CA2500311A1 - Modified release dosage forms - Google Patents

Modified release dosage forms Download PDF

Info

Publication number: CA2500311A1
Authority: CA; Canada
Prior art keywords: shell; core; active ingredient; dosage form; release
Prior art date: 2002-09-28
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

CA002500311A

Other languages

English (en)

French (fr)

Inventor

Shun-Por Li

Der-Yang Lee

Gerard P. Mcnally

Daniel Mcteigue

Narendra Parikh

Harry S. Sowden

David Wynn

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Kenvue Brands LLC

Original Assignee

Individual

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-09-28

Filing date

2003-03-21

Publication date

2004-04-08

2002-09-28 Priority claimed from PCT/US2002/031117 external-priority patent/WO2003026629A2/en

2003-03-21 Application filed by Individual filed Critical Individual

2003-03-21 Priority claimed from PCT/US2003/008891 external-priority patent/WO2004028504A1/en

2004-04-08 Publication of CA2500311A1 publication Critical patent/CA2500311A1/en

Status Abandoned legal-status Critical Current

Links

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229960003656 ricinoleic acid Drugs 0.000 description 1
FEUQNCSVHBHROZ-UHFFFAOYSA-N ricinoleic acid Natural products CCCCCCC(O[Si](C)(C)C)CC=CCCCCCCCC(=O)OC FEUQNCSVHBHROZ-UHFFFAOYSA-N 0.000 description 1
229960000371 rofecoxib Drugs 0.000 description 1
RZJQGNCSTQAWON-UHFFFAOYSA-N rofecoxib Chemical compound C1=CC(S(=O)(=O)C)=CC=C1C1=C(C=2C=CC=CC=2)C(=O)OC1 RZJQGNCSTQAWON-UHFFFAOYSA-N 0.000 description 1
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235000019333 sodium laurylsulphate Nutrition 0.000 description 1
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125000001424 substituent group Chemical group 0.000 description 1
235000019408 sucralose Nutrition 0.000 description 1
BAQAVOSOZGMPRM-QBMZZYIRSA-N sucralose Chemical compound O[C@@H]1[C@@H](O)[C@@H](Cl)[C@@H](CO)O[C@@H]1O[C@@]1(CCl)[C@@H](O)[C@H](O)[C@@H](CCl)O1 BAQAVOSOZGMPRM-QBMZZYIRSA-N 0.000 description 1
229950005175 sudoxicam Drugs 0.000 description 1
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MLKXDPUZXIRXEP-MFOYZWKCSA-N sulindac Chemical compound CC1=C(CC(O)=O)C2=CC(F)=CC=C2\C1=C/C1=CC=C(S(C)=O)C=C1 MLKXDPUZXIRXEP-MFOYZWKCSA-N 0.000 description 1
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230000009967 tasteless effect Effects 0.000 description 1
229960000351 terfenadine Drugs 0.000 description 1
IMCGHZIGRANKHV-AJNGGQMLSA-N tert-butyl (3s,5s)-2-oxo-5-[(2s,4s)-5-oxo-4-propan-2-yloxolan-2-yl]-3-propan-2-ylpyrrolidine-1-carboxylate Chemical compound O1C(=O)[C@H](C(C)C)C[C@H]1[C@H]1N(C(=O)OC(C)(C)C)C(=O)[C@H](C(C)C)C1 IMCGHZIGRANKHV-AJNGGQMLSA-N 0.000 description 1
229960002180 tetracycline Drugs 0.000 description 1
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235000019364 tetracycline Nutrition 0.000 description 1
150000003522 tetracyclines Chemical class 0.000 description 1
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230000008719 thickening Effects 0.000 description 1
KUAZQDVKQLNFPE-UHFFFAOYSA-N thiram Chemical compound CN(C)C(=S)SSC(=S)N(C)C KUAZQDVKQLNFPE-UHFFFAOYSA-N 0.000 description 1
229960001017 tolmetin Drugs 0.000 description 1
UPSPUYADGBWSHF-UHFFFAOYSA-N tolmetin Chemical compound C1=CC(C)=CC=C1C(=O)C1=CC=C(CC(O)=O)N1C UPSPUYADGBWSHF-UHFFFAOYSA-N 0.000 description 1
239000008379 tooth decay inhibitor Substances 0.000 description 1
239000008378 tooth mineralizer Substances 0.000 description 1
239000008377 tooth whitener Substances 0.000 description 1
230000000699 topical effect Effects 0.000 description 1
238000012549 training Methods 0.000 description 1
230000007704 transition Effects 0.000 description 1
ILJSQTXMGCGYMG-UHFFFAOYSA-N triacetic acid Chemical compound CC(=O)CC(=O)CC(O)=O ILJSQTXMGCGYMG-UHFFFAOYSA-N 0.000 description 1
229960002622 triacetin Drugs 0.000 description 1
QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
229940078499 tricalcium phosphate Drugs 0.000 description 1
229910000391 tricalcium phosphate Inorganic materials 0.000 description 1
235000019731 tricalcium phosphate Nutrition 0.000 description 1
PVNIQBQSYATKKL-UHFFFAOYSA-N tripalmitin Chemical compound CCCCCCCCCCCCCCCC(=O)OCC(OC(=O)CCCCCCCCCCCCCCC)COC(=O)CCCCCCCCCCCCCCC PVNIQBQSYATKKL-UHFFFAOYSA-N 0.000 description 1
150000004043 trisaccharides Chemical class 0.000 description 1
239000002996 urinary tract agent Substances 0.000 description 1
235000015112 vegetable and seed oil Nutrition 0.000 description 1
239000008158 vegetable oil Substances 0.000 description 1
238000007601 warm air drying Methods 0.000 description 1
230000004584 weight gain Effects 0.000 description 1
235000019786 weight gain Nutrition 0.000 description 1
235000021119 whey protein Nutrition 0.000 description 1

