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AR018197A1 - Compuestos de piperidina, un procedimiento para su preparacion, una composicion y uso del mismo para la preparacion de un medicamento - Google Patents

Compuestos de piperidina, un procedimiento para su preparacion, una composicion y uso del mismo para la preparacion de un medicamento

Info

Publication number
AR018197A1
AR018197A1 ARP990101908A ARP990101908A AR018197A1 AR 018197 A1 AR018197 A1 AR 018197A1 AR P990101908 A ARP990101908 A AR P990101908A AR P990101908 A ARP990101908 A AR P990101908A AR 018197 A1 AR018197 A1 AR 018197A1
Authority
AR
Argentina
Prior art keywords
preparation
procedure
composition
same
piperidine compounds
Prior art date
Application number
ARP990101908A
Other languages
English (en)
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27269380&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR018197(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9814316.7A external-priority patent/GB9814316D0/en
Priority claimed from GBGB9821732.6A external-priority patent/GB9821732D0/en
Priority claimed from GBGB9902935.7A external-priority patent/GB9902935D0/en
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of AR018197A1 publication Critical patent/AR018197A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4525—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Inorganic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Addiction (AREA)
  • Child & Adolescent Psychology (AREA)
  • Obesity (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Se describen compuestos de piperidina, que comprenden metanosulfonato de 4-(4-fluorfenil)-3-(3,4-metilendioxifenoximetil)-piperidina (paroxetina),procedimientos para preparados, composiciones farmacéuticas que los contienen, y su uso para la preparacion de un medicamento en el tratamiento oprevencion de varios trastornos.
ARP990101908A 1998-07-02 1999-04-26 Compuestos de piperidina, un procedimiento para su preparacion, una composicion y uso del mismo para la preparacion de un medicamento AR018197A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9814316.7A GB9814316D0 (en) 1998-07-02 1998-07-02 Novel compounds
GBGB9821732.6A GB9821732D0 (en) 1998-10-06 1998-10-06 Novel compound
GBGB9902935.7A GB9902935D0 (en) 1999-02-10 1999-02-10 Novel compound

Publications (1)

Publication Number Publication Date
AR018197A1 true AR018197A1 (es) 2001-10-31

Family

ID=27269380

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP990101885A AR011759A1 (es) 1998-07-02 1999-04-23 Compuesto derivado de fenoximetilpiperidina, procedimientos para su preparacion, una composicion farmaceutica, el uso del mismo para la preparacion de un medicamento, para la preparacion de un producto intermedio, un solvato y un envase
ARP990101908A AR018197A1 (es) 1998-07-02 1999-04-26 Compuestos de piperidina, un procedimiento para su preparacion, una composicion y uso del mismo para la preparacion de un medicamento

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ARP990101885A AR011759A1 (es) 1998-07-02 1999-04-23 Compuesto derivado de fenoximetilpiperidina, procedimientos para su preparacion, una composicion farmaceutica, el uso del mismo para la preparacion de un medicamento, para la preparacion de un producto intermedio, un solvato y un envase

Country Status (35)

Country Link
US (4) US6063927A (es)
EP (5) EP1020464B1 (es)
JP (1) JP2002519422A (es)
KR (1) KR20010053336A (es)
CN (1) CN1127502C (es)
AR (2) AR011759A1 (es)
AT (4) ATE251155T1 (es)
AU (4) AU3619199A (es)
BE (3) BE1012403A5 (es)
BR (1) BR9911682A (es)
CA (1) CA2269999A1 (es)
CH (1) CH689805A8 (es)
DE (5) DE19918588A1 (es)
DK (7) DK199900176U3 (es)
ES (4) ES2158778B1 (es)
FI (2) FI112077B (es)
FR (2) FR2780728B1 (es)
GB (5) GB2336364B (es)
GR (3) GR990100140A (es)
HK (1) HK1037877A1 (es)
HU (1) HUP0102334A3 (es)
IE (5) IE990344A1 (es)
IL (1) IL140628A (es)
IT (1) IT1312540B1 (es)
LU (1) LU90388B1 (es)
NL (4) NL1011875C2 (es)
NO (1) NO319030B1 (es)
NZ (1) NZ509180A (es)
PL (1) PL345214A1 (es)
PT (4) PT1089996E (es)
SE (1) SE9901462A0 (es)
SI (3) SI1020464T1 (es)
SK (1) SK20262000A3 (es)
TR (1) TR200100054T2 (es)
WO (1) WO2000001694A1 (es)

