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AR215666A1 - OLEANDOMYCIN DERIVATIVES, THERAPEUTICALLY RELEVANT DERIVATIVES, APPLICABLE AS INTERMEDIARIES FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE OLEANDOMYCINS; PROCEDURE FOR PREPARING SAID INTERMEDIARY DERIVATIVES; AND PROCEDURE FOR PREPARING THERAPEUTICALLY ACTIVE OLEANDOMYCIN DERIVATIVES; - Google Patents

OLEANDOMYCIN DERIVATIVES, THERAPEUTICALLY RELEVANT DERIVATIVES, APPLICABLE AS INTERMEDIARIES FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE OLEANDOMYCINS; PROCEDURE FOR PREPARING SAID INTERMEDIARY DERIVATIVES; AND PROCEDURE FOR PREPARING THERAPEUTICALLY ACTIVE OLEANDOMYCIN DERIVATIVES;

Info

Publication number
AR215666A1
AR215666A1 AR270472A AR27047277A AR215666A1 AR 215666 A1 AR215666 A1 AR 215666A1 AR 270472 A AR270472 A AR 270472A AR 27047277 A AR27047277 A AR 27047277A AR 215666 A1 AR215666 A1 AR 215666A1
Authority
AR
Argentina
Prior art keywords
derivatives
procedure
preparing
oleandomycin
therapeutically active
Prior art date
Application number
AR270472A
Other languages
Spanish (es)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of AR215666A1 publication Critical patent/AR215666A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AR270472A 1977-02-04 1977-12-22 OLEANDOMYCIN DERIVATIVES, THERAPEUTICALLY RELEVANT DERIVATIVES, APPLICABLE AS INTERMEDIARIES FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE OLEANDOMYCINS; PROCEDURE FOR PREPARING SAID INTERMEDIARY DERIVATIVES; AND PROCEDURE FOR PREPARING THERAPEUTICALLY ACTIVE OLEANDOMYCIN DERIVATIVES; AR215666A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/765,486 US4125705A (en) 1977-02-04 1977-02-04 Semi-synthetic 4-amino-oleandomycin derivatives

Publications (1)

Publication Number Publication Date
AR215666A1 true AR215666A1 (en) 1979-10-31

Family

ID=25073683

Family Applications (1)

Application Number Title Priority Date Filing Date
AR270472A AR215666A1 (en) 1977-02-04 1977-12-22 OLEANDOMYCIN DERIVATIVES, THERAPEUTICALLY RELEVANT DERIVATIVES, APPLICABLE AS INTERMEDIARIES FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE OLEANDOMYCINS; PROCEDURE FOR PREPARING SAID INTERMEDIARY DERIVATIVES; AND PROCEDURE FOR PREPARING THERAPEUTICALLY ACTIVE OLEANDOMYCIN DERIVATIVES;

Country Status (34)

Country Link
US (1) US4125705A (en)
JP (2) JPS5398981A (en)
AR (1) AR215666A1 (en)
AT (1) AT358169B (en)
AU (1) AU502293B1 (en)
BE (1) BE863618A (en)
BG (2) BG32116A3 (en)
CA (1) CA1106366A (en)
CH (1) CH629821A5 (en)
CS (3) CS200537B2 (en)
DD (1) DD134523A5 (en)
DE (1) DE2804509C2 (en)
DK (1) DK149628C (en)
ES (1) ES465322A1 (en)
FI (1) FI65262C (en)
FR (2) FR2383964A1 (en)
GB (1) GB1583921A (en)
GR (1) GR68692B (en)
HU (2) HU179744B (en)
IE (1) IE46395B1 (en)
IL (2) IL53959A0 (en)
IT (1) IT1094211B (en)
LU (1) LU79007A1 (en)
NL (1) NL175997C (en)
NO (2) NO145955C (en)
NZ (1) NZ186384A (en)
PH (2) PH14836A (en)
PL (3) PL113163B1 (en)
PT (1) PT67569B (en)
RO (3) RO79264A (en)
SE (2) SE445222B (en)
SU (3) SU805949A3 (en)
YU (3) YU39504B (en)
ZA (1) ZA78646B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4124755A (en) * 1978-01-03 1978-11-07 Pfizer Inc. 11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4133950A (en) * 1978-01-03 1979-01-09 Pfizer Inc. 4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters
US4413119A (en) * 1982-03-01 1983-11-01 Pfizer Inc. Semi-synthetic macrolides
US4363803A (en) * 1982-03-01 1982-12-14 Pfizer Inc. 3",4"-Oxyallylene erythromycin and oleandomycin, composition and method of use
JPH0240447U (en) * 1988-09-14 1990-03-19
US5141926A (en) * 1990-04-18 1992-08-25 Abbott Laboratories Erythromycin derivatives
JPH05155896A (en) * 1991-01-18 1993-06-22 Yamanouchi Pharmaceut Co Ltd New macrolide compound and its production

