(Q33530669)

27 July 2017

title

Comparative analysis of small molecules and histone substrate analogues as LSD1 lysine demethylase inhibitors (English)

1 reference

27 July 2017

Paul M Yen

0 references

Jeffrey C Culhane

1 reference

27 July 2017

Dongqing Wang

series ordinal

1 reference

27 July 2017

Philip A Cole

series ordinal

1 reference

27 July 2017

language of work or name

English

0 references

publication date

1 March 2010

1 reference

Journal of the American Chemical Society

27 July 2017

published in

1 reference

27 July 2017

volume

132

1 reference

27 July 2017

1 reference

27 July 2017

page(s)

3164-3176

1 reference

Identification of cell-active lysine specific demethylase 1-selective inhibitors

27 July 2017

cites work

1 reference

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21 June 2018

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21 June 2018

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Structural basis for the inhibition of the LSD1 histone demethylase by the antidepressant trans-2-phenylcyclopropylamine

21 June 2018

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Structural basis of histone demethylation by LSD1 revealed by suicide inactivation

21 June 2018

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Mechanistic analysis of a suicide inactivator of histone demethylase LSD1

21 June 2018

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Inhibition of lysine-specific demethylase 1 by polyamine analogues results in reexpression of aberrantly silenced genes

21 June 2018

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trans-2-Phenylcyclopropylamine is a mechanism-based inactivator of the histone demethylase LSD1.

21 June 2018

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21 June 2018

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Histone H3 lysine 4 demethylation is a target of nonselective antidepressive medications

21 June 2018

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A mechanism-based inactivator for histone demethylase LSD1.

21 June 2018

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21 June 2018

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Histone demethylation by a family of JmjC domain-containing proteins

21 June 2018

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The diverse functions of histone lysine methylation

21 June 2018

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Histone demethylation mediated by the nuclear amine oxidase homolog LSD1

21 June 2018

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Structure and mechanism of monoamine oxidase

21 June 2018

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Exploring distal regions of the A3 adenosine receptor binding site: sterically constrained N6-(2-phenylethyl)adenosine derivatives as potent ligands.

21 June 2018

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Esters of methanesulfonic acid as irreversible inhibitors of acetylcholinesterase

21 June 2018

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Coordinated histone modifications mediated by a CtBP co-repressor complex

21 June 2018

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A candidate X-linked mental retardation gene is a component of a new family of histone deacetylase-containing complexes

21 June 2018

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Structure-function relationships in flavoenzyme-dependent amine oxidations: a comparison of polyamine oxidase and monoamine oxidase

21 June 2018

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CoREST is an integral component of the CoREST- human histone deacetylase complex

21 June 2018

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Stable histone deacetylase complexes distinguished by the presence of SANT domain proteins CoREST/kiaa0071 and Mta-L1

21 June 2018

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Observation of two different chromophores in the resting state of monoamine oxidase B by fluorescence spectroscopy

21 June 2018

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Pharmacological and clinical implications of MAO-B inhibitors

21 June 2018

1 reference

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Mitochondrial monoamine oxidase. Mechanism of inhibition by phenylhydrazine and by aralkylhydrazines. Role of enzymatic oxidation

21 June 2018

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The monoamine oxidase catalyzed degradation of phenelzine-l-14C, an irreversible inhibitor of monoamine oxidase--I. Studies in vitro.

21 June 2018

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Therapeutic applications and mechanisms of action of monoamine oxidase inhibitor and heterocyclic antidepressant drugs

21 June 2018

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N,N-Dialkylated monophenolic trans-2-phenylcyclopropylamines: novel central 5-hydroxytryptamine receptor agonists

21 June 2018

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Deuterium isotope effect of phenelzine on the inhibition of rat liver mitochondrial monoamine oxidase activity

21 June 2018

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Regulation of histone H3 lysine 56 acetylation in Schizosaccharomyces pombe

21 June 2018

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Human histone demethylase LSD1 reads the histone code

31 October 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2843942

Conformationally restricted analogs of deoxynegamycin

31 October 2018

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https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2843942

Highly potent propargylamine and allylamine inhibitors of bovine plasma amine oxidase

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2843942

The pseudoirreversible inhibition of monoamine oxidase by allylamine

31 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20148560

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

A stable nonfluorescent derivative of resorufin for the fluorometric determination of trace hydrogen peroxide: applications in detecting the activity of phagocyte NADPH oxidase and other oxidases

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20148560

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/JA909996P

1 reference

27 July 2017

1 reference

27 July 2017

1 reference