09-20 | 1994-11-01 | Glaxo Group Limited | Medical use for tachykinin antagonists |
US5538982A (en) * | 1991-09-20 | 1996-07-23 | Glaxo Group Limited | Medical use for tachykinin antagonists |
US5798363A (en) * | 1991-09-20 | 1998-08-25 | Glaxo Group Limited | Use for tachykinin antagonists to treat emesis |
US7214692B2 (en) | 1991-09-20 | 2007-05-08 | Glaxo Group Limited | Medical use for tachykinin antagonists |
US7342028B2 (en) | 1991-09-20 | 2008-03-11 | Glaxo Group Limited | Medical use for tachykinin antagonists |
US5547964A (en) * | 1993-03-19 | 1996-08-20 | Glaxo Group Limited | Medical use for tachykinin antagonists |
US6329394B1 (en) | 1993-03-19 | 2001-12-11 | Glaxo Group Limited | Medical use for tachykinin antagonists |
US7043496B2 (en) | 2000-11-10 | 2006-05-09 | Masae Yanagi | Data managing method, data managing system, data managing apparatus, data handling apparatus, computer program, and recording medium |
Also Published As
Publication number | Publication date |
---|---|
ES2009718A4 (en) | 1989-10-16 |
FR2610323B1 (en) | 1989-06-23 |
FR2610323A1 (en) | 1988-08-05 |
EP0280603A1 (en) | 1988-08-31 |
JPS63196583A (en) | 1988-08-15 |
ZA88723B (en) | 1988-10-26 |
JPH0681754B2 (en) | 1994-10-19 |
DE280603T1 (en) | 1989-10-05 |
AU619731B2 (en) | 1992-02-06 |
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