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ATE280167T1 - INTERMEDIATE PRODUCTS AND A METHOD FOR PRODUCING BETA3 ADRENERGIC RECEPTOR AGONISTS - Google Patents

INTERMEDIATE PRODUCTS AND A METHOD FOR PRODUCING BETA3 ADRENERGIC RECEPTOR AGONISTS

Info

Publication number
ATE280167T1
ATE280167T1 AT00305987T AT00305987T ATE280167T1 AT E280167 T1 ATE280167 T1 AT E280167T1 AT 00305987 T AT00305987 T AT 00305987T AT 00305987 T AT00305987 T AT 00305987T AT E280167 T1 ATE280167 T1 AT E280167T1
Authority
AT
Austria
Prior art keywords
producing
receptor agonists
adrenergic receptor
intermediate products
beta3 adrenergic
Prior art date
Application number
AT00305987T
Other languages
German (de)
Inventor
Robert William Scott
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Application granted granted Critical
Publication of ATE280167T1 publication Critical patent/ATE280167T1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/73—Unsubstituted amino or imino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

A process is provided for preparing a compound of the formula: <CHEM> comprising deprotecting a compound of the formula <CHEM>
AT00305987T 1999-07-23 2000-07-14 INTERMEDIATE PRODUCTS AND A METHOD FOR PRODUCING BETA3 ADRENERGIC RECEPTOR AGONISTS ATE280167T1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US14541799P 1999-07-23 1999-07-23

Publications (1)

Publication Number Publication Date
ATE280167T1 true ATE280167T1 (en) 2004-11-15

Family

ID=22513018

Family Applications (1)

Application Number Title Priority Date Filing Date
AT00305987T ATE280167T1 (en) 1999-07-23 2000-07-14 INTERMEDIATE PRODUCTS AND A METHOD FOR PRODUCING BETA3 ADRENERGIC RECEPTOR AGONISTS

Country Status (6)

Country Link
US (2) US6297382B1 (en)
EP (1) EP1078924B1 (en)
JP (1) JP2001048864A (en)
AT (1) ATE280167T1 (en)
DE (1) DE60015036T2 (en)
ES (1) ES2228413T3 (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2471646A1 (en) 2002-02-27 2003-09-04 Yong Tao Processes and intermediates useful in preparing .beta.3-adrenergic receptor agonists
AU2003209527A1 (en) * 2002-02-27 2003-09-09 Pfizer Products Inc. Crystal forms of (r)-2-(2-(4-oxazol-4-yl-phenoxy)-ethylamino)-1-pyridin-3-yl-ethanol
US6864268B2 (en) 2002-02-27 2005-03-08 Pfizer Inc. β3 adrenergic receptor agonists
EP1424079A1 (en) * 2002-11-27 2004-06-02 Boehringer Ingelheim International GmbH Combination of a beta-3-receptor agonist and of a reuptake inhibitor of serotonin and/or norepinephrine
US7323462B2 (en) * 2002-12-10 2008-01-29 Pfizer Inc. Morpholine dopamine agonists
US7375100B2 (en) 2003-06-04 2008-05-20 Pfizer Inc 2-amino-pyridine derivatives useful for the treatment of diseases
GB0312832D0 (en) * 2003-06-04 2003-07-09 Pfizer Ltd 2-amino-pyridine derivatives useful for the treatment of diseases
US20050113318A1 (en) * 2003-07-31 2005-05-26 Robinson Cynthia B. Combination of dehydroepiandrosterone or dehydroepiandrosterone-sulfate with a beta-agonist bronchodilator for treatment of asthma or chronic obstructive pulmonary disease
US20050026884A1 (en) * 2003-07-31 2005-02-03 Robinson Cynthia B. Combination of dehydroepiandrosterone or dehydroepiandrosterone-sulfate with a beta-agonist bronchodilator for treatment of asthma or chronic obstructive pulmonary disease
US20090285900A1 (en) * 2003-07-31 2009-11-19 Robinson Cynthia B Combination of dehydroepiandrosterone or dehydroepiandrosterone-sulfate with a beta-agonist bronchodilator for treatment of asthma or chronic obstructive pulmonary disease
JP2008512470A (en) * 2004-09-10 2008-04-24 セラヴァンス， インコーポレーテッド Amidine-substituted arylaniline compounds

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5019578A (en) 1987-11-27 1991-05-28 Merck & Co., Inc. β-adrenergic agonists
US5030640A (en) 1989-01-05 1991-07-09 Merck & Co., Inc. Novel β-adrenergic agonists and pharmaceutical compositions thereof
US5977124A (en) 1995-05-10 1999-11-02 Pfizer Inc. β-adrenergic agonists
AR003509A1 (en) 1995-09-15 1998-08-05 Merck & Co Inc SYNTHESIS OF ALPHA-CHLORINE OR FLUORINE KETONES.
TR199901063T2 (en) * 1996-11-14 1999-08-23 Pfizer Inc. Process for substituted pyridines.
AU751015B2 (en) * 1997-12-19 2002-08-08 Bayer Corporation Novel sulfonamide substituted chroman derivatives useful as beta-3 adrenoreceptor agonists
US6090942A (en) * 1998-10-15 2000-07-18 Pfizer Inc. Process and intermediates for a β3 -adrenergic receptor agonist

Also Published As

Publication number Publication date
US6441181B1 (en) 2002-08-27
JP2001048864A (en) 2001-02-20
DE60015036T2 (en) 2006-03-02
EP1078924A1 (en) 2001-02-28
US20020045757A1 (en) 2002-04-18
EP1078924B1 (en) 2004-10-20
ES2228413T3 (en) 2005-04-16
US6297382B1 (en) 2001-10-02
DE60015036D1 (en) 2004-11-25

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Legal Events

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