(Q40883086)

24 September 2017

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title

5-HT 1B/D receptor antagonists (English)

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24 September 2017

Pauwels PJ

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24 September 2017

publication date

1 September 1997

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24 September 2017

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24 September 2017

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24 September 2017

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24 September 2017

page(s)

293-303

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Differential effects of clomipramine given locally or systemically on extracellular 5-hydroxytryptamine in raphe nuclei and frontal cortex. An in vivo brain microdialysis study

24 September 2017

cites work

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7 January 2021

Cell-specific coupling of the cloned human 5-HT1F receptor to multiple signal transduction pathways

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7 January 2021

Structure functional expression and spatial distribution of a cloned cDNA encoding a rat 5-HT1D-like receptor

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7 January 2021

Terminal serotonin autoreceptor function in the rat hippocampus is not modified by pertussis and cholera toxins

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7 January 2021

Long-term 5-HT reuptake blockade, but not monoamine oxidase inhibition, decreases the function of terminal 5-HT autoreceptors: an electrophysiological study in the rat brain

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7 January 2021

Effect of chronic antidepressant treatment on 5-HT1B presynaptic heteroreceptors inhibiting acetylcholine release

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7 January 2021

The mouse 5-hydroxytryptamine1B receptor is localized predominantly on axon terminals

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7 January 2021

5-HT and antidepressants: in vitro and in vivo release studies

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7 January 2021

Animal models for anxiety and response to serotonergic drugs

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7 January 2021

Autoradiographic characterisation and localisation of 5-HT1D compared to 5-HT1B binding sites in rat brain.

1 reference

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7 January 2021

Further characterization of the putative 5-HT receptor which mediates blockade of neurogenic plasma extravasation in rat dura mater

1 reference

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7 January 2021

5-HT1D receptor type is involved in stimulation of cell proliferation by serotonin in human small cell lung carcinoma

1 reference

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7 January 2021

1-(3-Trifluoromethylphenyl) piperazine (TFMPP) in the ventral tegmental area reduces the effect of desipramine in the forced swimming test in rats: possible role of serotonin receptors

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7 January 2021

Serotonin function in obsessive-compulsive disorder. A comparison of the effects of tryptophan and m-chlorophenylpiperazine in patients and healthy subjects

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7 January 2021

Neuropharmacology of 5-hydroxytryptamine1B/D receptor ligands

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7 January 2021

Evolution of a novel series of [(N,N-dimethylamino)propyl]- and piperazinylbenzanilides as the first selective 5-HT1D antagonists

1 reference

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7 January 2021

WAY-100635 and GR127935: Effects on 5-hydroxytryptamine-containing neurones

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7 January 2021

Brain serotonin receptors in Huntington's disease.

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7 January 2021

Serotonin-induced contraction in canine coronary artery and saphenous vein: role of a 5-HT1D-like receptor

1 reference

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7 January 2021

Response of cerebellar Purkinje cells to serotonin and the 5-HT1A agonists 8-OH-DPAT and ipsapirone in vitro

1 reference

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7 January 2021

The effect of paroxetine on 5-HT efflux in the rat dorsal raphe nucleus is potentiated by both 5-HT1A and 5-HT1B/D receptor antagonists

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Evidence that 5-hydroxytryptamine release in rat dorsal raphé nucleus is controlled by 5-HT1A, 5-HT1B and 5-HT1D autoreceptors.

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

5-HT and mechanisms of defence

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Blockade of porcine carotid vascular response to sumatriptan by GR 127935, a selective 5-HT1D receptor antagonist

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

In situ hybridization evidence for the synthesis of 5-HT1B receptor in serotoninergic neurons of anterior raphe nuclei in the rat brain

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

5-HT1b receptors in an animal model of depression

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Clinical and experimental effects of sumatriptan in humans

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Postsynaptic localization of 5-HT1D receptor binding sites in human caudate

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

The role of 5-HT1D and 5-HT1A receptors in mediating 5-hydroxytryptophan induced myoclonic jerks in guinea pigs

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Distinct 5-HT(1B) and 5-HT(1D) serotonin receptors in rat: Structural and pharmacological comparison of the two cloned receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Alignment of receptor nomenclature with the human genome: classification of 5-HT1B and 5-HT1D receptor subtypes.

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Cloning and characterisation of the rabbit 5-HT1D alpha and 5-HT1D beta receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

5-HT 1D receptors mediate SKF 99101H-induced hypothermia in the guinea pig.

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Of mice and flies: commonalities among 5-HT receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Detection and characterization of the serotonin 5-HT 1D receptor in rat and human brain

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Characterization of a novel 3H-5-hydroxytryptamine binding site subtype in bovine brain membranes

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Partial agonists, full agonists, antagonists: dilemmas of definition

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Species differences in the pharmacology of terminal 5-HT autoreceptors in mammalian brain

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

5-HT1D receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in calf substantia nigra

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

The effects of GR127935, a putative 5-HT1D receptor antagonist, on brain 5-HT metabolism, extracellular 5-HT concentration and behaviour in the guinea pig

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Variable participation of 5-HT1-like receptors and 5-HT2 receptors in serotonin-induced contraction of human isolated coronary arteries. 5-HT1-like receptors resemble cloned 5-HT1D beta receptors.

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Subunits beta gamma of heterotrimeric G protein activate beta 2 isoform of phospholipase C

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

On the importance of the "antagonist assumption" to how receptors express themselves.

