ZA200202122B - Kinase inhibitors as therapeutic agents. - Google Patents
Kinase inhibitors as therapeutic agents. Download PDFInfo
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- ZA200202122B ZA200202122B ZA200202122A ZA200202122A ZA200202122B ZA 200202122 B ZA200202122 B ZA 200202122B ZA 200202122 A ZA200202122 A ZA 200202122A ZA 200202122 A ZA200202122 A ZA 200202122A ZA 200202122 B ZA200202122 B ZA 200202122B
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
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- Health & Medical Sciences (AREA)
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- Pharmacology & Pharmacy (AREA)
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Applications Claiming Priority (1)
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| US15461899P | 1999-09-17 | 1999-09-17 |
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| ZA200202122B true ZA200202122B (en) | 2003-08-27 |
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| ZA200202122A ZA200202122B (en) | 1999-09-17 | 2002-03-14 | Kinase inhibitors as therapeutic agents. |
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| EP (1) | EP1268481B1 (no) |
| JP (1) | JP2003509427A (no) |
| KR (1) | KR20020063854A (no) |
| CN (1) | CN1390220A (no) |
| AR (1) | AR029766A1 (no) |
| AT (1) | ATE380814T1 (no) |
| AU (1) | AU7491400A (no) |
| BG (1) | BG106585A (no) |
| BR (1) | BR0014075A (no) |
| CA (1) | CA2385769A1 (no) |
| CY (1) | CY1107886T1 (no) |
| CZ (1) | CZ2002934A3 (no) |
| DE (1) | DE60037455T2 (no) |
| DK (1) | DK1268481T3 (no) |
| ES (1) | ES2299434T3 (no) |
| HK (1) | HK1053831A1 (no) |
| HU (1) | HUP0303363A2 (no) |
| IL (1) | IL148719A0 (no) |
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| NO (1) | NO20021329L (no) |
| NZ (1) | NZ517759A (no) |
| PL (1) | PL354241A1 (no) |
| PT (1) | PT1268481E (no) |
| SK (1) | SK3792002A3 (no) |
| TR (1) | TR200201506T2 (no) |
| WO (1) | WO2001019828A2 (no) |
| ZA (1) | ZA200202122B (no) |
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| WO2019051199A1 (en) | 2017-09-08 | 2019-03-14 | Incyte Corporation | 6-CYANO-INDAZOLE COMPOUNDS AS HEMATOPOIETIC PROGENITOR KINASE 1 (HPK1) MODULATORS |
| CN111386273B (zh) | 2017-09-27 | 2024-06-14 | 因赛特公司 | 可用作tam抑制剂的吡咯并三嗪衍生物的盐 |
| WO2019164847A1 (en) | 2018-02-20 | 2019-08-29 | Incyte Corporation | Indazole compounds and uses thereof |
| US10745388B2 (en) | 2018-02-20 | 2020-08-18 | Incyte Corporation | Indazole compounds and uses thereof |
| SG11202007917VA (en) | 2018-02-20 | 2020-09-29 | Incyte Corp | N-(phenyl)-2-(phenyl)pyrimidine-4-carboxamide derivatives and related compounds as hpk1 inhibitors for treating cancer |
| US11299473B2 (en) | 2018-04-13 | 2022-04-12 | Incyte Corporation | Benzimidazole and indole compounds and uses thereof |
| MX2021000127A (es) | 2018-06-29 | 2021-03-29 | Incyte Corp | Formulaciones de un inhibidor de axl/mer. |
| US10899755B2 (en) | 2018-08-08 | 2021-01-26 | Incyte Corporation | Benzothiazole compounds and uses thereof |
| ES2973117T3 (es) | 2018-09-25 | 2024-06-18 | Incyte Corp | Compuestos de pirazolo[4,3-d]pirimidina como moduladores de ALK2 y/o FGFR |
| JP2022543155A (ja) | 2019-08-06 | 2022-10-07 | インサイト・コーポレイション | Ｈｐｋ１阻害剤の固体形態 |
| CA3174539A1 (en) | 2020-03-06 | 2021-09-10 | Incyte Corporation | Combination therapy comprising axl/mer and pd-1/pd-l1 inhibitors |
| WO2024240088A1 (en) * | 2023-05-19 | 2024-11-28 | Chengdu Anticancer Bioscience , Ltd. | Compounds, compositions and methods of treating disorders |
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| KR20000076426A (ko) * | 1997-03-19 | 2000-12-26 | 스타르크, 카르크 | 피롤로[2,3-ｄ]피리미딘 및 티로신 키나제 저해제로서의 그의 용도 |
| UA71945C2 (en) * | 1999-01-27 | 2005-01-17 | Pfizer Prod Inc | Substituted bicyclic derivatives being used as anticancer agents |
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- 2000-09-15 CA CA002385769A patent/CA2385769A1/en not_active Abandoned
- 2000-09-15 JP JP2001523405A patent/JP2003509427A/ja not_active Withdrawn
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- 2000-09-15 AT AT00963510T patent/ATE380814T1/de active
- 2000-09-15 CN CN00815776A patent/CN1390220A/zh active Pending
- 2000-09-15 NZ NZ517759A patent/NZ517759A/en unknown
- 2000-09-15 WO PCT/US2000/025357 patent/WO2001019828A2/en active IP Right Grant
- 2000-09-15 SK SK379-2002A patent/SK3792002A3/sk unknown
- 2000-09-15 PL PL00354241A patent/PL354241A1/xx not_active Application Discontinuation
- 2000-09-15 ES ES00963510T patent/ES2299434T3/es not_active Expired - Lifetime
- 2000-09-15 BR BR0014075-9A patent/BR0014075A/pt not_active IP Right Cessation
- 2000-09-15 KR KR1020027003507A patent/KR20020063854A/ko not_active Application Discontinuation
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- 2000-09-15 DE DE60037455T patent/DE60037455T2/de not_active Expired - Lifetime
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| NZ517759A (en) | 2004-04-30 |
| PL354241A1 (en) | 2003-12-29 |
| DE60037455D1 (de) | 2008-01-24 |
| CZ2002934A3 (cs) | 2002-07-17 |
| TR200201506T2 (tr) | 2002-10-21 |
| KR20020063854A (ko) | 2002-08-05 |
| BR0014075A (pt) | 2002-07-16 |
| DE60037455T2 (de) | 2008-11-27 |
| IL148719A0 (en) | 2002-09-12 |
| CY1107886T1 (el) | 2013-06-19 |
| HUP0303363A2 (hu) | 2004-07-28 |
| WO2001019828A2 (en) | 2001-03-22 |
| ATE380814T1 (de) | 2007-12-15 |
| AU7491400A (en) | 2001-04-17 |
| CA2385769A1 (en) | 2001-03-22 |
| BG106585A (en) | 2003-03-31 |
| CN1390220A (zh) | 2003-01-08 |
| HK1053831A1 (zh) | 2003-11-07 |
| ES2299434T3 (es) | 2008-06-01 |
| PT1268481E (pt) | 2008-03-19 |
| WO2001019828A3 (en) | 2001-10-04 |
| NO20021329L (no) | 2002-05-21 |
| MXPA02002938A (es) | 2004-12-06 |
| AR029766A1 (es) | 2003-07-16 |
| EP1268481A2 (en) | 2003-01-02 |
| NO20021329D0 (no) | 2002-03-18 |
| SK3792002A3 (en) | 2003-09-11 |
| EP1268481B1 (en) | 2007-12-12 |
| DK1268481T3 (da) | 2008-05-05 |
| JP2003509427A (ja) | 2003-03-11 |
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