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AR219173A1 - Procedimiento para la preparacion de 4-(2-hidroxi-3-(amino)propoxi)-2-bencimidazolinonas - Google Patents

Procedimiento para la preparacion de 4-(2-hidroxi-3-(amino)propoxi)-2-bencimidazolinonas

Info

Publication number
AR219173A1
AR219173A1 AR277226A AR27722679A AR219173A1 AR 219173 A1 AR219173 A1 AR 219173A1 AR 277226 A AR277226 A AR 277226A AR 27722679 A AR27722679 A AR 27722679A AR 219173 A1 AR219173 A1 AR 219173A1
Authority
AR
Argentina
Prior art keywords
benzmidazolinones
propoxi
hydroxy
amino
procedure
Prior art date
Application number
AR277226A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB18438/77A external-priority patent/GB1595316A/en
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of AR219173A1 publication Critical patent/AR219173A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D303/00Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02Compounds containing oxirane rings
    • C07D303/12Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
    • C07D303/18Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by etherified hydroxyl radicals
    • C07D303/20Ethers with hydroxy compounds containing no oxirane rings
    • C07D303/22Ethers with hydroxy compounds containing no oxirane rings with monohydroxy compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/28Sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
AR277226A 1977-05-03 1979-07-06 Procedimiento para la preparacion de 4-(2-hidroxi-3-(amino)propoxi)-2-bencimidazolinonas AR219173A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB18438/77A GB1595316A (en) 1977-05-03 1977-05-03 4-(3-amino-2-hydroxy-propoxy)-benzimidazole derivatives and pharmaceutical compositions containing them
GB4915677 1977-11-25
GB220878 1978-01-19

Publications (1)

Publication Number Publication Date
AR219173A1 true AR219173A1 (es) 1980-07-31

Family

ID=27254036

Family Applications (2)

Application Number Title Priority Date Filing Date
AR272019A AR220335A1 (es) 1977-05-03 1978-05-31 Procedimiento para la preparacion de 4(2-hidroxi-3-(amino)-propoxi)-2-benzimidazolinonas y-tionas y compuestos para su exclusivo uso como intermediarios en dicho procedimiento
AR277226A AR219173A1 (es) 1977-05-03 1979-07-06 Procedimiento para la preparacion de 4-(2-hidroxi-3-(amino)propoxi)-2-bencimidazolinonas

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AR272019A AR220335A1 (es) 1977-05-03 1978-05-31 Procedimiento para la preparacion de 4(2-hidroxi-3-(amino)-propoxi)-2-benzimidazolinonas y-tionas y compuestos para su exclusivo uso como intermediarios en dicho procedimiento

Country Status (18)

Country Link
JP (1) JPS53135979A (es)
AR (2) AR220335A1 (es)
AU (1) AU3569678A (es)
DE (1) DE2819458A1 (es)
DK (1) DK190378A (es)
ES (1) ES469353A1 (es)
FI (1) FI781349A (es)
FR (1) FR2399414A1 (es)
GR (1) GR73669B (es)
IL (1) IL54591A0 (es)
IT (1) IT1096276B (es)
LU (1) LU79591A1 (es)
MC (1) MC1192A1 (es)
NL (1) NL7804794A (es)
NO (1) NO781556L (es)
NZ (1) NZ187066A (es)
PT (1) PT67980A (es)
SE (1) SE7805140L (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2801980A1 (de) * 1978-01-18 1979-07-19 Boehringer Mannheim Gmbh 4-hydroxy-2-benzimidazolin-thion- derivate, verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel
EP0003758A1 (de) * 1978-02-09 1979-09-05 Ciba-Geigy Ag Verätherte Hydroxy-benzodiheterocyclen und ihre Säureadditionssalze, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Präparate
DE2905877A1 (de) * 1979-02-16 1980-08-28 Boehringer Mannheim Gmbh Neue aminopropanolderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
CH661501A5 (fr) * 1982-01-26 1987-07-31 Oreal Composes derivant du amino-3 propanol-2 utilisables pour la teinture des cheveux, leur procede de preparation, composition de teinture les contenant et procede de teinture de cheveux correspondant.
DE3839743A1 (de) * 1988-11-25 1990-05-31 Hoechst Ag Verfahren zur herstellung von benzimidazolonen
US9784726B2 (en) 2013-01-08 2017-10-10 Atrogi Ab Screening method, a kit, a method of treatment and a compound for use in a method of treatment
GB201714736D0 (en) 2017-09-13 2017-10-25 Atrogi Ab New compounds and uses
GB201714734D0 (en) 2017-09-13 2017-10-25 Atrogi Ab New compounds and uses
GB201714740D0 (en) 2017-09-13 2017-10-25 Atrogi Ab New compounds and uses
GB201714745D0 (en) 2017-09-13 2017-10-25 Atrogi Ab New compounds and uses
GB202205895D0 (en) 2022-04-22 2022-06-08 Atrogi Ab New medical uses

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1058822A (en) * 1963-07-30 1967-02-15 Ici Ltd 3-amino-2-hydroxypropoxy heterocyclic derivatives
GB1363735A (en) * 1970-10-23 1974-08-14 Hoechst Ag Process for the manufacture of benzimidazolones
US4081447A (en) * 1975-04-09 1978-03-28 Abbott Laboratories 5-[2-Hydroxy-3-(3,4-dimethoxy phenethylamino)]-propoxy-3,4-dihydro carbostyril and pharmaceutically acceptable salts thereof
CH624395A5 (es) * 1976-01-08 1981-07-31 Ciba Geigy Ag

Also Published As

Publication number Publication date
DK190378A (da) 1978-11-04
JPS53135979A (en) 1978-11-28
ES469353A1 (es) 1980-01-01
FI781349A (fi) 1978-11-04
MC1192A1 (fr) 1979-02-23
IL54591A0 (en) 1978-07-31
NO781556L (no) 1978-11-06
FR2399414A1 (fr) 1979-03-02
GR73669B (es) 1984-03-28
AU3569678A (en) 1979-11-08
NZ187066A (en) 1981-02-11
DE2819458A1 (de) 1978-11-16
NL7804794A (nl) 1978-11-07
SE7805140L (sv) 1978-11-04
LU79591A1 (de) 1979-06-13
IT1096276B (it) 1985-08-26
PT67980B (es) 1980-05-05
IT7823000A0 (it) 1978-05-03
PT67980A (en) 1978-06-01
AR220335A1 (es) 1980-10-31

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