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3022219A (en) * 1958-03-07 1962-02-20 Pfizer & Co C Acyl esters of oleandomycin
US3179652A (en) * 1961-09-05 1965-04-20 Pfizer & Co C Antibiotic recovery process and salts produced thereby
US3836519A (en) * 1973-05-04 1974-09-17 Abbott Lab Sulfonyl derivatives of erythromycin
US3842069A (en) * 1973-06-21 1974-10-15 Abbott Lab 4"-deoxy-4"-oxoerythromycin b derivatives
US4036853A (en) * 1976-08-06 1977-07-19 Pfizer Inc. Semi-synthetic oleandomycin derivatives-C8 modifications

Also Published As

Publication number Publication date
DE2804509C2 (en) 1982-12-02
IE780240L (en) 1978-08-04
PL111160B1 (en) 1980-08-30
SU888824A3 (en) 1981-12-07
IT7820006A0 (en) 1978-02-03
PT67569B (en) 1979-06-18
RO79258A (en) 1982-06-25
PT67569A (en) 1978-02-01
BE863618A (en) 1978-08-03
JPS56135497A (en) 1981-10-22
YU39518B (en) 1984-12-31
DK149628C (en) 1987-02-02
RO79264A (en) 1982-06-25
DK51778A (en) 1978-08-05
HU179744B (en) 1982-12-28
PH16491A (en) 1983-10-28
FR2396022B1 (en) 1980-06-13
SU805949A3 (en) 1981-02-15
FI780355A (en) 1978-08-05
NO780390L (en) 1978-08-07
IE46395B1 (en) 1983-06-01
GR68692B (en) 1982-02-01
NL175997C (en) 1985-02-01
NO145955C (en) 1982-06-30
SE457085B (en) 1988-11-28
NL175997B (en) 1984-09-03
SE7800269L (en) 1978-08-05
CS200537B2 (en) 1980-09-15
FR2396022A1 (en) 1979-01-26
FI65262B (en) 1983-12-30
FR2383964B1 (en) 1981-11-27
YU151882A (en) 1982-10-31
JPS5827799B2 (en) 1983-06-11
DK149628B (en) 1986-08-18
SU1020004A3 (en) 1983-05-23
YU300377A (en) 1982-10-31
IL53959A0 (en) 1978-04-30
PL113163B1 (en) 1980-11-29
CS200538B2 (en) 1980-09-15
IL61606A0 (en) 1981-01-30
AT358169B (en) 1980-08-25
AU502293B1 (en) 1979-07-19
ES465322A1 (en) 1978-09-16
IT1094211B (en) 1985-07-26
GB1583921A (en) 1981-02-04
RO75387A (en) 1980-11-30
HU181395B (en) 1983-07-28
BG32117A4 (en) 1982-05-14
CS200536B2 (en) 1980-09-15
NO150439C (en) 1984-10-17
ATA72078A (en) 1980-01-15
JPS5398981A (en) 1978-08-29
NO811914L (en) 1978-08-07
CH629821A5 (en) 1982-05-14
US4125705A (en) 1978-11-14
NZ186384A (en) 1980-08-26
PH14836A (en) 1981-12-16
NL7801259A (en) 1978-08-08
NO150439B (en) 1984-07-09
NO145955B (en) 1982-03-22
JPS5652036B2 (en) 1981-12-09
ZA78646B (en) 1978-12-27
BG32116A3 (en) 1982-05-14
DE2804509A1 (en) 1978-08-10
PL110793B1 (en) 1980-07-31
SE445222B (en) 1986-06-09
FI65262C (en) 1984-04-10
YU151782A (en) 1982-10-31
LU79007A1 (en) 1979-09-06
YU39504B (en) 1984-12-31
DD134523A5 (en) 1979-03-07
YU39517B (en) 1984-12-31
FR2383964A1 (en) 1978-10-13
PL204041A1 (en) 1979-06-04
CA1106366A (en) 1981-08-04
SE8300869D0 (en) 1983-02-16

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