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Medicinal Preparation (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

CA002500311A 2002-09-28 2003-03-21 Modified release dosage forms Abandoned CA2500311A1 (en)

Applications Claiming Priority (11)

Application Number	Priority Date	Filing Date	Title
USPCT/US02/31129		2002-09-28
PCT/US2002/031117 WO2003026629A2 (en)	2001-09-28	2002-09-28	Modified release dosage forms
USPCT/US02/31163		2002-09-28
USPCT/US02/31117		2002-09-28
USPCT/US02/31024		2002-09-28
PCT/US2002/031024 WO2003026625A1 (en)	2001-09-28	2002-09-28	Modified release dosage forms
PCT/US2002/031062 WO2003026626A2 (en)	2001-09-28	2002-09-28	Modified release dosage forms
PCT/US2002/031129 WO2003026630A1 (en)	2001-09-28	2002-09-28	Dosage forms having an inner core and outer shell with different shapes
PCT/US2002/031163 WO2003026627A1 (en)	2001-09-28	2002-09-28	Composite dosage forms
USPCT/US02/31062		2002-09-28
PCT/US2003/008891 WO2004028504A1 (en)	2002-09-28	2003-03-21	Modified release dosage forms

Publications (1)

Publication Number	Publication Date
CA2500311A1 true CA2500311A1 (en)	2004-04-08

Family

ID=34271652

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
CA002500312A Abandoned CA2500312A1 (en)	2002-09-28	2003-03-21	Modified release dosage form
CA2500313A Expired - Fee Related CA2500313C (en)	2002-09-28	2003-03-21	Polymer composition and dosage forms comprising the same
CA002500311A Abandoned CA2500311A1 (en)	2002-09-28	2003-03-21	Modified release dosage forms

Family Applications Before (2)

Application Number	Title	Priority Date	Filing Date
CA002500312A Abandoned CA2500312A1 (en)	2002-09-28	2003-03-21	Modified release dosage form
CA2500313A Expired - Fee Related CA2500313C (en)	2002-09-28	2003-03-21	Polymer composition and dosage forms comprising the same

Country Status (8)

Country	Link
JP (3)	JP2006517182A (zh)
CN (3)	CN1700907A (zh)
AT (1)	ATE444739T1 (zh)
AU (4)	AU2003218359A1 (zh)
BR (5)	BR0314777A (zh)
CA (3)	CA2500312A1 (zh)
DE (2)	DE60335270D1 (zh)
MX (1)	MXPA05003283A (zh)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US12161754B2 (en)	2017-12-20	2024-12-10	Purdue Pharma L.P.	Abuse deterrent morphine sulfate dosage forms

