AR046036A1 - Composiciones de risedronato y metodos para su uso - Google Patents
Composiciones de risedronato y metodos para su usoInfo
- Publication number
- AR046036A1 AR046036A1 ARP040103537A ARP040103537A AR046036A1 AR 046036 A1 AR046036 A1 AR 046036A1 AR P040103537 A ARP040103537 A AR P040103537A AR P040103537 A ARP040103537 A AR P040103537A AR 046036 A1 AR046036 A1 AR 046036A1
- Authority
- AR
- Argentina
- Prior art keywords
- risedronate
- pharmaceutical composition
- accordance
- compositions
- methods
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/662—Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
- A61K31/663—Compounds having two or more phosphorus acid groups or esters thereof, e.g. clodronic acid, pamidronic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Physical Education & Sports Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
El uso de una composición farmacéutica para tratar o prevenir un trastorno óseo que contiene del 65 % al 110 % de la dosis efectiva acumulativa de risedronato que comprende administrar por vía oral al ser humano u otro mamífero de conformidad con un esquema de dosificación continua de uno, dos o tres días consecutivos al mes. Dicho uso en donde dicha composición farmacéutica se administra un día por mes en la forma de una dosis unitaria que comprende de 100 mg a 165 mg de risedronato, de preferencia 150 mg de risedronato. Dicho uso en donde el trastorno óseo es osteoporosis. Composición farmacéutica adecuada para administrarse de conformidad con dicho esquema de dosificación continua, dicha composición farmacéutica comprende: a) entre 65 % y 110 % de la dosis efectiva acumulativa de risedronato; y b) uno o más excipientes farmacéuticamente aceptables. Dicha composición farmacéutica en donde la forma de dosificación es una tableta.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10/897,897 US20050070504A1 (en) | 2001-12-21 | 2004-07-23 | Risedronate compositions and their methods of use |
Publications (1)
Publication Number | Publication Date |
---|---|
AR046036A1 true AR046036A1 (es) | 2005-11-23 |
Family
ID=34958880
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP040103537A AR046036A1 (es) | 2004-07-23 | 2004-09-29 | Composiciones de risedronato y metodos para su uso |
Country Status (20)
Country | Link |
---|---|
US (1) | US20050070504A1 (es) |
EP (1) | EP1776123A1 (es) |
JP (3) | JP5377852B2 (es) |
KR (2) | KR20080083219A (es) |
CN (1) | CN101146542A (es) |
AR (1) | AR046036A1 (es) |
AU (2) | AU2004322703B2 (es) |
BR (1) | BRPI0418973A (es) |
CA (1) | CA2564898A1 (es) |
IL (1) | IL180907A0 (es) |
IS (1) | IS8597A (es) |
MA (1) | MA28778B1 (es) |
MX (1) | MX2007000967A (es) |
NO (1) | NO20071058L (es) |
NZ (1) | NZ552799A (es) |
PE (1) | PE20060144A1 (es) |
RU (1) | RU2007103306A (es) |
TW (1) | TWI351286B (es) |
WO (1) | WO2006022755A1 (es) |
ZA (1) | ZA200701308B (es) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2003055496A1 (en) * | 2001-12-21 | 2003-07-10 | The Procter & Gamble Company | Method for the treatment of bone disorders |
PT1506041E (pt) * | 2002-05-10 | 2007-12-28 | Hoffmann La Roche | Ácido ibandrónico para o tratamento e a prevenção da osteoporose |
EP1790347B1 (en) * | 2002-12-20 | 2014-12-24 | F. Hoffmann-La Roche AG | High dose ibandronate formulation |
US20080287400A1 (en) * | 2004-05-24 | 2008-11-20 | Richard John Dansereau | Low Dosage Forms Of Risedronate Or Its Salts |
AU2011218625B2 (en) * | 2004-05-24 | 2014-03-20 | Theramex HQ UK Limited | Dosage forms of risedronate |
US7645459B2 (en) | 2004-05-24 | 2010-01-12 | The Procter & Gamble Company | Dosage forms of bisphosphonates |
US20080286359A1 (en) * | 2004-05-24 | 2008-11-20 | Richard John Dansereau | Low Dosage Forms Of Risedronate Or Its Salts |
US8071574B2 (en) * | 2005-02-22 | 2011-12-06 | John Dennis Bobyn | Implant improving local bone formation |
US7473684B2 (en) | 2005-09-16 | 2009-01-06 | Selamine Limited | Bisphosphonate formulation |
