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HK1011542A1 - Reductive alkylation of glycopeptide antibiotics - Google Patents

Reductive alkylation of glycopeptide antibiotics Download PDF

Info

Publication number
HK1011542A1
HK1011542A1 HK98112780A HK98112780A HK1011542A1 HK 1011542 A1 HK1011542 A1 HK 1011542A1 HK 98112780 A HK98112780 A HK 98112780A HK 98112780 A HK98112780 A HK 98112780A HK 1011542 A1 HK1011542 A1 HK 1011542A1
Authority
HK
Hong Kong
Prior art keywords
copper
glycopeptide antibiotic
mmol
complex
glycopeptide
Prior art date
Application number
HK98112780A
Other languages
German (de)
English (en)
French (fr)
Chinese (zh)
Other versions
HK1011542B (en
Inventor
Alan Berglund Richard
Anne Lockwood Nancy
Eugene Magadanz Howard
Zheng Hua
Original Assignee
Eli Lilly And Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly And Company filed Critical Eli Lilly And Company
Publication of HK1011542A1 publication Critical patent/HK1011542A1/en
Publication of HK1011542B publication Critical patent/HK1011542B/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K9/00Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HK98112780.2A 1996-11-21 1998-12-03 Reductive alkylation of glycopeptide antibiotics HK1011542B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US3159696P 1996-11-21 1996-11-21
US31596P 1996-11-21

Publications (2)

Publication Number Publication Date
HK1011542A1 true HK1011542A1 (en) 1999-07-16
HK1011542B HK1011542B (en) 2005-08-19

Family

ID=

Also Published As

Publication number Publication date
TW585868B (en) 2004-05-01
AU723941B2 (en) 2000-09-07
TR199901679T2 (xx) 1999-09-21
ZA9710428B (en) 1999-05-19
CO4650045A1 (es) 1998-09-03
EA002925B1 (ru) 2002-10-31
CZ179499A3 (cs) 2000-01-12
NO325365B1 (no) 2008-04-14
CN1244802A (zh) 2000-02-16
HU227641B1 (en) 2011-10-28
EG23855A (en) 2007-11-11
KR20000057156A (ko) 2000-09-15
AR010621A1 (es) 2000-06-28
BR9713523A (pt) 2000-03-21
EP0845478B1 (en) 2005-01-12
NZ335840A (en) 2000-09-29
EP0845478A1 (en) 1998-06-03
UA58526C2 (uk) 2003-08-15
HUP0000268A2 (hu) 2000-08-28
ID18900A (id) 1998-05-20
NO992415D0 (no) 1999-05-20
JP2001504494A (ja) 2001-04-03
IL129991A0 (en) 2000-02-29
DE69732215T2 (de) 2006-01-12
JP4308912B2 (ja) 2009-08-05
CA2272240C (en) 2011-02-08
CZ300528B6 (cs) 2009-06-10
ATE286910T1 (de) 2005-01-15
DE69732215D1 (de) 2005-02-17
PE17499A1 (es) 1999-02-19
HUP0000268A3 (en) 2001-04-28
CN100463917C (zh) 2009-02-25
KR100514276B1 (ko) 2005-09-13
EA199900480A1 (ru) 2000-02-28
CA2272240A1 (en) 1998-05-28
BR9713523B1 (pt) 2010-07-27
NO992415L (no) 1999-05-20
WO1998022121A1 (en) 1998-05-28
PL190780B1 (pl) 2006-01-31
AU5449798A (en) 1998-06-10
MY117383A (en) 2004-06-30

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20161119