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ATE402173T1 - Stereoselektive synthese bestimmter trifluormethylsubstituierter alkohole - Google Patents

Stereoselektive synthese bestimmter trifluormethylsubstituierter alkohole

Info

Publication number
ATE402173T1
ATE402173T1 AT05724524T AT05724524T ATE402173T1 AT E402173 T1 ATE402173 T1 AT E402173T1 AT 05724524 T AT05724524 T AT 05724524T AT 05724524 T AT05724524 T AT 05724524T AT E402173 T1 ATE402173 T1 AT E402173T1
Authority
AT
Austria
Prior art keywords
stereoselective synthesis
substituted alcohols
sup
trifluoromethyl
certain trifluoromethyl
Prior art date
Application number
AT05724524T
Other languages
English (en)
Inventor
Jinhua J Song
Zhulin Tan
Nathan K Yee
Chris Hugh Senanayake
Jinghua Xu
Fabrice Gallou
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Application granted granted Critical
Publication of ATE402173T1 publication Critical patent/ATE402173T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT05724524T 2004-03-18 2005-03-04 Stereoselektive synthese bestimmter trifluormethylsubstituierter alkohole ATE402173T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US55426604P 2004-03-18 2004-03-18

Publications (1)

Publication Number Publication Date
ATE402173T1 true ATE402173T1 (de) 2008-08-15

Family

ID=34962572

Family Applications (1)

Application Number Title Priority Date Filing Date
AT05724524T ATE402173T1 (de) 2004-03-18 2005-03-04 Stereoselektive synthese bestimmter trifluormethylsubstituierter alkohole

Country Status (8)

Country Link
US (1) US7179919B2 (de)
EP (1) EP1727818B1 (de)
JP (1) JP4672720B2 (de)
AT (1) ATE402173T1 (de)
CA (1) CA2557896A1 (de)
DE (1) DE602005008402D1 (de)
ES (1) ES2310815T3 (de)
WO (1) WO2005090343A1 (de)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4324480B2 (ja) * 2002-03-26 2009-09-02 ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド グルココルチコイドミメティクス、その製法、医薬組成物、及び使用
AU2003255259A1 (en) * 2002-08-29 2004-03-19 Boehringer Ingelheim Pharmaceuticals, Inc. -3 (sulfonamidoethyl) -indole derivatives for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative diseases
UY28526A1 (es) * 2003-09-24 2005-04-29 Boehringer Ingelheim Pharma Miméticos de glucocorticoides, métodos de preparación composiciones farmacéuticas y usos de los mismos
US7638515B2 (en) 2003-10-08 2009-12-29 Bayer Schering Pharma Aktiengesellschaft Tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents
US7662821B2 (en) 2003-10-08 2010-02-16 Bayer Schering Pharma Ag Tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents
RS20060250A (en) 2003-10-08 2008-08-07 Schering Aktiengesellschaft, 1-amino-2-oxy-substituted tetrahydronaphtalene derivatives, method for the production thereof, and their use as antiphlogistics
US7795272B2 (en) * 2004-03-13 2010-09-14 Boehringer Ingelheim Pharmaceutical, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof
US20080153859A1 (en) 2004-04-05 2008-06-26 Hartmut Rehwinkel Multiply-substituted tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents
DE102004055633A1 (de) * 2004-11-12 2006-05-18 Schering Ag 5-substituierte Chinolin- und Isochinolin-Derivate, ein Verfahren zu ihrer Herstellung und ihre Verwendung als Entzündungshemmer
US7417056B2 (en) 2004-11-12 2008-08-26 Schering Ag 5-substituted quinoline and isoquinoline derivatives, a process for their production and their use as anti-inflammatory agents
CA2592514A1 (en) * 2004-12-27 2006-07-06 Boehringer Ingelheim Pharmaceuticals, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
ES2333820T3 (es) * 2005-09-30 2010-03-01 Boehringer Ingelheim International Gmbh Sintesis estereoselectiva de determinados alcoholes trifluorometilo-sustituidos.
EP1834948A1 (de) 2006-03-15 2007-09-19 Bayer Schering Pharma Aktiengesellschaft Tetrahydronaphthalinderivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Entzündungshemmer
WO2008070507A2 (en) * 2006-12-06 2008-06-12 Boehringer Ingelheim International Gmbh Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
MX2010013095A (es) * 2008-06-06 2010-12-21 Boehringer Ingelheim Int Mimeticos de glucocorticoides, metodos para su fabricacion, composiciones farmaceuticas y usos de los mismos.
US20110130567A1 (en) * 2009-06-03 2011-06-02 Boehringer Ingelheim International Gmbh Steroselective synthesis of certain trifluoromethyl-substituted alcohols
SG11202109435YA (en) * 2019-02-06 2021-09-29 Air Liquide Compound and method for producing lithium-containing film

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4324480B2 (ja) 2002-03-26 2009-09-02 ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド グルココルチコイドミメティクス、その製法、医薬組成物、及び使用

Also Published As

Publication number Publication date
WO2005090343A1 (en) 2005-09-29
EP1727818B1 (de) 2008-07-23
CA2557896A1 (en) 2005-09-29
DE602005008402D1 (de) 2008-09-04
EP1727818A1 (de) 2006-12-06
JP4672720B2 (ja) 2011-04-20
US20050209488A1 (en) 2005-09-22
ES2310815T3 (es) 2009-01-16
US7179919B2 (en) 2007-02-20
JP2007529520A (ja) 2007-10-25

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