EP3047847A1 (en) * | 2005-10-12 | 2016-07-27 | OPKO Renal, LLC | Methods and articles for treating 25-hydroxyvitamin d insufficiency and deficiency |
GB0624090D0 (en) * | 2006-12-01 | 2007-01-10 | Selamine Ltd | Ramipril amine salts |
GB0624087D0 (en) * | 2006-12-01 | 2007-01-10 | Selamine Ltd | Ramipril combination salt |
GB0624084D0 (en) * | 2006-12-01 | 2007-01-10 | Selamine Ltd | Ramipril amino acid salts |
KR100844256B1 (ko) | 2007-03-23 | 2008-07-07 | 코오롱제약주식회사 | 리세드로네이트와 비타민 d를 포함하는 대사성 골질환치료용 약제조성물 및 이의 제조방법 |
JP2011529901A (ja) * | 2008-07-31 | 2011-12-15 | 味の素株式会社 | リセドロネートまたはその塩の低投与量形態 |
KR101379664B1 (ko) * | 2008-09-23 | 2014-04-02 | 한림제약(주) | 리세드론산 또는 그의 염 및 비타민 d를 포함하는 약학 조성물 |
KR101102364B1 (ko) | 2009-09-18 | 2012-01-03 | 한림제약(주) | 비스포스포네이트 유도체 및 고용량의 콜레칼시페롤을 포함하는 약학 조성물 |
PT106978A (pt) * | 2013-05-31 | 2014-12-02 | Tecnimede Sociedade Tecnico Medicinal S A | Composição sólida oral contendo ácido ibandrónico e vitamina d |
Family Cites Families (30)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA777769A (en) * | 1963-03-18 | 1968-02-06 | H. Roy Clarence | Substituted methylene diphosphonic acid compounds and detergent compositions |
IT1201087B (it) * | 1982-04-15 | 1989-01-27 | Gentili Ist Spa | Bifosfonati farmacologicamente attivi,procedimento per la loro preparazione e relative composizioni farmaceutiche |
FR2531088B1 (fr) * | 1982-07-29 | 1987-08-28 | Sanofi Sa | Produits anti-inflammatoires derives de l'acide methylenediphosphonique et leur procede de preparation |
IL77243A (en) * | 1984-12-21 | 1996-11-14 | Procter & Gamble | Pharmaceutical compositions containing geminal diphosphonic acid compounds and certain such novel compounds |
US4761406A (en) * | 1985-06-06 | 1988-08-02 | The Procter & Gamble Company | Regimen for treating osteoporosis |
DE3623397A1 (de) * | 1986-07-11 | 1988-01-14 | Boehringer Mannheim Gmbh | Neue diphosphonsaeurederivate, verfahren zu deren herstellung und diese verbindungen enthaltende arzneimittel |
CA1339805C (en) * | 1988-01-20 | 1998-04-07 | Yasuo Isomura | (cycloalkylamino)methylenebis(phosphonic acid) and medicines containing the same as an active |
CA1336328C (en) * | 1988-04-11 | 1995-07-18 | Walter G. Leonard | Method of increasing bone density in humans |
US4922007A (en) * | 1989-06-09 | 1990-05-01 | Merck & Co., Inc. | Process for preparing 4-amino-1-hydroxybutylidene-1,1-bisphosphonic acid or salts thereof |
US5227506A (en) * | 1989-09-06 | 1993-07-13 | Merck & Co., Inc. | Acyloxymethyl esters of bisphosphonic acids as bone resorption inhibitors |
NL8902727A (nl) * | 1989-11-06 | 1991-06-03 | Philips Nv | Objecthouder voor ondersteuning van een object in een geladen deeltjesbundelsysteem. |
WO1994000130A1 (en) * | 1992-06-30 | 1994-01-06 | Procter & Gamble Pharmaceuticals, Inc. | Compositions for the treatment of arthritis containing phosphonates and nsaids |
US5646134A (en) * | 1994-04-21 | 1997-07-08 | Merck & Co., Inc. | Alendronate therapy to prevent loosening of, or pain associated with, orthopedic implant devices |
US6008206A (en) * | 1994-09-21 | 1999-12-28 | Merck & Co., Inc. | Sodium alendronate preparation for local administration |
US6750216B2 (en) * | 1996-03-08 | 2004-06-15 | Adolor Corporation | Kappa agonist compounds and pharmaceutical formulations thereof |
US5730715A (en) * | 1996-06-14 | 1998-03-24 | Becton Dickinson And Company | Method for the iontophoretic administration of bisphosphonates |
GB2324726A (en) * | 1997-05-01 | 1998-11-04 | Merck & Co Inc | Combination Therapy for the Treatment of Osteoporosis |
DE69826660T2 (de) * | 1997-06-11 | 2005-10-06 | The Procter & Gamble Company, Cincinnati | Filmüberzogene tablette für verbesserte verträglichkeit im oberen magen-darmtrakt |
US5994329A (en) * | 1997-07-22 | 1999-11-30 | Merck & Co., Inc. | Method for inhibiting bone resorption |
US6432932B1 (en) * | 1997-07-22 | 2002-08-13 | Merck & Co., Inc. | Method for inhibiting bone resorption |
US6015801A (en) * | 1997-07-22 | 2000-01-18 | Merck & Co., Inc. | Method for inhibiting bone resorption |
