AR216496A1 - PROCEDURE FOR PREPARING N- (BENZOTHIAZOL-2-IL) -OXAMIDIC ACID DERIVATIVES - Google Patents
PROCEDURE FOR PREPARING N- (BENZOTHIAZOL-2-IL) -OXAMIDIC ACID DERIVATIVESInfo
- Publication number
- AR216496A1 AR216496A1 AR270289A AR27028977A AR216496A1 AR 216496 A1 AR216496 A1 AR 216496A1 AR 270289 A AR270289 A AR 270289A AR 27028977 A AR27028977 A AR 27028977A AR 216496 A1 AR216496 A1 AR 216496A1
- Authority
- AR
- Argentina
- Prior art keywords
- benzothiazol
- preparing
- procedure
- acid derivatives
- oxamidic acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/62—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to atoms of the carbocyclic ring
- C07D317/66—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pulmonology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19762656468 DE2656468A1 (en) | 1976-12-14 | 1976-12-14 | N- (BENZTHIAZOL-2-YL) -OXAMID ACID DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF |
Publications (1)
Publication Number | Publication Date |
---|---|
AR216496A1 true AR216496A1 (en) | 1979-12-28 |
Family
ID=5995427
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AR270289A AR216496A1 (en) | 1976-12-14 | 1977-12-07 | PROCEDURE FOR PREPARING N- (BENZOTHIAZOL-2-IL) -OXAMIDIC ACID DERIVATIVES |
Country Status (17)
Country | Link |
---|---|
JP (1) | JPS5377058A (en) |
AR (1) | AR216496A1 (en) |
AT (1) | AT360523B (en) |
AU (1) | AU510730B2 (en) |
BE (1) | BE861794A (en) |
CS (1) | CS203179B2 (en) |
DD (1) | DD133329A5 (en) |
DE (1) | DE2656468A1 (en) |
ES (1) | ES465034A1 (en) |
FI (1) | FI57594C (en) |
FR (1) | FR2374317A1 (en) |
GB (1) | GB1538822A (en) |
HU (1) | HU175340B (en) |
NL (1) | NL7713580A (en) |
SE (1) | SE7714074L (en) |
SU (1) | SU680647A3 (en) |
ZA (1) | ZA777236B (en) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2676775A (en) * | 1949-10-24 | 1954-04-27 | Gustav O Schulz | Electric flatiron cord holder |
DE3017976A1 (en) * | 1980-05-10 | 1981-11-19 | Dr. Karl Thomae Gmbh, 7950 Biberach | SUBSTITUTED 2-AMINO-5-HALOGEN-BENZOTHIAZOLES, METHOD FOR THE PRODUCTION THEREOF AND MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS |
US4321372A (en) | 1980-06-16 | 1982-03-23 | Pfizer Inc. | Antiulcer thiazol-2-ylcarbamoyl-carboxylic acids, esters and amides |
DE3027527A1 (en) | 1980-07-19 | 1982-02-18 | Basf Ag, 6700 Ludwigshafen | NEW OXAMID ACID DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND THERAPEUTIC AGENTS CONTAINING THEM |
GB2090826B (en) * | 1981-01-09 | 1985-06-12 | Usv Pharma Corp | New heterocyclic compounds useful as anti-allergie agents |
DE3135250A1 (en) * | 1981-09-05 | 1983-03-17 | Basf Ag, 6700 Ludwigshafen | TRICYCLIC THIAZOLYLOXAMATES, METHOD FOR THE PRODUCTION THEREOF AND THERAPEUTIC AGENTS CONTAINING THEM |
US4826860A (en) * | 1987-03-16 | 1989-05-02 | Warner-Lambert Company | Substituted 2-aminobenzothiazoles and derivatives useful as cerebrovascular agents |
