(Q35609958)

9 August 2017

title

[3H]xanthine amine congener of 1,3-dipropyl-8-phenylxanthine: an antagonist radioligand for adenosine receptors (English)

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9 August 2017

Jacobson KA

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9 August 2017

Ukena D

series ordinal

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9 August 2017

Kirk KL

series ordinal

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9 August 2017

Daly JW

series ordinal

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9 August 2017

language of work or name

English

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publication date

1 June 1986

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Proceedings of the National Academy of Sciences of the United States of America

9 August 2017

published in

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9 August 2017

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9 August 2017

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9 August 2017

page(s)

4089-4093

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Adenosine receptor binding: structure-activity analysis generates extremely potent xanthine antagonists

9 August 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=323672

Adenosine receptors: targets for future drugs

12 July 2018

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LIGAND: A versatile computerized approach for characterization of ligand-binding systems

12 July 2018

1 reference

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Adenosine receptors in brain membranes: binding of N6-cyclohexyl[3H]adenosine and 1,3-diethyl-8-[3H]phenylxanthine

12 July 2018

1 reference

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Reciprocal modulation of agonist and antagonist binding to inhibitory adenosine receptors by 5'-guanylylimidodiphosphate and monovalent cations

12 July 2018

1 reference

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Guanine nucleotide and cation regulation of radioligand binding to R i adenosine receptors of rat fat cells

12 July 2018

1 reference

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Evaluation of the binding of the A-1 selective adenosine radioligand, cyclopentyladenosine (CPA), to rat brain tissue

12 July 2018

1 reference

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A functionalized congener approach to adenosine receptor antagonists: amino acid conjugates of 1,3-dipropylxanthine

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=323672

Functionalized congeners of 1,3-dipropyl-8-phenylxanthine: potent antagonists for adenosine receptors that modulate membrane adenylate cyclase in pheochromocytoma cells, platelets and fat cells

12 July 2018

1 reference

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A novel 8-phenyl-substituted xanthine derivative is a selective antagonist at adenosine A1-receptors in vivo

12 July 2018

1 reference

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Evidence for an A2 adenosine receptor in guinea pig lung

12 July 2018

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Binding of [3H]cyclohexyladenosine to adenosine recognition sites in guinea pig ileal membranes: comparison with binding in brain membranes

12 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=323672

Functionalized congeners of adenosine: preparation of analogues with high affinity for A1-adenosine receptors

12 July 2018

1 reference

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Functionalized congeners of 1,3-dialkylxanthines: preparation of analogues with high affinity for adenosine receptors

12 July 2018

1 reference

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Synthesis of xanthines as adenosine antagonists, a practical quantitative structure-activity relationship application

12 July 2018

1 reference

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Demonstration of Ri-type adenosine receptors in bovine myocardium by radioligand binding

12 July 2018

1 reference

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3H5?-N-ethylcarboxamide adenosine binds to both Ra and Ri adenosine receptors in rat striatum

12 July 2018

1 reference

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A rapid filtration assay for soluble receptors using polyethylenimine-treated filters

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=323672

Functional identification of adenylate cyclase-coupled adenosine receptors in rat brain microvessels

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=323672

Subclasses of Adenosine Receptors in Brain Membranes from Adult Tissue and from Primary Cultures of Chick Embryo

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=323672

Two affinity states of Ri adenosine receptors in brain membranes. Analysis of guanine nucleotide and temperature effects on radioligand binding.

25 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=323672

Guanine nucleotide and cation regulation of the binding of [3H]cyclohexyladenosine and [3H]diethylphenylxanthine to adenosine A1 receptors in brain membranes

25 September 2018

1 reference

12 December 2020

Adenosine receptor agonists: binding and adenylate cyclase stimulation in rat liver plasma membranes

1 reference

12 December 2020

Agonist and antagonist affinities for inhibitory adenosine receptors are reciprocally affected by 5'-guanylylimidodiphosphate or N-ethylmaleimide

1 reference

12 December 2020

Characterization of adenosine receptors in rat brain by (?)[3H]N6-phenylisopropyladenosine

1 reference

12 December 2020

Identifiers

DOI

10.1073/PNAS.83.11.4089

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9 August 2017

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9 August 2017

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