US6331533B1 (en) * | 1998-11-16 | 2001-12-18 | Merck & Co., Inc. | Method for inhibiting dental resorptive lesions |
US6225801B1 (en) * | 1999-01-14 | 2001-05-01 | Lucent Technologies Inc. | Article comprising electronic circuits and devices with magnetically programmable electrical resistance |
JP2001253827A (ja) * | 2000-02-15 | 2001-09-18 | Pfizer Prod Inc | 骨粗鬆症を治療するための組成物および方法 |
US6468559B1 (en) * | 2000-04-28 | 2002-10-22 | Lipocine, Inc. | Enteric coated formulation of bishosphonic acid compounds and associated therapeutic methods |
NZ523086A (en) * | 2000-06-20 | 2007-07-27 | Novartis Ag | Method of administering bisphosphonates |
US6593310B1 (en) * | 2000-11-21 | 2003-07-15 | Arthropharm Pty. Ltd. | Treatment of osteoporosis |
EP1458400A1 (en) * | 2001-12-13 | 2004-09-22 | Merck & Co., Inc. | Liquid bisphosphonate formulations for bone disorders |
PT1506041E (pt) * | 2002-05-10 | 2007-12-28 | Hoffmann La Roche | Ácido ibandrónico para o tratamento e a prevenção da osteoporose |
US20040188316A1 (en) * | 2003-03-26 | 2004-09-30 | The Procter & Gamble Company | Kit for pharmaceutical use |
-
2004
- 2004-07-23 US US10/897,897 patent/US20050070504A1/en not_active Abandoned
- 2004-09-25 WO PCT/US2004/031975 patent/WO2006022755A1/en active Application Filing
- 2004-09-25 JP JP2007522476A patent/JP5377852B2/ja not_active Expired - Lifetime
- 2004-09-25 RU RU2007103306/14A patent/RU2007103306A/ru unknown
- 2004-09-25 CN CNA2004800436570A patent/CN101146542A/zh active Pending
- 2004-09-25 CA CA002564898A patent/CA2564898A1/en not_active Abandoned
- 2004-09-25 EP EP04789250A patent/EP1776123A1/en not_active Ceased
- 2004-09-25 KR KR1020087021196A patent/KR20080083219A/ko active Search and Examination
- 2004-09-25 MX MX2007000967A patent/MX2007000967A/es unknown
- 2004-09-25 KR KR1020077001602A patent/KR20070038115A/ko not_active Application Discontinuation
- 2004-09-25 AU AU2004322703A patent/AU2004322703B2/en not_active Withdrawn - After Issue
- 2004-09-25 BR BRPI0418973-6A patent/BRPI0418973A/pt not_active Application Discontinuation
- 2004-09-25 NZ NZ552799A patent/NZ552799A/en not_active IP Right Cessation
- 2004-09-29 AR ARP040103537A patent/AR046036A1/es unknown
- 2004-09-30 PE PE2004000960A patent/PE20060144A1/es not_active Application Discontinuation
- 2004-11-30 TW TW093136901A patent/TWI351286B/zh not_active IP Right Cessation
-
2007
- 2007-01-23 IL IL180907A patent/IL180907A0/en unknown
- 2007-01-24 IS IS8597A patent/IS8597A/is unknown
- 2007-02-01 MA MA29645A patent/MA28778B1/fr unknown
- 2007-02-14 ZA ZA200701308A patent/ZA200701308B/en unknown
- 2007-02-22 NO NO20071058A patent/NO20071058L/no not_active Application Discontinuation
-
2011
- 2011-03-02 AU AU2011200905A patent/AU2011200905A1/en not_active Abandoned
-
2013
- 2013-08-16 JP JP2013169220A patent/JP5761274B2/ja not_active Expired - Lifetime
-
2014
- 2014-10-21 JP JP2014214604A patent/JP5910698B2/ja not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
JP2015038135A (ja) | 2015-02-26 |
IS8597A (is) | 2007-01-24 |
MA28778B1 (fr) | 2007-08-01 |
JP2013231087A (ja) | 2013-11-14 |
JP5377852B2 (ja) | 2013-12-25 |
MX2007000967A (es) | 2007-07-11 |
US20050070504A1 (en) | 2005-03-31 |
AU2011200905A1 (en) | 2011-03-24 |
AU2004322703A1 (en) | 2006-03-02 |
JP5910698B2 (ja) | 2016-04-27 |
NO20071058L (no) | 2007-02-22 |
ZA200701308B (en) | 2008-07-30 |
BRPI0418973A (pt) | 2007-12-04 |
RU2007103306A (ru) | 2008-09-10 |
TWI351286B (en) | 2011-11-01 |
CN101146542A (zh) | 2008-03-19 |
NZ552799A (en) | 2010-04-30 |
PE20060144A1 (es) | 2006-04-17 |
KR20070038115A (ko) | 2007-04-09 |
WO2006022755A1 (en) | 2006-03-02 |
AU2004322703B2 (en) | 2010-12-02 |
KR20080083219A (ko) | 2008-09-16 |
JP5761274B2 (ja) | 2015-08-12 |
EP1776123A1 (en) | 2007-04-25 |
TW200603816A (en) | 2006-02-01 |
CA2564898A1 (en) | 2006-03-02 |
IL180907A0 (en) | 2007-07-04 |
JP2008507513A (ja) | 2008-03-13 |
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Legal Events
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FB | Suspension of granting procedure |