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CH689805A8 (fr) * 1998-07-02 2000-02-29 Smithkline Beecham Plc Méthanesulfonate de paroxétine, procédé pour sa préparation et compositions pharmaceutiques le contenant.
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WO2000078290A2 (en) * 1999-06-22 2000-12-28 Smithkline Beecham P.L.C. Pharmaceutical composition comprising a salt of paroxetine
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NZ523902A (en) * 2000-08-28 2004-05-28 Synthon Bv Paroxetine compositions and processes for making the same
DE20100529U1 (de) * 2001-01-11 2001-05-10 Synthon Bv Pharmazeutische Tablette umfassend Paroxetinmesylat
NL1017421C2 (nl) * 2001-02-21 2002-01-15 Synthon Bv Werkwijze voor het vervaardigen van paroxetine.
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JP4625637B2 (ja) 2002-02-22 2011-02-02 シャイア エルエルシー 活性物質送達系及び活性物質を保護し投与する方法
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US20080033050A1 (en) 2006-08-04 2008-02-07 Richards Patricia Allison Tewe Method of treating thermoregulatory disfunction with paroxetine
JP2010520879A (ja) * 2007-03-09 2010-06-17 ノバルティス アーゲー ３−（１ｈ−インドール−３−イル）−４−［２−（４−メチル−ピペラジン−１−イル）−キナゾリン−４−イル］−ピロール−２，５−ジオンの塩
US8119688B2 (en) * 2007-09-19 2012-02-21 Xy, Llc Differential evaporation potentiated disinfectant system
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FR2926552B1 (fr) * 2008-01-23 2010-03-26 Biocodex Procede de preparation de particules de stiripentol ayant une granulometrie definie
CN103961333B (zh) * 2014-05-07 2020-02-21 浙江华海药业股份有限公司 甲磺酸帕罗西汀胶囊及其制备方法
CN104523645A (zh) * 2014-11-20 2015-04-22 美吉斯制药（厦门）有限公司 甲磺酸帕罗西汀片芯及其包衣片的制备方法
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DE20100529U1 (de) * 2001-01-11 2001-05-10 Synthon Bv Pharmazeutische Tablette umfassend Paroxetinmesylat

Also Published As

Publication number Publication date
GB9909505D0 (en) 1999-06-23
DE69911774D1 (de) 2003-11-06
AR011759A1 (es) 2000-09-13
DE60000003T2 (de) 2002-03-21
BR9911682A (pt) 2001-12-26
GR3034328T3 (en) 2000-12-29
GB9920332D0 (en) 1999-11-03
US20010023253A1 (en) 2001-09-20
GB0026487D0 (en) 2000-12-13
SI0970955T1 (en) 2001-02-28
IL140628A0 (en) 2002-02-10
SE9901462L (es)
DK199900554A (da) 2000-01-03
NL1012272C1 (nl) 1999-07-12
CA2269999A1 (en) 2000-01-02
EP1020464A1 (en) 2000-07-19
GR990100140A (el) 2000-03-31
GB2352395B (en) 2004-02-11
NO991944L (no) 2000-01-03
PT970955E (pt) 2000-11-30
ATE251155T1 (de) 2003-10-15
IES20000894A2 (en) 2001-05-30
SE9901462A0 (sv) 2000-01-03
SI1020464T1 (en) 2001-12-31
ES2157881T3 (es) 2001-09-01
CN1315949A (zh) 2001-10-03
PT102291A (pt) 2000-05-31
FI990922A (fi) 2000-01-03
DE29907248U1 (de) 1999-09-09
GB0119695D0 (en) 2001-10-03
GB0216752D0 (en) 2002-08-28
US6063927A (en) 2000-05-16
IL140628A (en) 2004-06-20
ES2149044T3 (es) 2000-10-16
KR20010053336A (ko) 2001-06-25
FR2780728A1 (fr) 2000-01-07
AU2392899A (en) 2000-01-20
DK1089996T3 (da) 2004-02-09
LU90388B1 (fr) 2001-01-29
NL1011875A1 (nl) 2000-01-07
IE20000633A1 (en) 2001-10-17
DK199900234U4 (da) 2000-12-22
GB2367003A (en) 2002-03-27
NL1012271A1 (nl) 1999-07-12
PT1089996E (pt) 2004-02-27
EP1089996A1 (en) 2001-04-11
DE19918588A1 (de) 2000-01-27
IES20000893A2 (en) 2001-05-30
HK1037877A1 (en) 2002-02-22
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AU713877B3 (en) 1999-12-09
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NO319030B1 (no) 2005-06-06
FI112077B (fi) 2003-10-31
ITMI990866A1 (it) 2000-10-23
IES81166B2 (en) 2000-05-31
PT1020464E (pt) 2001-10-30
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GB2336364A (en) 1999-10-20
FI990922A0 (fi) 1999-04-23
GB2377637A (en) 2003-01-22
SK20262000A3 (sk) 2001-07-10
FR2802098A1 (fr) 2001-06-15
NL1012271C2 (nl) 1999-09-23
ATE202777T1 (de) 2001-07-15
AU3619199A (en) 2000-01-24
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DK199900234U1 (da) 2000-12-22
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CH689805A8 (fr) 2000-02-29
DK199900176U3 (da) 1999-08-13
IES990343A2 (en) 2000-01-02
SE9901462D0 (sv) 1999-04-23
EP1288214A1 (en) 2003-03-05
AU732211C (en) 2004-05-06
NL1011874C1 (nl) 1999-07-12
ES2158778A1 (es) 2001-09-01
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GB2336364B (en) 2000-05-10
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JP2002519422A (ja) 2002-07-02
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AU713131B3 (en) 1999-11-25
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DE60000003D1 (de) 2001-08-09
DE69900007T2 (de) 2001-06-07
FI4209U1 (fi) 1999-11-10
BE1011664A6 (fr) 1999-11-09
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NZ509180A (en) 2001-06-29
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GB2352395A (en) 2001-01-31
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EP0970955A1 (en) 2000-01-12
WO2000001694A1 (en) 2000-01-13
US20020193406A1 (en) 2002-12-19
NL1011875C2 (nl) 2000-03-24
AT3185U2 (de) 1999-11-25
CH689805A5 (fr) 1999-11-30
SI1089996T1 (en) 2004-04-30
FR2780728B1 (fr) 2001-02-16
PL345214A1 (en) 2001-12-03
GR1003350B (el) 2000-03-29
ATE195121T1 (de) 2000-08-15
DE69900007D1 (de) 2000-09-07
PT102291B (pt) 2002-07-31
GB2339428A (en) 2000-01-26
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