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Publication number	Priority date	Publication date	Assignee	Title
CA2470463C (en)	2004-06-09	2012-09-18	Lornamead Brands, Inc.	Tooth whitening products and methods of making the same
SA07280459B1 (ar) *	2006-08-25	2011-07-20	بيورديو فارما إل. بي.	أشكال جرعة صيدلانية للتناول عن طريق الفم مقاومة للعبث تشتمل على مسكن شبه أفيوني
WO2009153635A1 (en) *	2008-06-19	2009-12-23	University Of Witwatersrand, Johannesburg	A chronotherapeutic pharmaceutical dosage form
JPWO2011118454A1 (ja) *	2010-03-23	2013-07-04	リンテック株式会社	固形製剤
US9693957B2 (en) *	2011-07-08	2017-07-04	The University Of North Carolina At Chapel Hill	Metal bisphosphonate nanoparticles for anti-cancer therapy and imaging and for treating bone disorders
MX359529B (es) *	2012-02-07	2018-10-01	Mcneil Ppc Inc	Tabletas recubiertas de desintegración rápida.
WO2013183497A1 (ja) *	2012-06-05	2013-12-12	武田薬品工業株式会社	有核錠
WO2016044704A1 (en) *	2014-09-19	2016-03-24	The Procter & Gamble Company	Pulsed release phenylephrine dosage forms
BR112020013374A2 (pt) *	2017-12-29	2020-12-01	Exentis Knowledge Gmbh	sistema de administração de medicamentos
US11752107B2 (en) *	2021-07-30	2023-09-12	Evecxia Therapeutics, Inc.	5-hydroxytryptophan gastroretentive dosage forms
CN115295864B (zh) *	2021-11-09	2023-08-11	深圳市德方创域新能源科技有限公司	正极补锂添加剂及其制备方法与应用

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EP0662824A1 (en) *	1992-09-30	1995-07-19	Pfizer Inc.	Article containing a core and a coating having a non constant thickness
GB9402203D0 (en) *	1994-02-04	1994-03-30	Smithkline Beecham Plc	Pharmaceutical formulation
DE4431653C2 (de) *	1994-09-06	2000-01-20	Lohmann Therapie Syst Lts	Manteltablette zur kontrollierten Freisetzung von Wirkstoffen, ein Verfahren zu ihrer Herstellung und ihre Verwendung
IT1282576B1 (it) *	1996-02-06	1998-03-31	Jagotec Ag	Compressa farmaceutica atta a cedere la sostanza attiva in tempi successivi e predeterminabili
US6602521B1 (en) *	1998-09-29	2003-08-05	Impax Pharmaceuticals, Inc.	Multiplex drug delivery system suitable for oral administration
EP1275373A4 (en) *	2000-04-17	2007-04-04	Astellas Pharma Inc	DRUG DISPERSION SYSTEM FOR THE AVOIDANCE OF PHARMACOKINETIC INTERACTIONS BETWEEN ACTIVE SUBSTANCES AND METHODOLOGY THEREOF
IL157075A0 (en) *	2001-02-13	2004-02-08	Astrazeneca Ab	Novel modified release formulation

