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HK1033277A1 - Emulsion preconcentrates containing cyclosporin or a macrolide - Google Patents

Emulsion preconcentrates containing cyclosporin or a macrolide Download PDF

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Publication number
HK1033277A1
HK1033277A1 HK01104070A HK01104070A HK1033277A1 HK 1033277 A1 HK1033277 A1 HK 1033277A1 HK 01104070 A HK01104070 A HK 01104070A HK 01104070 A HK01104070 A HK 01104070A HK 1033277 A1 HK1033277 A1 HK 1033277A1
Authority
HK
Hong Kong
Prior art keywords
macrolide
containing cyclosporin
emulsion preconcentrates
emulsion
preconcentrates containing
Prior art date
Application number
HK01104070A
Other languages
English (en)
Chinese (zh)
Other versions
HK1033277B (en
Inventor
Ambuhl Michael
Luckel Barbara
Richter Friedrich
Haberlin Barbara
Meinzer Armin
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27269231&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1033277(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9804742.6A external-priority patent/GB9804742D0/en
Priority claimed from GBGB9805104.8A external-priority patent/GB9805104D0/en
Priority claimed from GBGB9805199.8A external-priority patent/GB9805199D0/en
Application filed by Novartis Ag filed Critical Novartis Ag
Priority to HK03106974.4A priority Critical patent/HK1056310B/xx
Priority to HK03106973.5A priority patent/HK1056309B/xx
Publication of HK1033277A1 publication Critical patent/HK1033277A1/xx
Publication of HK1033277B publication Critical patent/HK1033277B/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13Cyclosporins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P41/00Drugs used in surgical methods, e.g. surgery adjuvants for preventing adhesion or for vitreum substitution

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dispersion Chemistry (AREA)
  • Oncology (AREA)
  • Surgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Communicable Diseases (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Transplantation (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
HK01104070.4A 1998-03-06 1999-03-04 Emulsion preconcentrates containing cyclosporin or a macrolide HK1033277B (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
HK03106974.4A HK1056310B (en) 1998-03-06 2001-06-13 Emulsion preconcentrates containing cyclosporin or a macrolide
HK03106973.5A HK1056309B (en) 1998-03-06 2001-06-13 Emulsion preconcentrates containing cyclosporin or a macrolide

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
GBGB9804742.6A GB9804742D0 (en) 1998-03-06 1998-03-06 Organic compounds
GB9804742 1998-03-06
GBGB9805104.8A GB9805104D0 (en) 1998-03-10 1998-03-10 Organic compounds
GB9805104 1998-03-10
GBGB9805199.8A GB9805199D0 (en) 1998-03-11 1998-03-11 Organic compounds
GB9805199 1998-03-11
PCT/EP1999/001415 WO1999044584A1 (en) 1998-03-06 1999-03-04 Emulsion preconcentrates containing cyclosporin or a macrolide

Related Parent Applications (2)

Application Number Title Priority Date Filing Date
HK03106974.4A Division HK1056310B (en) 1998-03-06 2001-06-13 Emulsion preconcentrates containing cyclosporin or a macrolide
HK03106973.5A Division HK1056309B (en) 1998-03-06 2001-06-13 Emulsion preconcentrates containing cyclosporin or a macrolide

Related Child Applications (2)

Application Number Title Priority Date Filing Date
HK03106974.4A Addition HK1056310B (en) 1998-03-06 2001-06-13 Emulsion preconcentrates containing cyclosporin or a macrolide
HK03106973.5A Addition HK1056309B (en) 1998-03-06 2001-06-13 Emulsion preconcentrates containing cyclosporin or a macrolide

Publications (2)

Publication Number Publication Date
HK1033277A1 true HK1033277A1 (en) 2001-08-24
HK1033277B HK1033277B (en) 2003-10-31

Family

ID=

Also Published As

Publication number Publication date
IT1313550B1 (it) 2002-09-09
IL138248A0 (en) 2001-10-31
KR20010041657A (ko) 2001-05-25
PE20000324A1 (es) 2000-04-13
JP2004189753A (ja) 2004-07-08
WO1999044584A1 (en) 1999-09-10
FR2853546B1 (fr) 2006-04-07
TWI236912B (en) 2005-08-01
CZ20003222A3 (cs) 2000-12-13
TW200422057A (en) 2004-11-01
ID25908A (id) 2000-11-09
EP1354582A2 (en) 2003-10-22
TR200002586T2 (tr) 2000-11-21
AU2836199A (en) 1999-09-20
ITMI990452A1 (it) 2000-09-05
FR2775596A1 (fr) 1999-09-10
DE69920668T2 (de) 2005-10-06
CA2322845A1 (en) 1999-09-10
EP1059913A1 (en) 2000-12-20
FR2775596B1 (fr) 2004-12-24
NO331800B1 (no) 2012-04-02
DE19983012T1 (de) 2001-02-01
FR2800277B1 (fr) 2004-06-25
SK285139B6 (sk) 2006-07-07
IL138248A (en) 2006-06-11
GB2350791A (en) 2000-12-13
AU749217B2 (en) 2002-06-20
JP2002505271A (ja) 2002-02-19
BR9908597A (pt) 2000-11-14
HUP0101080A2 (hu) 2001-08-28
HUP0101080A3 (en) 2001-12-28
ATE277599T1 (de) 2004-10-15
NZ506644A (en) 2004-02-27
TWI248368B (en) 2006-02-01
CN1195495C (zh) 2005-04-06
HK1034038A1 (en) 2001-10-12
NO20004299D0 (no) 2000-08-29
GB2350791B (en) 2003-04-02
FR2881956A1 (fr) 2006-08-18
CA2322845C (en) 2009-12-08
KR100443306B1 (ko) 2004-08-09
CO4930289A1 (es) 2000-06-27
BE1013423A5 (fr) 2002-01-15
CN1292684A (zh) 2001-04-25
TWI257870B (en) 2006-07-11
FR2800277A1 (fr) 2001-05-04
BE1012400A5 (fr) 2000-10-03
NO20004299L (no) 2000-08-29
GB0021495D0 (en) 2000-10-18
EP1354582A3 (en) 2004-06-09
CZ301967B6 (cs) 2010-08-18
BE1013648A5 (fr) 2002-05-07
AR015729A1 (es) 2001-05-16
FR2853546A1 (fr) 2004-10-15
SK13192000A3 (sk) 2001-02-12
MY129274A (en) 2007-03-30
EP1059913B1 (en) 2004-09-29
ES2228014T3 (es) 2005-04-01
PT1059913E (pt) 2005-01-31
DE69920668D1 (de) 2004-11-04

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Legal Events

Date Code Title Description
PF Patent in force
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20130304