AT331970B - Verfahren zur herstellung neuer alpha- aminobenzylpenicillinderivate - Google Patents
Verfahren zur herstellung neuer alpha- aminobenzylpenicillinderivateInfo
- Publication number
- AT331970B AT331970B AT399573A AT399573A AT331970B AT 331970 B AT331970 B AT 331970B AT 399573 A AT399573 A AT 399573A AT 399573 A AT399573 A AT 399573A AT 331970 B AT331970 B AT 331970B
- Authority
- AT
- Austria
- Prior art keywords
- aminobenzylpenicillin
- derivatives
- producing new
- new alpha
- alpha
- Prior art date
Links
- AVKUERGKIZMTKX-NJBDSQKTSA-N ampicillin Chemical class C1([C@@H](N)C(=O)N[C@H]2[C@H]3SC([C@@H](N3C2=O)C(O)=O)(C)C)=CC=CC=C1 AVKUERGKIZMTKX-NJBDSQKTSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
- C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
- C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
- C07D499/68—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with aromatic rings as additional substituents on the carbon chain
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP4511872A JPS5547036B2 (de) | 1972-05-08 | 1972-05-08 | |
| JP8342472A JPS4941396A (de) | 1972-08-21 | 1972-08-21 | |
| JP8510272A JPS4942692A (de) | 1972-08-25 | 1972-08-25 | |
| JP8510372A JPS4942693A (de) | 1972-08-25 | 1972-08-25 | |
| JP12595272A JPS4981388A (de) | 1972-12-15 | 1972-12-15 | |
| JP1991773A JPS49108092A (de) | 1973-02-18 | 1973-02-18 | |
| JP3813273A JPS49125386A (de) | 1973-04-04 | 1973-04-04 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ATA399573A ATA399573A (de) | 1975-12-15 |
| AT331970B true AT331970B (de) | 1975-12-15 |
Family
ID=27563884
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT399573A AT331970B (de) | 1972-05-08 | 1973-05-07 | Verfahren zur herstellung neuer alpha- aminobenzylpenicillinderivate |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US3953428A (de) |
| AR (2) | AR204813A1 (de) |
| AT (1) | AT331970B (de) |
| BE (1) | BE799202A (de) |
| CA (1) | CA1050971A (de) |
| DE (1) | DE2322750A1 (de) |
| DK (1) | DK139754B (de) |
| FI (1) | FI58131C (de) |
| FR (1) | FR2183895B1 (de) |
| GB (1) | GB1407566A (de) |
Families Citing this family (28)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4202900A (en) * | 1972-09-27 | 1980-05-13 | Ciba-Geigy Corporation | Derivatives of penam-3-carboxylic acid and a pharmaceutical composition containing the same |
| JPS5751837B2 (de) * | 1973-04-05 | 1982-11-04 | ||
| US3994874A (en) * | 1973-11-07 | 1976-11-30 | Richardson-Merrell Inc. | 6-[(2-Oxo-1-pyridinyl)acylamino]penicillin derivatives |
| US3954734A (en) * | 1974-01-21 | 1976-05-04 | Parke, Davis & Company | Novel antibacterial amide compounds and process means for producing the same |
| IL47168A (en) * | 1974-05-09 | 1979-07-25 | Toyama Chemical Co Ltd | Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the same |
| US3989687A (en) * | 1974-09-27 | 1976-11-02 | Richardson-Merrell Inc. | 4-Oxo-1-pyridinyl penicillin derivatives |
| GB1568962A (en) * | 1975-10-31 | 1980-06-11 | Beecham Group Ltd | Reparation and compositions containing them (heterocyclic-carbonylamino)pencillins methods for their p |
| NZ184434A (en) * | 1976-06-30 | 1979-03-28 | Dainippon Pharmaceutical Co | Penicillins with a substituted p-hydroxy-benzyl side-chain, and injectable pharmaceutical compositions |
| GB1579362A (en) * | 1977-03-16 | 1980-11-19 | Beecham Group Ltd | 6-(a-heterocyclylcarbonyl amino-acetamido)-penicillins and compositions containing them |
| EP0001041A3 (de) * | 1977-07-27 | 1979-06-27 | Sandoz Ag | Alpha(Pyridonecarboxylamino)Alpha-acetamid-substituierte Penicilline und Cephalosporine, Verfahren zu ihrer Herstellung, ihre Verwendung als Arzneimittel; Pyridone für ihre Herstellung |
| GB2010250B (en) * | 1977-12-06 | 1982-07-14 | Nippon Chemiphar Co | Penicillin and cephalosporin derivatives and a process for producing the same |
| US4231928A (en) * | 1979-04-24 | 1980-11-04 | Bristol-Myers Company | Antibacterial agents |
