ATE399779T1 - Zwischenprodukte für die herstellung von neuraminidase-inhibitor-konjugaten - Google Patents
Zwischenprodukte für die herstellung von neuraminidase-inhibitor-konjugatenInfo
- Publication number
- ATE399779T1 ATE399779T1 AT02759906T AT02759906T ATE399779T1 AT E399779 T1 ATE399779 T1 AT E399779T1 AT 02759906 T AT02759906 T AT 02759906T AT 02759906 T AT02759906 T AT 02759906T AT E399779 T1 ATE399779 T1 AT E399779T1
- Authority
- AT
- Austria
- Prior art keywords
- sub
- neuraminidase
- production
- intermediate products
- inhibitor conjugates
- Prior art date
Links
- 229940123424 Neuraminidase inhibitor Drugs 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 239000002911 sialidase inhibitor Substances 0.000 title abstract 2
- 239000013067 intermediate product Substances 0.000 title 1
- 150000000180 1,2-diols Chemical class 0.000 abstract 1
- 125000006242 amine protecting group Chemical group 0.000 abstract 1
- 125000006244 carboxylic acid protecting group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 125000006239 protecting group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pulmonology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrane Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AUPR757401 | 2001-09-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE399779T1 true ATE399779T1 (de) | 2008-07-15 |
Family
ID=3831510
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT02759906T ATE399779T1 (de) | 2001-09-07 | 2002-08-30 | Zwischenprodukte für die herstellung von neuraminidase-inhibitor-konjugaten |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US7230114B2 (de) |
| EP (1) | EP1423385B1 (de) |
| JP (1) | JP4463553B2 (de) |
| AT (1) | ATE399779T1 (de) |
| BR (1) | BR0212261A (de) |
| CA (1) | CA2456239C (de) |
| DE (1) | DE60227386D1 (de) |
| DK (1) | DK1423385T3 (de) |
| ES (1) | ES2307776T3 (de) |
| MX (1) | MXPA04002141A (de) |
| PT (1) | PT1423385E (de) |
| WO (1) | WO2003022841A1 (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN111018901B (zh) * | 2013-09-09 | 2021-09-03 | 中国科学院上海有机化学研究所 | 扎那米韦和拉那米韦的中间体及其合成方法 |
| CN113461631B (zh) * | 2021-06-29 | 2022-10-14 | 上海应用技术大学 | 一种1,3,4-恶二唑类神经氨酸酶抑制剂及其制备方法与应用 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9516276D0 (en) * | 1995-08-08 | 1995-10-11 | Biota Scient Management | Chemical compounds |
| EP0885391B1 (de) | 1996-03-01 | 2003-04-23 | Biota Scientific Management Pty. Ltd. | Verfahren zum nachweis von influenza-virus und dazu verwendbare verbindungen |
| ES2198002T3 (es) * | 1996-08-13 | 2004-01-16 | Sankyo Company, Limited | Compuestos de acido neuraminico. |
| AUPR001000A0 (en) * | 2000-09-08 | 2000-10-05 | Biota Scientific Management Pty Ltd | Novel chemical compounds and their use |
-
2002
- 2002-08-30 US US10/488,791 patent/US7230114B2/en not_active Expired - Fee Related
- 2002-08-30 AT AT02759906T patent/ATE399779T1/de not_active IP Right Cessation
- 2002-08-30 WO PCT/AU2002/001187 patent/WO2003022841A1/en active IP Right Grant
- 2002-08-30 DE DE60227386T patent/DE60227386D1/de not_active Expired - Lifetime
- 2002-08-30 JP JP2003526916A patent/JP4463553B2/ja not_active Expired - Fee Related
- 2002-08-30 ES ES02759906T patent/ES2307776T3/es not_active Expired - Lifetime
- 2002-08-30 DK DK02759906T patent/DK1423385T3/da active
- 2002-08-30 MX MXPA04002141A patent/MXPA04002141A/es active IP Right Grant
- 2002-08-30 PT PT02759906T patent/PT1423385E/pt unknown
- 2002-08-30 BR BR0212261-8A patent/BR0212261A/pt not_active IP Right Cessation
- 2002-08-30 EP EP02759906A patent/EP1423385B1/de not_active Expired - Lifetime
- 2002-08-30 CA CA2456239A patent/CA2456239C/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| PT1423385E (pt) | 2008-09-24 |
| CA2456239C (en) | 2010-11-30 |
| ES2307776T3 (es) | 2008-12-01 |
| JP4463553B2 (ja) | 2010-05-19 |
| US20050032853A1 (en) | 2005-02-10 |
| EP1423385A4 (de) | 2004-12-01 |
| MXPA04002141A (es) | 2004-07-23 |
| WO2003022841A1 (en) | 2003-03-20 |
| BR0212261A (pt) | 2004-10-19 |
| DE60227386D1 (de) | 2008-08-14 |
| DK1423385T3 (da) | 2008-11-03 |
| EP1423385A1 (de) | 2004-06-02 |
| US7230114B2 (en) | 2007-06-12 |
| CA2456239A1 (en) | 2003-03-20 |
| EP1423385B1 (de) | 2008-07-02 |
| JP2005501921A (ja) | 2005-01-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |