ATE338044T1 - Herstellung von 1h-imidazoc4,5-c)chinolin-4- aminen ber 1h-imidazoc4,5-c)chinolin-4- phthalimidzwischenprodukte - Google Patents

Herstellung von 1h-imidazoc4,5-c)chinolin-4- aminen ber 1h-imidazoc4,5-c)chinolin-4- phthalimidzwischenprodukte

Info

Publication number: ATE338044T1
Authority: AT; Austria
Prior art keywords: quinoline; imidazoc4; production; intermediate products; amines via
Prior art date: 2002-07-23

Application number

AT03766003T

Other languages

English (en)

Inventor

Valeriano Merli

Silvia Mantovani

Stefano Bianchi

Original Assignee

Teva Gyogyszergyar Zartkoeruen

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-07-23

Filing date

2003-07-23

Publication date

2006-09-15

2003-07-23 Application filed by Teva Gyogyszergyar Zartkoeruen filed Critical Teva Gyogyszergyar Zartkoeruen

2006-09-15 Application granted granted Critical

2006-09-15 Publication of ATE338044T1 publication Critical patent/ATE338044T1/de

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Virology (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

AT03766003T 2002-07-23 2003-07-23 Herstellung von 1h-imidazoc4,5-c)chinolin-4- aminen ber 1h-imidazoc4,5-c)chinolin-4- phthalimidzwischenprodukte ATE338044T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US39760702P	2002-07-23	2002-07-23

Publications (1)

Publication Number	Publication Date
ATE338044T1 true ATE338044T1 (de)	2006-09-15

Family

ID=30771087

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT03766003T ATE338044T1 (de)	2002-07-23	2003-07-23	Herstellung von 1h-imidazoc4,5-c)chinolin-4- aminen ber 1h-imidazoc4,5-c)chinolin-4- phthalimidzwischenprodukte

Country Status (17)

Country	Link
US (3)	US6852861B2 (de)
EP (1)	EP1543002B1 (de)
JP (1)	JP2006502121A (de)
KR (1)	KR20050028047A (de)
CN (1)	CN1315828C (de)
AT (1)	ATE338044T1 (de)
AU (1)	AU2003259226A1 (de)
CA (1)	CA2493227A1 (de)
DE (1)	DE60308040T2 (de)
DK (1)	DK1543002T3 (de)
ES (1)	ES2271650T3 (de)
HR (1)	HRP20050159A2 (de)
IL (1)	IL166309A (de)
MX (1)	MXPA05000893A (de)
PL (1)	PL374884A1 (de)
PT (1)	PT1543002E (de)
WO (1)	WO2004009593A1 (de)