| JPS5651488A (en) * | 1979-10-02 | 1981-05-09 | Meiji Seika Kaisha Ltd | Penicillin derivative and its preparation |
| US5281612A (en) * | 1982-09-09 | 1994-01-25 | Warner-Lambert Company | Naphthyridine antibacterial agents |
| IE55898B1 (en) * | 1982-09-09 | 1991-02-14 | Warner Lambert Co | Antibacterial agents |
| IT1215277B (it) * | 1985-05-27 | 1990-01-31 | Pomezia Roma A | Derivato chinolin-lattaminico ad attivita' antibatterica ed inibitrice delle b-lattamasi. |
| US5273973A (en) * | 1988-10-24 | 1993-12-28 | Norwich Eaton Pharmaceuticals, Inc. | Antimicrobial quinolonyl esters |
| US5328908A (en) * | 1988-10-24 | 1994-07-12 | Procter & Gamble Pharmaceuticals, Inc. | Antimicrobial quinolone thioureas |
| CA2001203C (en) * | 1988-10-24 | 2001-02-13 | Thomas P. Demuth, Jr. | Novel antimicrobial dithiocarbamoyl quinolones |
| EP0997466A1 (de) * | 1988-10-24 | 2000-05-03 | PROCTER & GAMBLE PHARMACEUTICALS, INC. | Antimikrobielle Laktamchinolone |
| US5491139A (en) * | 1988-10-24 | 1996-02-13 | The Procter & Gamble Company | Antimicrobial quinolonyl lactams |
| US5180719A (en) * | 1988-10-24 | 1993-01-19 | Norwich Eaton Pharmaceuticals, Inc. | Antimicrobial quinolonyl lactam esters |
| ES2147721T3 (es) * | 1990-04-18 | 2000-10-01 | Procter & Gamble Pharma | Quinolonil lactamas antimicrobianas. |
| FR2713637B1 (fr) * | 1993-12-15 | 1996-01-05 | Cird Galderma | Nouveaux composés bi-aromatiques dérivés d'amide, compositions pharmaceutiques et cosmétiques les contenant et utilisations. |
| US6143760A (en) | 1997-08-25 | 2000-11-07 | Neurogen Corporation | Substituted 4-oxo-napthyridine-3-carboxamides: GABA brain receptor ligands |
| PL338783A1 (en) * | 1997-08-25 | 2000-11-20 | Neurogen Corp | Substituted 4-oxo-naphtyridin-3-carboxamides as ligands of cerebral gaba receptors |
| US7939558B2 (en) * | 2004-06-04 | 2011-05-10 | The Regents Of The University Of California | Compounds having activity in increasing ion transport by mutant-CFTR and uses thereof |
| US8669370B2 (en) | 2011-01-26 | 2014-03-11 | Sanofi | Substituted 3-heteroaroylamino-propionic acid derivatives and their use as pharmaceuticals |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1180745A (en) * | 1966-10-04 | 1970-02-11 | Beecham Group Ltd | Penicillins |
| US3668198A (en) * | 1970-06-01 | 1972-06-06 | Squibb & Sons Inc | {60 -ureido-2,4,6-cycloheptatrienylmethylpenicillins |
| US3711471A (en) * | 1971-02-03 | 1973-01-16 | Bristol Myers Co | Purification of 6-{8 d-{60 -(3-guanyl-1-ureido)phenylacetamido{9 {0 penicillanic acid |
-
1973
- 1973-01-01 AR ARJA247904A patent/AR204813A1/es active
- 1973-01-01 AR AR251189A patent/AR204162A1/es active
- 1973-04-30 CA CA169,846A patent/CA1050971A/en not_active Expired
- 1973-05-01 US US05/356,120 patent/US3953428A/en not_active Expired - Lifetime
- 1973-05-05 DE DE2322750A patent/DE2322750A1/de not_active Withdrawn
- 1973-05-07 AT AT399573A patent/AT331970B/de not_active IP Right Cessation
- 1973-05-07 BE BE130836A patent/BE799202A/xx unknown
- 1973-05-07 DK DK248973AA patent/DK139754B/da not_active IP Right Cessation
- 1973-05-07 FI FI1458/73A patent/FI58131C/fi active
- 1973-05-08 GB GB2195173A patent/GB1407566A/en not_active Expired
- 1973-05-08 FR FR7316416A patent/FR2183895B1/fr not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| CA1050971A (en) | 1979-03-20 |
| ATA399573A (de) | 1975-12-15 |
| DE2322750A1 (de) | 1973-11-29 |
| FI58131B (fi) | 1980-08-29 |
| GB1407566A (en) | 1975-09-24 |
| AU5504573A (en) | 1974-11-07 |
| AR204162A1 (es) | 1975-11-28 |
| DK139754C (de) | 1979-09-24 |
| US3953428A (en) | 1976-04-27 |
| FI58131C (fi) | 1980-12-10 |
| AR204813A1 (es) | 1976-03-05 |
| DK139754B (da) | 1979-04-09 |
| FR2183895B1 (de) | 1976-07-02 |
| BE799202A (fr) | 1973-08-31 |
| FR2183895A1 (de) | 1973-12-21 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ELA | Expired due to lapse of time | ||
| ELJ | Ceased due to non-payment of the annual fee |