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AR077332A1 - Procesos para la alquilacion de pirazoles - Google Patents

Procesos para la alquilacion de pirazoles

Info

Publication number
AR077332A1
AR077332A1 ARP100102714A ARP100102714A AR077332A1 AR 077332 A1 AR077332 A1 AR 077332A1 AR P100102714 A ARP100102714 A AR P100102714A AR P100102714 A ARP100102714 A AR P100102714A AR 077332 A1 AR077332 A1 AR 077332A1
Authority
AR
Argentina
Prior art keywords
compound
formula
pirazoles
rental
processes
Prior art date
Application number
ARP100102714A
Other languages
English (en)
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of AR077332A1 publication Critical patent/AR077332A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Steroid Compounds (AREA)

Abstract

Reivindicacion 1: Un proceso para la preparacion de un compuesto de la formula (1) donde R1 es haloalquilo C1-4; R2 es alquilo opcionalmente sustituido, arilo opcionalmente sustituido o heteroarilo opcionalmente sustituido; y R3 es metilo o etilo; donde un compuesto de la formula (2) donde R1 y R2 son tales como se definieron para el compuesto de la formula (1); se hace reaccionar con un compuesto de la formula (3) donde R3 es tal como se definio para el compuesto de la formula (1).
ARP100102714A 2009-07-31 2010-07-27 Procesos para la alquilacion de pirazoles AR077332A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23013409P 2009-07-31 2009-07-31
US36157010P 2010-07-06 2010-07-06

Publications (1)

Publication Number Publication Date
AR077332A1 true AR077332A1 (es) 2011-08-17

Family

ID=42782270

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP100102714A AR077332A1 (es) 2009-07-31 2010-07-27 Procesos para la alquilacion de pirazoles

Country Status (12)

Country Link
US (1) US8563747B2 (es)
EP (1) EP2459538B1 (es)
JP (1) JP5956334B2 (es)
CN (1) CN102471279A (es)
AR (1) AR077332A1 (es)
BR (1) BR112012008128B8 (es)
DK (1) DK2459538T3 (es)
ES (1) ES2525489T3 (es)
IL (1) IL217387A (es)
MX (1) MX2012001067A (es)
TW (1) TW201107296A (es)
WO (1) WO2011012620A2 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW201105636A (en) 2009-07-28 2011-02-16 Syngenta Participations Ag Processes relating to the alkylation of pyrazoles
PT2603494T (pt) * 2010-08-10 2017-02-03 Syngenta Participations Ag Processo para a preparação de 3-haloalquilopirazóis
JP5140776B1 (ja) * 2012-09-05 2013-02-13 タマ化学工業株式会社 １−置換−３−フルオロアルキルピラゾール−４−カルボン酸エステルの製造方法
JP6676038B2 (ja) 2014-08-19 2020-04-08 バイエル・アニマル・ヘルス・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ａｎｉｍａｌ Ｈｅａｌｔｈ Ｇｍｂｈ ヘキサフルオロプロペンから出発する５−フルオロ−１ｈ−ピラゾール類の調製のための方法

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0759560B2 (ja) * 1987-10-19 1995-06-28 三井東圧化学株式会社 １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法
GB9405229D0 (en) * 1994-03-17 1994-04-27 Rhone Poulenc Agriculture Compositions of matter
US5498624A (en) * 1995-05-03 1996-03-12 Monsanto Company Selected pyrazolyl derivatives
JP2000044541A (ja) 1998-08-03 2000-02-15 Mitsui Chemicals Inc １，３−ジアルキルピラゾール−４−カルボン酸エステルの製造法
JP4568404B2 (ja) 2000-05-17 2010-10-27 三井化学アグロ株式会社 ピラゾールカルボン酸エステル誘導体の製造法
EP1829865A3 (en) 2002-03-05 2007-09-19 Syngeta Participations AG O-Cyclopropyl-carboxanilides and their use as fungicides
GB0224316D0 (en) 2002-10-18 2002-11-27 Syngenta Participations Ag Chemical compounds
JP2008502636A (ja) * 2004-06-18 2008-01-31 ビーエーエスエフ　アクチェンゲゼルシャフト Ｎ−（オルト−フェニル）−１−メチル−３−ジフルオロメチルピラゾール−４−カルボキシアニリドおよびそれらの殺菌剤としての使用
CA2582141C (en) * 2004-10-21 2013-06-11 Harald Walter Process for the preparation of pyrazoles
EP1854788B8 (en) * 2005-02-25 2012-12-26 Sagami Chemical Research Institute Method for producing 1-substituted-3-fluoroalkyl pyrazole-4-carboxylate
SI1940813T1 (sl) * 2005-10-25 2011-02-28 Syngenta Participations Ag Heterociklični amidni derivati, uporabni kot mikrobiocidi
GB0526044D0 (en) 2005-12-21 2006-02-01 Syngenta Ltd Novel herbicides
WO2008053044A2 (de) 2006-11-03 2008-05-08 Basf Se Hetarylcarbonsäure-n-(biphen-2-yl)amid-verbindungen
KR101543705B1 (ko) 2007-03-16 2015-08-11 신젠타 리미티드 살균제의 신규한 고체 형태
CA2684563C (en) * 2007-05-11 2013-08-13 Eli Lilly And Company 2-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-3-phenyl pyrazines and pyridines and 3-[4-(pyrazol-4-ylalkyl)piperazin-1-yl]-2-phenyl pyridines as 5-ht7 receptor antagonists
US8124787B2 (en) 2007-05-31 2012-02-28 Syngenta Crop Protection, Inc. Process for the production of pyrazoles
UA103323C2 (ru) 2008-05-08 2013-10-10 Басф Се Способ получения арилкарбоксамидов
GB0812028D0 (en) 2008-07-01 2008-08-06 Syngenta Participations Ag Fungicidal compositions

Also Published As

Publication number Publication date
BR112012008128B8 (pt) 2019-07-16
IL217387A (en) 2016-02-29
WO2011012620A2 (en) 2011-02-03
ES2525489T3 (es) 2014-12-23
TW201107296A (en) 2011-03-01
US8563747B2 (en) 2013-10-22
CN102471279A (zh) 2012-05-23
BR112012008128A2 (pt) 2015-09-22
MX2012001067A (es) 2012-03-16
WO2011012620A3 (en) 2011-06-09
EP2459538A2 (en) 2012-06-06
IL217387A0 (en) 2012-02-29
JP5956334B2 (ja) 2016-07-27
BR112012008128B1 (pt) 2017-10-31
JP2013500945A (ja) 2013-01-10
US20120130085A1 (en) 2012-05-24
EP2459538B1 (en) 2014-10-15
DK2459538T3 (en) 2015-01-05

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