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KR20060120069A (ko)	2003-10-03	2006-11-24	쓰리엠 이노베이티브 프로퍼티즈 컴파니	피라졸로피리딘 및 그의 유사체
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CN1906192A (zh)	2003-11-14	2007-01-31	3M创新有限公司	羟胺取代的咪唑环化合物
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US8691837B2 (en)	2003-11-25	2014-04-08	3M Innovative Properties Company	Substituted imidazo ring systems and methods
JP2007513170A (ja) *	2003-12-04	2007-05-24	スリーエムイノベイティブプロパティズカンパニー	スルホン置換イミダゾ環エーテル
JP2007517035A (ja) *	2003-12-29	2007-06-28	スリーエムイノベイティブプロパティズカンパニー	アリールアルケニルおよびアリールアルキニル置換されたイミダゾキノリン
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AU2004312508A1 (en) *	2003-12-30	2005-07-21	3M Innovative Properties Company	Imidazoquinolinyl, imidazopyridinyl, and imidazonaphthyridinyl sulfonamides
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US20090270443A1 (en) *	2004-09-02	2009-10-29	Doris Stoermer	1-amino imidazo-containing compounds and methods
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EP1804583A4 (de) *	2004-10-08	2009-05-20	3M Innovative Properties Co	Adjuvans für dna-impfstoffe
JP2008523076A (ja) *	2004-12-08	2008-07-03	スリーエムイノベイティブプロパティズカンパニー	免疫調節性の組成物、合剤、および方法
AU2004326103A1 (en) *	2004-12-27	2006-07-06	Usv Limited	A process for preparation of 4-Amino-1-isobutyl-1H-imidazo[4,5-c]-quinoline (Imiquimod)
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US8436176B2 (en) *	2004-12-30	2013-05-07	Medicis Pharmaceutical Corporation	Process for preparing 2-methyl-1-(2-methylpropyl)-1H-imidazo[4,5-c][1,5]naphthyridin-4-amine
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JP2008526751A (ja) *	2004-12-30	2008-07-24	武田薬品工業株式会社	１−（２−メチルプロピル）−１ｈ−イミダゾ［４，５−ｃ］［１，５］ナフチリジン−４−アミンエタンスルホナート及び１−（２−メチルプロピル）−１ｈ−イミダゾ［４，５−ｃ］［１，５］ナフチリジン−４−アミンメタンスルホナート
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EP1850849A2 (de) *	2005-02-23	2007-11-07	Coley Pharmaceutical Group, Inc.	Verfahren zur vorzugsweisen herbeiführung der biosynthese von interferon
US8178677B2 (en) *	2005-02-23	2012-05-15	3M Innovative Properties Company	Hydroxyalkyl substituted imidazoquinolines
WO2006091568A2 (en)	2005-02-23	2006-08-31	Coley Pharmaceutical Group, Inc.	Hydroxyalkyl substituted imidazonaphthyridines
JP2008531567A (ja) *	2005-02-23	2008-08-14	コーリーファーマシューティカルグループ，インコーポレイテッド	ヒドロキシアルキル置換イミダゾキノリン化合物および方法
WO2006107851A1 (en)	2005-04-01	2006-10-12	Coley Pharmaceutical Group, Inc.	1-substituted pyrazolo (3,4-c) ring compounds as modulators of cytokine biosynthesis for the treatment of viral infections and neoplastic diseases
EP1869043A2 (de)	2005-04-01	2007-12-26	Coley Pharmaceutical Group, Inc.	Pyrazolopyridin-1,4-diamine und analoge davon
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US8476292B2 (en) *	2005-09-09	2013-07-02	3M Innovative Properties Company	Amide and carbamate derivatives of N-{2-[4-amino-2-(ethoxymethyl)-1H-imidazo[4,5-c] quinolin-1-Yl]-1,1-dimethylethyl}methanesulfonamide and methods
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CN103582496B (zh)	2011-06-03	2016-05-11	3M创新有限公司	具有聚乙二醇链段的异双官能连接基以及由其制成的免疫应答调节剂缀合物
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2003
- 2003-07-23 PL PL03374884A patent/PL374884A1/xx unknown
- 2003-07-23 DE DE60308040T patent/DE60308040T2/de not_active Expired - Fee Related
- 2003-07-23 JP JP2004523380A patent/JP2006502121A/ja active Pending
- 2003-07-23 CN CNB038219174A patent/CN1315828C/zh not_active Expired - Fee Related
- 2003-07-23 WO PCT/US2003/023153 patent/WO2004009593A1/en active IP Right Grant
- 2003-07-23 AU AU2003259226A patent/AU2003259226A1/en not_active Abandoned
- 2003-07-23 CA CA002493227A patent/CA2493227A1/en not_active Abandoned
- 2003-07-23 AT AT03766003T patent/ATE338044T1/de not_active IP Right Cessation
- 2003-07-23 HR HR20050159A patent/HRP20050159A2/hr not_active Application Discontinuation
- 2003-07-23 MX MXPA05000893A patent/MXPA05000893A/es unknown
- 2003-07-23 EP EP03766003A patent/EP1543002B1/de not_active Expired - Lifetime
- 2003-07-23 DK DK03766003T patent/DK1543002T3/da active
- 2003-07-23 ES ES03766003T patent/ES2271650T3/es not_active Expired - Lifetime
- 2003-07-23 PT PT03766003T patent/PT1543002E/pt unknown
- 2003-07-23 US US10/626,036 patent/US6852861B2/en not_active Expired - Fee Related
- 2003-07-23 KR KR1020057001185A patent/KR20050028047A/ko not_active Ceased
2004
- 2004-12-23 US US11/023,021 patent/US7153967B2/en not_active Expired - Fee Related
2005
- 2005-01-14 IL IL166309A patent/IL166309A/en not_active IP Right Cessation
2006
- 2006-11-15 US US11/600,673 patent/US20070060755A1/en not_active Abandoned

Also Published As

Publication number	Publication date
US20050113404A1 (en)	2005-05-26
EP1543002B1 (de)	2006-08-30
CN1681814A (zh)	2005-10-12
JP2006502121A (ja)	2006-01-19
ES2271650T3 (es)	2007-04-16
US7153967B2 (en)	2006-12-26
PL374884A1 (en)	2005-11-14
HRP20050159A2 (en)	2005-08-31
AU2003259226A1 (en)	2004-02-09
KR20050028047A (ko)	2005-03-21
IL166309A0 (en)	2006-01-15
WO2004009593A1 (en)	2004-01-29
DK1543002T3 (da)	2006-12-27
MXPA05000893A (es)	2005-09-30
CN1315828C (zh)	2007-05-16
DE60308040D1 (de)	2006-10-12
EP1543002A1 (de)	2005-06-22
US20040138459A1 (en)	2004-07-15
DE60308040T2 (de)	2007-04-19
US6852861B2 (en)	2005-02-08
IL166309A (en)	2010-04-15
PT1543002E (pt)	2006-11-30
CA2493227A1 (en)	2004-01-29
US20070060755A1 (en)	2007-03-15

Publication	Publication Date	Title
ATE338044T1 (de)	2006-09-15	Herstellung von 1h-imidazoc4,5-c)chinolin-4- aminen ber 1h-imidazoc4,5-c)chinolin-4- phthalimidzwischenprodukte
PL378168A1 (pl)	2006-03-06	Dihydropterydynony, sposoby ich wytwarzania i ich zastosowanie w postaci leków
WO2003104473A8 (de)	2004-04-08	Galactosyl-isomalt, verfahren zu seiner herstellung und verwendung
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MXPA03010322A (es)	2004-02-17	PROCEDIMIENTO PARA LA PREPARACIoN DE POLIISOCIANATOS.
HRP20080057T3 (en)	2008-02-29	9,10-alpha,alpha-oh-taxane analogs and methods for production thereof
IL165558A0 (en)	2006-01-15	N-benzoylureidocinnamate derivatives method for production and use thereof
HRP20051005A2 (en)	2006-09-30	Process for the preparation of nonpeptide substituted spirobenzoazepine derivatives
DE60106057D1 (de)	2004-11-04	Verfahren zur herstellung von baccatin iii-derivativen
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