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Immunolabeling of central serotonin 5-HT1D beta receptors in the rat, mouse, and guinea pig with a specific anti-peptide antiserum

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Constitutive activity of receptors coupled to guanine nucleotide regulatory proteins

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Detection of a novel serotonin receptor subtype (5-HT1E) in human brain: interaction with a GTP-binding protein

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

The orphan receptor cDNA RDC4 encodes a 5-HT1D serotonin receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Increase of central 5-HT1B binding sites following 5,7-dihydroxytryptamine axotomy in the adult rat

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Ketanserin-sensitive depressant actions of 5-HT receptor agonists in the neonatal rat spinal cord

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Is there a relationship between 5-HT1B receptors and the mechanisms of action of antidepressant drugs in the learned helplessness paradigm in rats?

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

CP-93,129, a potent and selective 5-HT1B receptor agonist blocks neurogenic plasma extravasation within rat but not guinea-pig dura mater

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Conversion of the human 5-HT1D beta serotonin receptor to the rat 5-HT1B ligand-binding phenotype by Thr355Asn site directed mutagenesis

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

A pharmacological analysis of the 5-HT receptor mediating inhibition of 5-HT release in the guinea-pig frontal cortex

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Inhibition of noradrenaline release via presynaptic 5-HT1D alpha receptors in human atrium

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Inhibition of noradrenaline release from the sympathetic nerves of the human saphenous vein via presynaptic 5-HT receptors similar to the 5-HT 1D subtype

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Serotonin autoreceptor subsensitivity and antidepressant activity

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

The unique effect of methiothepin on the terminal serotonin autoreceptor in the rat hypothalamus could be an example of inverse agonism

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Effects of acute and repeated administration of citalopram on extracellular levels of serotonin in rat brain

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Neurogenic versus vascular mechanisms of sumatriptan and ergot alkaloids in migraine

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Role of the serotonin receptor subtype 5-HT1D on basal and stimulated growth hormone secretion.

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

A single amino-acid difference confers major pharmacological variation between human and rodent 5-HT1B receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

The 5-HT1D receptor antagonist GR 127,935 is an agonist at cloned human 5-HT1D alpha receptor sites

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Functional effects of the 5-HT1D receptor antagonist GR 127,935 at human 5-HT1D alpha, 5-HT1D beta, 5-HT1A and opossum 5-HT1B receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Pharmacology of cloned human 5-HT1D receptor-mediated functional responses in stably transfected rat C6-glial cell lines: further evidence differentiating human 5-HT1D and 5-HT1B receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

How Efficacious are 5-HT 1B/D Receptor Ligands: an Answer from GTPγS Binding Studies with Stably Transfected C6-glial Cell Lines

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Promotion of cell growth by stimulation of cloned human 5-HT1D receptor sites in transfected C6-glial cells is highly sensitive to intrinsic activity at 5-HT1D receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Prevention of learned helplessness: in vivo correlation with cortical serotonin

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

5-HT1D receptors regulate 5-HT release in the rat raphe nuclei. In vivo voltammetry and in vitro superfusion studies

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Differences in the effects of ketanserin and GR127935 on 5-HT-receptor mediated responses in rabbit saphenous vein and guinea-pig jugular vein

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

The use of nitrates, calcium channel blockers and ACE inhibitors in primary care in the Northern Region: a pharmacoepidemiological study

1 reference

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7 January 2021

Enhanced aggressive behavior in mice lacking 5-HT1B receptor.

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

The 5-hydroxytryptamine 5-HT1D receptor subtype is negatively coupled to adenylate cyclase in calf substantia nigra

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

High-affinity serotonin binding sites: autoradiographic evidence for their location on retinal afferents in the rat superior colliculus

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Stimulation of central 5-HT1D receptors causes hypothermia in the guinea-pig.

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Effects of the 5-HT1D receptor antagonist GR127935 on extracellular levels of 5-HT in the guinea-pig frontal cortex as measured by microdialysis.

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

GR127935 is a potent antagonist of the 5-HT1-like receptor mediating contraction in the canine coronary artery

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Pharmacological characterisation of [35S]-GTPgammaS binding to Chinese hamster ovary cell membranes stably expressing cloned human 5-HT1D receptor subtypes

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Influence of the endothelium and nitric oxide on the contractile responses evoked by 5-HT1D receptor agonists in the rabbit isolated saphenous vein

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

The human and dog 5-HT1D receptors can both activate and inhibit adenylate cyclase in transfected cells

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Quantitative autoradiography of multiple 5-HT1 receptor subtypes in the brain of control or 5,7-dihydroxytryptamine-treated rats

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Molecular cloning and characterization of a rat brain cDNA encoding a 5-hydroxytryptamine1B receptor

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

[3H]sumatriptan labels both 5-HT1D and 5-HT1F receptor binding sites in the guinea pig brain: an autoradiographic study

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

The serotonin 5-HT1D receptor: a progress review

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Serotonin-1 receptor binding sites in the human basal ganglia are decreased in Huntington's chorea but not in Parkinson's disease: a quantitative in vitro autoradiography study

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Molecular pharmacology of 5-HT1D recognition sites: radioligand binding studies in human, pig and calf brain membranes.

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

The activity of 5-HT1D receptor ligands at cloned human 5-HT1D alpha and 5-HT1D beta receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Evidence for hyperdensity of 5HT1B binding sites in the substantia nigra of the rat after 5,7-dihydroxytryptamine intraventricular injection

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Recombinant saphenous vein 5-HT1B receptors of the rabbit: comparative pharmacology with human 5-HT1B receptors

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

Ketanserin and ritanserin discriminate between recombinant human 5-HT1D alpha and 5-HT1D beta receptor subtypes

1 reference

https://api.crossref.org/works/10.1016%2FS0306-3623%2896%2900460-0

7 January 2021

10.1016/S0306-3623(96)00460-0

Identifiers

DOI

1 reference

24 September 2017

1 reference