ATE170187T1 - Pyrrolothienopyrazin-verbindungen als 5ht3- rezeptoren-antagonisten - Google Patents

Pyrrolothienopyrazin-verbindungen als 5ht3- rezeptoren-antagonisten

Info

Publication number: ATE170187T1
Authority: AT; Austria
Prior art keywords: compounds; pyrrolothienopyrazine; receptor antagonists; medicaments; image
Prior art date: 1992-06-05

Application number

AT93401416T

Other languages

English (en)

Inventor

Sylvain Rault

Jean-Charles Lancelot

Vincente Juan-Carlos Pilo

Max Robba

Beatrice Guardiola-Lemaitre

Pierre Renard

Gerard Adam

Original Assignee

Adir

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1992-06-05

Filing date

1993-06-03

Publication date

1998-09-15

1993-06-03 Application filed by Adir filed Critical Adir

1998-09-15 Application granted granted Critical

1998-09-15 Publication of ATE170187T1 publication Critical patent/ATE170187T1/de

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Animal Behavior & Ethology (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Neurology (AREA)
General Health & Medical Sciences (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Hospice & Palliative Care (AREA)
Anesthesiology (AREA)
Otolaryngology (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

AT93401416T 1992-06-05 1993-06-03 Pyrrolothienopyrazin-verbindungen als 5ht3- rezeptoren-antagonisten ATE170187T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR9206800A FR2691967B1 (fr)	1992-06-05	1992-06-05	Nouveaux composes pyrrolothienopyraziniques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent.

Publications (1)

Publication Number	Publication Date
ATE170187T1 true ATE170187T1 (de)	1998-09-15

Family

ID=9430449

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT93401416T ATE170187T1 (de)	1992-06-05	1993-06-03	Pyrrolothienopyrazin-verbindungen als 5ht3- rezeptoren-antagonisten

Country Status (11)

Country	Link
EP (1)	EP0573360B1 (de)
JP (1)	JPH0794460B2 (de)
AT (1)	ATE170187T1 (de)
AU (1)	AU659738B2 (de)
CA (1)	CA2097779A1 (de)
DE (1)	DE69320542T2 (de)
DK (1)	DK0573360T3 (de)
ES (1)	ES2123038T3 (de)
FR (1)	FR2691967B1 (de)
NZ (1)	NZ247791A (de)
ZA (1)	ZA933942B (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US10040802B2 (en)	2015-03-12	2018-08-07	Merck Sharp & Dohme Corp.	Thienopyrazine inhibitors of IRAK4 activity

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4997433A (en) *	1990-01-16	1991-03-05	Marlowe Goble E	Endosteal fixation stud and system
FR2659332B1 (fr) *	1990-03-08	1994-04-29	Adit Et Cie	Nouvelles pyrrolo [1,2-a] thieno [3,2-f] diazepines [1,4], leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
FR2660310B1 (fr) *	1990-03-27	1992-06-05	Adir	Nouveaux derives de la 4h-pyrrolo[1,2a] thieno[2,3-f] diazepine[1,4], leur procede de preparation et les compositions pharmaceutiques les renfermant.

1992
- 1992-06-05 FR FR9206800A patent/FR2691967B1/fr not_active Expired - Fee Related
1993
- 1993-06-03 DK DK93401416T patent/DK0573360T3/da active
- 1993-06-03 DE DE69320542T patent/DE69320542T2/de not_active Expired - Fee Related
- 1993-06-03 ES ES93401416T patent/ES2123038T3/es not_active Expired - Lifetime
- 1993-06-03 AT AT93401416T patent/ATE170187T1/de not_active IP Right Cessation
- 1993-06-03 EP EP93401416A patent/EP0573360B1/de not_active Expired - Lifetime
- 1993-06-04 NZ NZ247791A patent/NZ247791A/en unknown
- 1993-06-04 ZA ZA933942A patent/ZA933942B/xx unknown
- 1993-06-04 AU AU40059/93A patent/AU659738B2/en not_active Ceased
- 1993-06-04 CA CA002097779A patent/CA2097779A1/fr not_active Abandoned
- 1993-06-04 JP JP5134922A patent/JPH0794460B2/ja not_active Expired - Lifetime

Also Published As

Publication number	Publication date
JPH06172363A (ja)	1994-06-21
NZ247791A (en)	1994-12-22
AU659738B2 (en)	1995-05-25
FR2691967A1 (fr)	1993-12-10
JPH0794460B2 (ja)	1995-10-11
CA2097779A1 (fr)	1993-12-06
DE69320542T2 (de)	1999-04-29
EP0573360B1 (de)	1998-08-26
FR2691967B1 (fr)	1995-06-09
DE69320542D1 (de)	1998-10-01
DK0573360T3 (da)	1999-05-25
EP0573360A1 (de)	1993-12-08
AU4005993A (en)	1993-12-09
ZA933942B (en)	1993-12-30
ES2123038T3 (es)	1999-01-01

Publication	Publication Date	Title
ES2081187T3 (es)	1996-02-16	Nuevas naftil-alquil-aminas, su procedimiento de preparacion y composiciones farmaceuticas que las contienen.
DK0580502T3 (da)	1999-05-31	3-(hydroxybenzylidenyl)-indolin-2-oner og farmaceutiske sammensætninger indeholdende disse
DE69318238D1 (de)	1998-06-04	Benzopyran-Verbindungen, Verfahren zu ihrer Herstellung und ihre Verwendung als Zellenschutzmittel
NO870199D0 (no)	1987-01-16	Alalogifremgangsmaate for fremstilling av nye, terapeutisk virksomme dihydrobenzofuran- og chroman-carboxamidderivater.
ES2077473T3 (es)	1995-11-16	Nuevos compuestos tiocromanicos, su procedimiento de preparacion y composiciones farmaceuticas que los contienen.
DE69320542D1 (de)	1998-10-01	Pyrrolothienopyrazin-Verbindungen als 5HT3-Rezeptoren-Antagonisten
ES2123728T3 (es)	1999-01-16	Derivados de pirrolo-pirazina de actividad 5-ht3.
ES2076054T3 (es)	1995-10-16	Nuevas amino-alquil-cromonas, su procedimiento de preparacion y composiciones farmaceuticas que las contienen.

Legal Events

Date	Code	Title	Description
1999-04-15	UEP	Publication of translation of european patent specification
2001-03-15	REN	Ceased due to non-payment of the annual fee