FI91859C (en) * | 1987-06-17 | 1994-08-25 | Eisai Co Ltd | Analogue method for the preparation of an active benzothiazole derivative as an antiallergic agent |
CZ2003182A3 (en) | 2000-06-21 | 2003-06-18 | F. Hoffmann-La Roche Ag | Benzothiazole derivatives |
US7087761B2 (en) | 2003-01-07 | 2006-08-08 | Hoffmann-La Roche Inc. | Cyclization process for substituted benzothiazole derivatives |
PT1753760E (en) | 2004-05-24 | 2008-02-12 | Hoffmann La Roche | 4-hydroxy-4-methyl-piperidine-1-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-amide |
JP4633123B2 (en) | 2004-11-05 | 2011-02-16 | エフ.ホフマン−ラ ロシュ アーゲー | Method for producing isonicotinic acid derivative |
EP1863818B1 (en) | 2005-03-23 | 2010-03-10 | F.Hoffmann-La Roche Ag | Acetylenyl-pyrazolo-pvrimidine derivatives as mglur2 antagonists |
ES2340321T3 (en) | 2005-09-27 | 2010-06-01 | F.Hoffmann-La Roche Ag | OXADIAZOLILPIRAZOLO-PIRIMIDINAS, AS ANGLGIST OF MGLUR2. |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4150140A (en) * | 1976-12-23 | 1979-04-17 | The Upjohn Company | Benzothiazolyl oxanic acids, esters and salts |
-
1976
- 1976-12-14 DE DE19762656468 patent/DE2656468A1/en not_active Withdrawn
-
1977
- 1977-12-03 HU HU77BO1695A patent/HU175340B/en unknown
- 1977-12-05 ZA ZA00777236A patent/ZA777236B/en unknown
- 1977-12-07 SU SU772550552A patent/SU680647A3/en active
- 1977-12-07 AR AR270289A patent/AR216496A1/en active
- 1977-12-07 GB GB50911/77A patent/GB1538822A/en not_active Expired
- 1977-12-07 CS CS778173A patent/CS203179B2/en unknown
- 1977-12-08 DD DD7700202483A patent/DD133329A5/en unknown
- 1977-12-08 AU AU31377/77A patent/AU510730B2/en not_active Expired
- 1977-12-08 NL NL7713580A patent/NL7713580A/en not_active Application Discontinuation
- 1977-12-12 SE SE7714074A patent/SE7714074L/en not_active Application Discontinuation
- 1977-12-12 FI FI773738A patent/FI57594C/en not_active IP Right Cessation
- 1977-12-13 AT AT890777A patent/AT360523B/en not_active IP Right Cessation
- 1977-12-13 BE BE183407A patent/BE861794A/en unknown
- 1977-12-13 FR FR7737467A patent/FR2374317A1/en active Granted
- 1977-12-14 JP JP15041777A patent/JPS5377058A/en active Pending
- 1977-12-14 ES ES465034A patent/ES465034A1/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
AT360523B (en) | 1981-01-12 |
ES465034A1 (en) | 1978-09-01 |
GB1538822A (en) | 1979-01-24 |
FR2374317B1 (en) | 1980-11-07 |
ATA890777A (en) | 1980-06-15 |
FI57594C (en) | 1980-09-10 |
ZA777236B (en) | 1978-11-29 |
HU175340B (en) | 1980-07-28 |
DD133329A5 (en) | 1978-12-27 |
JPS5377058A (en) | 1978-07-08 |
FR2374317A1 (en) | 1978-07-13 |
FI57594B (en) | 1980-05-30 |
AU510730B2 (en) | 1980-07-10 |
SE7714074L (en) | 1978-06-15 |
SU680647A3 (en) | 1979-08-15 |
AU3137777A (en) | 1979-06-14 |
FI773738A (en) | 1978-06-15 |
DE2656468A1 (en) | 1978-06-15 |
CS203179B2 (en) | 1981-02-27 |
BE861794A (en) | 1978-06-13 |
NL7713580A (en) | 1978-06-16 |
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