2003
- 2003-03-21 AU AU2003218359A patent/AU2003218359A1/en not_active Abandoned
- 2003-03-21 CA CA002500312A patent/CA2500312A1/en not_active Abandoned
- 2003-03-21 AT AT03714356T patent/ATE444739T1/de not_active IP Right Cessation
- 2003-03-21 CN CN03825324.0A patent/CN1700907A/zh active Pending
- 2003-03-21 AU AU2003220466A patent/AU2003220466A1/en not_active Abandoned
- 2003-03-21 BR BR0314777-0A patent/BR0314777A/pt not_active Application Discontinuation
- 2003-03-21 CA CA2500313A patent/CA2500313C/en not_active Expired - Fee Related
- 2003-03-21 CA CA002500311A patent/CA2500311A1/en not_active Abandoned
- 2003-03-21 JP JP2004539769A patent/JP2006517182A/ja active Pending
- 2003-03-21 MX MXPA05003283A patent/MXPA05003283A/es unknown
- 2003-03-21 JP JP2004539767A patent/JP2006517514A/ja active Pending
- 2003-03-21 AU AU2003220472A patent/AU2003220472A1/en not_active Abandoned
- 2003-03-21 CN CN03825331.3A patent/CN1700908A/zh active Pending
- 2003-03-21 AU AU2003225944A patent/AU2003225944A1/en not_active Abandoned
- 2003-03-21 BR BR0314781-9A patent/BR0314781A/pt not_active Application Discontinuation
- 2003-03-21 JP JP2004539770A patent/JP2006517183A/ja active Pending
- 2003-03-21 BR BR0314547-6A patent/BR0314547A/pt not_active Application Discontinuation
- 2003-03-21 CN CN03823065.8A patent/CN1684671A/zh active Pending
- 2003-03-21 DE DE60335270T patent/DE60335270D1/de not_active Expired - Lifetime
- 2003-03-21 BR BR0314804-1A patent/BR0314804A/pt not_active Application Discontinuation
- 2003-03-21 DE DE60329614T patent/DE60329614D1/de not_active Expired - Lifetime
- 2003-03-21 BR BR0314787-8A patent/BR0314787A/pt not_active IP Right Cessation

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US12161754B2 (en)	2017-12-20	2024-12-10	Purdue Pharma L.P.	Abuse deterrent morphine sulfate dosage forms

Also Published As

Publication number	Publication date
DE60329614D1 (de)	2009-11-19
BR0314781A (pt)	2005-07-26
ATE444739T1 (de)	2009-10-15
CN1700908A (zh)	2005-11-23
JP2006517183A (ja)	2006-07-20
MXPA05003283A (es)	2005-11-23
AU2003225944A1 (en)	2004-04-19
BR0314777A (pt)	2005-07-26
AU2003220472A1 (en)	2004-04-19
CN1700907A (zh)	2005-11-23
JP2006517514A (ja)	2006-07-27
BR0314804A (pt)	2005-08-02
AU2003220466A1 (en)	2004-04-19
DE60335270D1 (de)	2011-01-20
CA2500312A1 (en)	2004-04-08
CA2500313C (en)	2011-06-07
BR0314547A (pt)	2005-08-09
AU2003218359A1 (en)	2004-04-19
CN1684671A (zh)	2005-10-19
CA2500313A1 (en)	2004-04-08
BR0314787A (pt)	2005-07-26
JP2006517182A (ja)	2006-07-20

Publication	Publication Date	Title
US20030232082A1 (en)	2003-12-18	Modified release dosage forms
CA2499882C (en)	2010-11-09	Modified release dosage form with two cores
CA2663871C (en)	2015-05-19	Multi-core solid dosage form comprising a transparent coating between said cores
CA2500311A1 (en)	2004-04-08	Modified release dosage forms
US20080206337A1 (en)	2008-08-28	Method of making dosage forms comprising polymeric compositions
US20050196446A1 (en)	2005-09-08	Polymeric compositions and dosage forms comprising the same
US20050196447A1 (en)	2005-09-08	Polymeric compositions and dosage forms comprising the same
US20050196442A1 (en)	2005-09-08	Polymeric compositions and dosage forms comprising the same
CA2556922C (en)	2012-05-15	Polymeric compositions and dosage forms comprising the same
CA2612989A1 (en)	2007-11-08	Osmotic dosage form
US20060233882A1 (en)	2006-10-19	Osmotic dosage form
AU2002337772A1 (en)	2003-04-07	Modified release dosage forms
KR20070017128A (ko)	2007-02-08	중합체성 조성물 및 이를 포함하는 투여 형태

Legal Events

Date	Code	Title	Description
2009-03-23	FZDE	Discontinued

CA2500311A1 - Modified release dosage forms - Google Patents

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Applications Claiming Priority (11)

Publications (1)

Family

ID=34271652

Family Applications (3)

Family Applications Before (2)

Country Status (8)

Cited By (1)

Families Citing this family (11)

Family Cites Families (7)

Cited By (1)

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